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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-(piperazin-1-yl)ethyl)benzamide 1157847-25-0 C27H38N8O3
—— 11-chloroacetyl-6-isopropyl-2-phenyl-5,6-dihydropyrimido[4,5-b][1,5]benzodiazepin-5-one 78438-66-1 C22H19ClN4O2
—— 4-(9-isopropyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-05-9 C27H39N7O3
—— 7-(tert-butyldimethylsilyloxy)-2-chloro-9-cyclopentyl-7-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-46-1 C19H31ClN4O2Si
—— 4-chloro-9-methyl-6-phenyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one 1228425-06-6 C14H13ClN4O
—— isopropyl-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoate 1157849-16-5 C24H31N5O4
—— 11-(2-Bromopropionyl)-6-methyl-2-phenyl-5,6-dihydropyrimido[4,5-b][1,5]benzodiazepin-5-one 78438-71-8 C21H17BrN4O2
—— 2-Azamethylindolizidin 22023-52-5 C8H16N2
—— Oktahydro-didethio-desacetyl-aranotin 20484-99-5 C18H26N2O6
—— 4-chloro-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one 1228425-26-0 C8H9ClN4O
—— (S)-4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-41-3 C28H37N7O3
—— (S)-(isoquinolin-8-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-46-8 C20H20N6O
—— 4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethylpiperidin-4-yl)-3-methoxybenzamide 1157847-59-0 C31H45N7O3
—— 2'-Chloro-5'-(2,2-difluoroethyl)-8'-methylspiro[cyclopropane-1,7'-pteridine]-6'-one 1452229-41-2 C11H11ClF2N4O
—— (S)-4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-4-yl)benzamide 1157848-52-6 C29H39N7O3
—— 5-(2-morpholin-4-yl-ethyl)-5,11-dihydro-benzo[<i>e</i>]pyrido[3,2-<i>b</i>][1,4]diazepin-6-one 4929-28-6 C18H20N4O2
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-(2,2-difluoroethoxy)-N-(1-methylpiperidin-4-yl)benzamide 1157847-70-5 C30H41F2N7O3
—— 4-(9’-cyclopentyl-5’-methyl-6’-oxo-5’,6',8’,9’-tetrahydrospiro[cyclopropane-1,7’-pyrimido[4,5-b][1,4]diazepine]-2’-ylamino)-N-((trans)-4-(4-methylpiperazin-1-yl)cyclohexyl)3-methoxybenzamide 1137212-79-3 C34H48N8O3
—— 2-chloro-5-cyclopropylspiro[8H-pteridine-7,3'-oxolane]-6-one 1452229-22-9 C12H13ClN4O2
—— 6,6-bis-(1H-indol-3-yl)-6H-indeno[1,2-b]pyrido[3,2-e]pyrazine 1526911-64-7 C30H19N5
—— 4-(9-cyclohexyl-7-cyclopropyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-08-2 C29H39N7O3
—— 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-piperidin-3-yl)benzamide 1157848-36-6 C30H41N7O3
—— 11-chloroacetyl-2-phenyl-6-n-propyl-5,6-dihydropyrimido[4,5-b][1,5]benzodiazepin-5-one 78438-65-0 C22H19ClN4O2
—— 9-cyclopentyl-2-(2-methoxy-4-(morpholine-4-carbonyl)phenylamino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-10-9 C25H32N6O4
—— 5-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)picolinonitrile 1157849-00-7 C19H21N7O
—— (S)-4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)-benzamide 1157848-21-9 C30H41N7O3
—— 4-(9-cyclopentyl-5-methyl-6-oxo-7-(pent-2-ynyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-64-0 C32H43N7O3
—— 4-((S)-7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-piperidin-3-yl)benzamide 1157848-46-8 C29H39N7O3
—— 4-(9-cyclopentyl-7-(2-fluoroallyl)-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-76-4 C30H40FN7O3
—— (R)-4-(7-allyl-9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-68-4 C31H43N7O3
—— (R)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro [cyclobutane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1157848-27-5 C29H39N7O3
—— 9-cyclopentyl-2-(3-fluoro-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-04-1 C20H24FN5O2
—— 7-methoxy-3-(2-methyl-imidazol-1-yl)-5-phenyl-3<i>H</i>-benzo[<i>e</i>][1,4]diazepin-2-ylamine 73302-47-3 C20H19N5O
—— 4-((S)-7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-1-methylpiperidin-3-yl)benzamide 1157848-43-5 C30H41N7O3
—— N-(1-acetylpiperidin-4-yl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide 1157847-43-2 C30H41N7O4
—— (R)-4-(9-cyclopentyl-5-methyl-6-oxo-7-(prop-2-ynyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-58-2 C30H39N7O3
—— (+/-)-2-methoxy-N-(4-oxo-2-pyrimidin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-nicotinamide 1175078-29-1 C19H19N7O3
—— (R)-4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1157847-56-7 C29H41N7O3
—— (S)-1-tert-butoxycarbonyl-4-(3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl))phenoxypiperidine 1092114-66-3 C28H38N6O4
—— 4-(9-cyclohexyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-09-3 C27H37N7O3
—— 4-(9-cyclopentyl-7-methoxy-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157848-79-7 C23H29N5O5
—— 2-(3-aminophenylamino)-9-cyclopentyl-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-07-4 C19H24N6O
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-(methylsulfonyl)piperidin-4-yl)benzamide 1157847-44-3 C29H41N7O5S
—— 4-(9-cyclopentyl-5-methyl-6-oxo-7-(prop-2-ynyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-54-8 C30H39N7O3
—— 4-(9-cyclopentyl-7-hydroxy-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid 1157848-81-1 C22H27N5O5
—— N-(1-(cyanomethyl)piperidin-4-yl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide 1157849-11-0 C30H40N8O3
—— 4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide 1157848-19-5 C29H40N8O3
—— 4-(4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamido)-N,N-dimethylpiperidine-1-carboxamide 1157849-12-1 C31H44N8O4
—— 6-hexyl-9-methyl-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>b</i>]quinazoline-5,13-dione 71982-01-9 C23H25N3O2
—— (S)-4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1157847-57-8 C29H41N7O3