| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide | 1157847-87-4 | C29H41N7O3 |
| —— | 3-methoxy-4-(5'-methyl-9'-(2-methylcyclopentyl)-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-(1-methylpiperidin-4-yl)benzamide | 1157848-26-4 | C30H41N7O3 |
| —— | 4-(9-cyclobutyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-03-7 | C28H39N7O3 |
| —— | 6-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)nicotinonitrile | 1157848-99-1 | C19H21N7O |
| —— | 6-Isopropyl-11-[(4-methyl-1-piperazinyl)acetyl]-5,6-dihydropyrimido[4,5-b][1,5]benzodiazepin-5-one | 78438-27-4 | C21H26N6O2 |
| —— | (S)-9-cyclopentyl-5,7,7-trimethyl-2-(1-(4-nitrophenyl)ethylamino)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1204831-82-2 | C23H30N6O3 |
| —— | 4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(piperidin-4-yl)benzamide | 1157849-20-1 | C29H39N7O3 |
| —— | (R)-2-(4-(4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamido)piperidin-1-yl)ethyl dihydrogen phosphate | 1137868-47-3 | C30H41FN7O7P |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(2-(dimethylamino)-2-oxoethyl)piperidin-4-yl)-3-methoxybenzamide | 1137868-51-9 | C30H40F2N8O4 |
| —— | (S)-4-(7-(but-2-ynyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-61-7 | C31H41N7O3 |
| —— | (S)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)benzamide | 1157848-14-0 | C29H39N7O3 |
| —— | (R)-4-(7-(but-2-ynyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-62-8 | C31H41N7O3 |
| —— | 4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157848-83-3 | C24H29N5O4 |
| —— | (S)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-85-5 | C30H41N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1157847-53-4 | C23H30N6O3 |
| —— | (S)-4-(9-cyclopentyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide | 1157847-77-2 | C28H39N7O3 |
| —— | 4-(9-cyclohexyl-7-(2-fluoroallyl)-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-77-5 | C31H42FN7O3 |
| —— | 4-(9-cyclopentyl-7-methoxy-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-80-0 | C29H41N7O4 |
| —— | 4-((S)-7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-piperidin-3-yl)benzamide | 1157848-45-7 | C29H39N7O3 |
| —— | 1092793-64-0 | C22H19ClFN7O | |
| —— | 4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-84-4 | C30H41N7O3 |
| —— | 6-(4,4-Dimethyl-2,6-dioxo-cyclohexenyl)-5,6-dihydro-7-hydroxy-pteridin | 6742-16-1 | C14H16N4O3 |
| —— | 4-chloro-6,9-dimethyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one | 1228425-22-6 | C9H11ClN4O |
| —— | 4-(7-(but-2-ynyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-60-6 | C31H41N7O3 |
| —— | (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide | 1157847-49-8 | C28H39N7O3 |
| —— | 4-(7-(cyanomethyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-30-0 | C29H38N8O3 |
| —— | 11-trifluoromethyl-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>b</i>]quinazoline-5,13-dione | 71981-88-9 | C17H10F3N3O2 |
| —— | (S)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylpyrrolidin-3-yl)benzamide | 1157848-18-4 | C28H37N7O3 |
| —— | (S)-4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide | 1137868-46-2 | C28H37FN8O3 |
| —— | 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethylazetidin-3-yl)-3-methoxybenzamide | 1137868-62-2 | C27H35F2N7O3 |
| —— | 9-cyclopentyl-5-methyl-2-(2-(trifluoromethyl)phenylamino)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1157848-96-8 | C20H22F3N5O |
| —— | (S)-4-(9-cyclopentyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide | 1157847-79-4 | C29H42N8O3 |
| —— | (S)-4-(7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157848-40-2 | C24H29N5O4 |
| —— | 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(pyrrolidin-1-yl)benzamide | 946825-69-0 | C27H35N7O3 |
| —— | N-(cyanomethyl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 946825-49-6 | C25H31N7O3 |
| —— | 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylthio)-N-methylbenzoic acid | 946826-00-2 | C22H26N4O3S |
| —— | 1,5,6,7-tetrachloro-3-(2,4-dichlorophenyl)-1,2,4-benzothiadiazine | 89983-57-3 | C13H4Cl6N2S |
| —— | 4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[5,4-b][1,4]diazepine]-2'-ylamino)-N-(1-ethyl-4-piperidyl)-3-methoxy-benzamide | 1001345-35-2 | C31H43N7O3 |
| —— | 4-(9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide | 1157849-27-8 | C27H38N8O3 |
| —— | N-(azepan-4-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1137867-49-2 | C27H35F2N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-(dimethylamino)ethyl)-3-methoxybenzamide | 1001344-49-5 | C27H39N7O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-fluoro-N-(1-isopropylazetidin-3-yl)-5-methoxybenzamide | 1137868-68-8 | C27H34F3N7O3 |
| —— | N-(azepan-4-yl)-4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1157847-65-8 | C30H43N7O3 |
| —— | 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide | 1157847-19-2 | C25H33N7O3 |
| —— | 4-(9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide | 1157849-13-2 | C26H35N7O3 |
| —— | (RS)-9-cyclopentyl-5,7,7-trimethyl-2-(1-(pyridin-4-yl)ethylamino)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1204831-58-2 | C22H30N6O |
| —— | (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpyrrolidin-3-yl)benzamide | 1157847-45-4 | C28H39N7O3 |
| —— | 4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-4-yl)benzamide | 1157847-62-5 | C29H41N7O3 |
| —— | (R)-4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)-benzamide | 1157848-22-0 | C30H41N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N,3-dimethoxybenzamide | 1157847-50-1 | C24H32N6O4 |