| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 12,13-dihydro-11,13-dioxo-12-phenyl-9H,11H-pyrimido<4,3-c>pyrrolo<1,2-a><1,4>benzodiazepine | 154227-80-2 | C21H15N3O2 |
| —— | (S)-5-(3-Hydroxymethylphenyl)-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092114-34-5 | C18H20N4O2S |
| —— | (2S)-18-nitro-6,14,22-triazapentacyclo[12.8.0.02,6.08,13.016,21]docosa-1(22),8,10,12,16(21),17,19-heptaene-7,15-dione | 1359681-73-4 | C19H14N4O4 |
| —— | (S)-9-ethylamino-5-[1-(pyridin-4-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092111-70-0 | C23H31N7O |
| —— | 1-Methyl-3-morpholin-4-yl-5,10-dihydro-2,4,5,10-tetraaza-dibenzo[a,d]cyclohepten-11-one | 126806-87-9 | C16H17N5O2 |
| —— | 8-amino-3-(carbomethoxy)-1-methyl-5-(3,4,5-trimethoxyphenyl)-1H-pyrimido<4,5-c>-1,2-diazepin-6(7H)-one | 70311-81-8 | C19H21N5O6 |
| —— | (+/-)-pyridine-2-carboxylic acid (4-oxo-2-pyrimidin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-amide | 1175077-84-5 | C18H17N7O2 |
| —— | 10-chloro-6-methyl-2-(1-methyl-4-piperidyl)-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one | 1001346-40-2 | C14H20ClN5O |
| —— | (S)-9-Ethylamino-5-[3-(1,3-oxazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092111-60-8 | C21H22N6O2 |
| —— | (S)-5-(3-Bromophenyl)-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092111-58-4 | C18H20BrN5O |
| —— | (rac)-2-chloro-9-cyclopentyl-7-(2-hydroxy-ethyl)-5-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062245-00-4 | C15H21ClN4O2 |
| —— | 4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid | 1062241-30-8 | C20H23N5O4 |
| —— | 2-chloro-7,7-difluoro-5-methyl-9-phenethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1201693-78-8 | C16H15ClF2N4O |
| —— | 4-(7,7-difluoro-5-methyl-6-oxo-9-phenethyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid | 1201693-29-9 | C24H23F2N5O4 |
| —— | (rac)-4-(9-Cyclopentyl-5,7-diethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid | 1062241-07-9 | C24H31N5O4 |
| —— | 2-chloro-9-cyclopentyl-7,7-dichloro-5-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1201693-91-5 | C13H15Cl3N4O |
| —— | (rac)-2-chloro-9-cyclopropyl-5,7,8-trimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062244-92-1 | C13H17ClN4O |
| —— | (rac)-4-(4-cyclopentyl-9-methyl-10-oxo-1,2,3,3a,4,9,10,10a-octahydro-4,5,7,9-tetraaza-benzo[f]azulen-6-ylamino)-3-methoxy-benzoic acid | 1062245-98-0 | C24H29N5O4 |
| —— | 2-chloro-7,7-difluoro-5-methyl-9-((3R)-3-methylcyclopentyl)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137869-57-8 | C14H17ClF2N4O |
| —— | 4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1137868-34-8 | C23H26FN5O4 |
| —— | (R)-4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-35-5 | C30H41N7O3 |
| —— | 4-(9-cyclopentyl-7-fluoro-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1137868-22-4 | C22H26FN5O4 |
| —— | 4-(7,7-difluoro-5-methyl-9-((3R)-3-methylcyclopentyl)-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1137868-15-5 | C22H25F2N5O4 |
| —— | 2-chloro-9-cyclopentyl-7-fluoro-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137869-64-7 | C14H18ClFN4O |
| —— | 2-chloro-9-cyclohexyl-7-ethyl-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1157849-36-9 | C17H25ClN4O |
| —— | 4-(9-cyclohexyl-7-fluoro-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1137869-72-7 | C23H28FN5O4 |
| —— | 4-(9-cyclopentyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157847-73-8 | C24H31N5O4 |
| —— | (rac)-4-(9-Cyclopentyl-5-methyl-6-oxo-7-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid | 1062241-13-7 | C24H31N5O4 |
| —— | (rac)-6-chloro-4-cyclopentyl-9-methyl-2,3,3a,4,9,10a-hexahydro-1H-4,5,7,9-tetraazabenzo[f]azulen-10-one | 1062245-95-7 | C16H21ClN4O |
| —— | 2-chloro-9-cyclopentyl-7-ethyl-7-fluoro-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137869-79-4 | C15H20ClFN4O |
| —— | (R)-2-chloro-5-methyl-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-b]pyrrolo[1,2-d][1,4]diazepin-6(7H)-one | 1062246-11-0 | C11H13ClN4O |
| —— | 2-chloro-9-cyclopentyl-7-ethyl-7-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1157849-33-6 | C15H21ClN4O |
| —— | 9-butyl-2-chloro-5-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062244-78-3 | C12H17ClN4O |
| —— | (rac)-2-chloro-9-cyclopentyl-7-ethyl-5-ethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062244-09-0 | C16H23ClN4O |
| —— | 2-chloro-9-cyclopentyl-5-methyl-7-(prop-2-ynyl)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1157849-41-6 | C16H19ClN4O |
| —— | (rac)-2-chloro-5-methyl-9-(2,2-dimethyl-cyclopentyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062245-49-1 | C15H21ClN4O |
| —— | (rac)-2-chloro-5-methyl-9-(3-methyl-cyclopentyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062245-37-7 | C14H19ClN4O |
| —— | (rac)-2-chloro-5-methyl-9-(2-methyl-cyclopentyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one | 1062245-29-7 | C14H19ClN4O |
| —— | 10-chloro-2-cyclobutyl-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one | 1001346-15-1 | C12H15ClN4O |
| —— | 4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157848-32-2 | C24H29N5O4 |
| —— | 4-(7-(but-2-ynyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157848-59-3 | C25H29N5O4 |
| —— | 4-(9-cyclopentyl-5-methyl-6-oxo-7-(prop-2-ynyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157848-53-7 | C24H27N5O4 |
| —— | 4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157847-82-9 | C25H33N5O4 |
| —— | 2-chloro-9-cyclohexyl-7-fluoro-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137869-71-6 | C15H20ClFN4O |
| —— | 10-chloro-2-cyclohexyl-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one | 1001345-64-7 | C14H19ClN4O |
| —— | 4-(9-benzyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid | 1062244-36-3 | C23H23N5O4 |
| —— | 4-(9-cyclopentyl-7-ethyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1137868-27-9 | C23H28FN5O4 |
| —— | (rac)-4-(9-Cyclopentyl-7-ethyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid | 1062241-02-4 | C23H29N5O4 |
| —— | 2-chloro-9-cyclohexyl-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1157849-31-4 | C16H23ClN4O |
| —— | 4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157847-54-5 | C24H31N5O4 |