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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 12,13-dihydro-11,13-dioxo-12-phenyl-9H,11H-pyrimido<4,3-c>pyrrolo<1,2-a><1,4>benzodiazepine 154227-80-2 C21H15N3O2
—— (S)-5-(3-Hydroxymethylphenyl)-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-34-5 C18H20N4O2S
—— (2S)-18-nitro-6,14,22-triazapentacyclo[12.8.0.02,6.08,13.016,21]docosa-1(22),8,10,12,16(21),17,19-heptaene-7,15-dione 1359681-73-4 C19H14N4O4
—— (S)-9-ethylamino-5-[1-(pyridin-4-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-70-0 C23H31N7O
—— 1-Methyl-3-morpholin-4-yl-5,10-dihydro-2,4,5,10-tetraaza-dibenzo[a,d]cyclohepten-11-one 126806-87-9 C16H17N5O2
—— 8-amino-3-(carbomethoxy)-1-methyl-5-(3,4,5-trimethoxyphenyl)-1H-pyrimido<4,5-c>-1,2-diazepin-6(7H)-one 70311-81-8 C19H21N5O6
—— (+/-)-pyridine-2-carboxylic acid (4-oxo-2-pyrimidin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-amide 1175077-84-5 C18H17N7O2
—— 10-chloro-6-methyl-2-(1-methyl-4-piperidyl)-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-40-2 C14H20ClN5O
—— (S)-9-Ethylamino-5-[3-(1,3-oxazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-60-8 C21H22N6O2
—— (S)-5-(3-Bromophenyl)-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-58-4 C18H20BrN5O
—— (rac)-2-chloro-9-cyclopentyl-7-(2-hydroxy-ethyl)-5-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-00-4 C15H21ClN4O2
—— 4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062241-30-8 C20H23N5O4
—— 2-chloro-7,7-difluoro-5-methyl-9-phenethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1201693-78-8 C16H15ClF2N4O
—— 4-(7,7-difluoro-5-methyl-6-oxo-9-phenethyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1201693-29-9 C24H23F2N5O4
—— (rac)-4-(9-Cyclopentyl-5,7-diethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062241-07-9 C24H31N5O4
—— 2-chloro-9-cyclopentyl-7,7-dichloro-5-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1201693-91-5 C13H15Cl3N4O
—— (rac)-2-chloro-9-cyclopropyl-5,7,8-trimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-92-1 C13H17ClN4O
—— (rac)-4-(4-cyclopentyl-9-methyl-10-oxo-1,2,3,3a,4,9,10,10a-octahydro-4,5,7,9-tetraaza-benzo[f]azulen-6-ylamino)-3-methoxy-benzoic acid 1062245-98-0 C24H29N5O4
—— 2-chloro-7,7-difluoro-5-methyl-9-((3R)-3-methylcyclopentyl)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1137869-57-8 C14H17ClF2N4O
—— 4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1137868-34-8 C23H26FN5O4
—— (R)-4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-35-5 C30H41N7O3
—— 4-(9-cyclopentyl-7-fluoro-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1137868-22-4 C22H26FN5O4
—— 4-(7,7-difluoro-5-methyl-9-((3R)-3-methylcyclopentyl)-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1137868-15-5 C22H25F2N5O4
—— 2-chloro-9-cyclopentyl-7-fluoro-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1137869-64-7 C14H18ClFN4O
—— 2-chloro-9-cyclohexyl-7-ethyl-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-36-9 C17H25ClN4O
—— 4-(9-cyclohexyl-7-fluoro-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1137869-72-7 C23H28FN5O4
—— 4-(9-cyclopentyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157847-73-8 C24H31N5O4
—— (rac)-4-(9-Cyclopentyl-5-methyl-6-oxo-7-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062241-13-7 C24H31N5O4
—— (rac)-6-chloro-4-cyclopentyl-9-methyl-2,3,3a,4,9,10a-hexahydro-1H-4,5,7,9-tetraazabenzo[f]azulen-10-one 1062245-95-7 C16H21ClN4O
—— 2-chloro-9-cyclopentyl-7-ethyl-7-fluoro-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1137869-79-4 C15H20ClFN4O
—— (R)-2-chloro-5-methyl-7a,8,9,10-tetrahydro-5H-pyrimido[5,4-b]pyrrolo[1,2-d][1,4]diazepin-6(7H)-one 1062246-11-0 C11H13ClN4O
—— 2-chloro-9-cyclopentyl-7-ethyl-7-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-33-6 C15H21ClN4O
—— 9-butyl-2-chloro-5-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-78-3 C12H17ClN4O
—— (rac)-2-chloro-9-cyclopentyl-7-ethyl-5-ethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-09-0 C16H23ClN4O
—— 2-chloro-9-cyclopentyl-5-methyl-7-(prop-2-ynyl)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-41-6 C16H19ClN4O
—— (rac)-2-chloro-5-methyl-9-(2,2-dimethyl-cyclopentyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-49-1 C15H21ClN4O
—— (rac)-2-chloro-5-methyl-9-(3-methyl-cyclopentyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-37-7 C14H19ClN4O
—— (rac)-2-chloro-5-methyl-9-(2-methyl-cyclopentyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-29-7 C14H19ClN4O
—— 10-chloro-2-cyclobutyl-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-15-1 C12H15ClN4O
—— 4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157848-32-2 C24H29N5O4
—— 4-(7-(but-2-ynyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157848-59-3 C25H29N5O4
—— 4-(9-cyclopentyl-5-methyl-6-oxo-7-(prop-2-ynyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157848-53-7 C24H27N5O4
—— 4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157847-82-9 C25H33N5O4
—— 2-chloro-9-cyclohexyl-7-fluoro-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1137869-71-6 C15H20ClFN4O
—— 10-chloro-2-cyclohexyl-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001345-64-7 C14H19ClN4O
—— 4-(9-benzyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062244-36-3 C23H23N5O4
—— 4-(9-cyclopentyl-7-ethyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1137868-27-9 C23H28FN5O4
—— (rac)-4-(9-Cyclopentyl-7-ethyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062241-02-4 C23H29N5O4
—— 2-chloro-9-cyclohexyl-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-31-4 C16H23ClN4O
—— 4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157847-54-5 C24H31N5O4