N-protected/N-substituted alpha-amino aldehydes, which are useful as pharmaceuticals and pharmaceutical intermediates, can be stored and shipped in a more stable form as N-protected/N-substituted-beta-amino hydroxy sulfonates which can be readily converted back into the aldehyde under mild conditions. The present invention relates to N-protected/N-substituted-beta-amino hydroxy sulfonates and their preparation and use.
N-保护/N-取代的α-
氨基醛可以用作药物和药物中间体,并且可以以更稳定的形式作为N-保护/N-取代-β-
氨基羟基
磺酸盐进行储存和运输,在温和条件下可以轻松地转化回
醛类。本发明涉及N-保护/N-取代-β-
氨基羟基
磺酸盐及其制备和使用。