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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— (S)-9-ethylamino-5-[1-(2-chloropyridin-4-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-72-2 C23H30ClN7O
—— 5-cyclopropyl-8-methoxy-1-(pyrazine-2-carbonyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one 1307894-44-5 C19H20N4O3
—— 4-(9-butyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062244-79-4 C20H25N5O4
—— 4-(9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062244-28-3 C22H27N5O4
—— 2-(methoxymethyl)-6-(pyridin-2-ylethynyl)-2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one 1312539-08-4 C20H17N3O2
—— 9-((4-fluorophenyl)ethynyl)-2-methyl-3,4-dihydro-1H-pyrazino[2,1-b]quinazolin-6(2H)-one 1312449-84-5 C20H16FN3O
—— (S)-2-ethylamino-6-(2-(methoxymethyl)-3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-41-6 C23H27N7O3
—— (rac)-4-(9-cyclopentyl-5,7,8-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1062244-62-5 C23H29N5O4
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-1-methylpyrrolidin-3-yl)benzamide 946822-87-3 C28H39N7O3
—— (S)-5-[(2-cyanopyridin-5-yl)methyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-53-9 C19H21N7O
—— (S)-5-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)nicotinic acid 1092113-53-5 C17H17N5O3S
—— 3-(Methylsulfanyl)-6-phenyl-4H-[1,2,4]triazino[1,6-c]quinazolin-1(6H)-one 61602-85-5 C17H14N4OS
—— (S)-5-[(5-cyanopyridin-2-yl)methyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-90-3 C18H18N6OS
—— 4-((S)-9-cyclopentyl-6,7,8,9-tetrahydro-5,7-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946822-78-2 C23H30N6O3
—— 10-methyl-9-methylthio-6-(4-methylphenyl)-6,7,10,12-tetrahydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-dione 1072880-11-5 C23H20N4O2S
—— 2-(2-methoxypropan-2-yl)-6-(pyridin-2-ylethynyl)-2,3-dihydropyrrolo[2,1-b]quinazolin-9(1H)-one 1416009-82-9 C22H21N3O2
—— [(2,2'-bipyridine)2Ru(tetrapyrido[3.2-a:2'3'-c:3'',2''-h:2''',3'''-j]phenazine)Os(2,2'-bipyridine)2](4+) 176388-07-1 C64H44N14OsRu
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-isopropylpiperidin-4-yl)-3-methoxybenzamide 946823-29-6 C31H45N7O3
—— 2-methyl-9-(pyridin-2-ylethynyl)-3,4-dihydro-1H-pyrazino[2,1-b]quinazolin-6(2H)-one 1312449-86-7 C19H16N4O
—— (S)-5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-19-0 C20H21N7O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-isopropylazetidin-3-yl)-3-methoxybenzamide 946823-13-8 C29H41N7O3
—— 3-((4-fluorophenyl)ethynyl)-8-propyl-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312450-43-3 C24H23FN2O
—— N-[2-({4-[2-(4-chlorobenzyl)pyrrolidin-1-yl]-6-isopropyl-7-oxo-6,7-dihydro-5H-pyrrolo[3,4-d]pyrimidin-2-yl}amino)ethyl]acetamide 1079654-00-4 C24H31ClN6O2
—— (S)-6-(2-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-6-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-24-4 C20H20N6O2S
—— 2,2-difluoro-11-(pyridin-2-ylethynyl)-2,3,5,6,14,14a-hexahydropyrrolo[1',2':4,5][1,4]diazepino[7,1-b]quinazolin-8(1H)-one 1416011-14-7 C22H18F2N4O*ClH
—— 4-[(2-cyclopentyl-4,4,6-trimethyl-5-oxo-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-10-yl)amino]-N-(1-ethyl-4-piperidyl)-3-methoxy-benzamide 946823-34-3 C30H43N7O3
—— 2-(1-acetylindolin-5-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-41-2 C25H32N6O2
—— 3-[(5-methyl-6-oxo-8-propan-2-yl-7H-pteridin-2-yl)amino]-N-(1-methylpiperidin-4-yl)-5-methylsulfonylbenzamide 1044269-90-0 C24H33N7O4S
—— 4-((R)-9-cyclopentyl-6,7,8,9-tetrahydro-5,8-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 946823-27-4 C28H39N7O3
—— (R)-3-fluoro-pyrrolidine-1-carboxylic acid 2-[4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoylamino]-ethyl ester 946823-00-3 C30H40FN7O5
—— 8-ethyl-3-((4-fluorophenyl)ethynyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312450-42-2 C23H21FN2O
—— 2-chloro-9-cyclopentyl-5-ethyl-7-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1137213-27-4 C15H21ClN4O
—— (S)-6-(3-ethyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-22-0 C21H23N7O2
—— 8-methyl-3-((5-methylthiazol-2-yl)ethynyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312450-37-5 C20H19N3OS
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methylbenzamide 946823-42-3 C23H30N6O2
—— (S)-5-[3-(4-methyl-5-thioxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-22-1 C20H20N6O2S2
—— 5-cyclopropyl-8-fluoro-1-(2-hydroxy-2-(4-methoxyphenyl)ethyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one 1307894-04-7 C22H25FN2O3
—— 4-(9-cyclopentyl-8-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1137206-54-2 C27H37N7O3
—— cyclopropylmethyl (14Z,9E)-66-chloro-5-oxo-11H-7-oxa-4-aza-1(4,1)-imidazola-6(1,3)-benzenacycloundecaphan-9-ene-3-carboxylate 1534386-98-5 C21H22ClN3O4
—— 3-((3-fluorophenyl)ethynyl)-8-(methoxymethyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312450-58-0 C23H21FN2O2
—— 4-(6,7,8,9-tetrahydro-9-(tetrahydro-2H-pyran-4-yl)-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946823-18-3 C24H32N6O4
—— 2-(2-oxoindolin-5-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-06-9 C23H28N6O2
—— 4-(9-cyclopentyl-8-isopropyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1137206-34-8 C29H41N7O3
—— 10-methyl-9-methylthio-6-(4-nitrophenyl)-6,7,10,12-tetrahydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-dione 1072880-06-8 C22H17N5O4S
—— 2-Chloro-9-(2-cyclopropylethyl)-5-methyl-7,8-dihydropyrimido[4,5-b][1,4]diazepin-6-one 1396319-68-8 C13H17ClN4O
—— N-(4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)-N-methylacetamide 946823-50-3 C24H32N6O2
—— (S)-2-ethylamino-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-25-3 C21H23N7O2
—— 3-((3-fluorophenyl)ethynyl)-8-(hydroxymethyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312455-50-7 C22H19FN2O2
—— (S)-9-ethylamino-5-{3-[5-((1S)-1-hydroxyethyl)-1,3,4-oxadiazol-2-yl]phenyl}-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-07-6 C22H25N7O3
—— N-(4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)-2,2,2-trifluoroacetamide 946823-40-1 C23H27F3N6O2