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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 11-butyl-4-chloro-10-(4-methylphenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-48-4 C22H25ClN4O
11-butyl-4-chloro-10-(4-methylphenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-ethyl-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-45-1 C17H23ClN4O
11-butyl-4-chloro-10-ethyl-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-propyl-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-44-0 C18H25ClN4O
11-butyl-4-chloro-10-propyl-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-(2-methoxyphenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-46-2 C22H25ClN4O2
11-butyl-4-chloro-10-(2-methoxyphenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-(4-cyanophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-56-4 C22H22ClN5O
11-butyl-4-chloro-10-(4-cyanophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-(3-nitrophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-58-6 C21H22ClN5O3
11-butyl-4-chloro-10-(3-nitrophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-(4-methoxyphenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-47-3 C22H25ClN4O2
11-butyl-4-chloro-10-(4-methoxyphenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-(4-fluorophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-54-2 C21H22ClFN4O
11-butyl-4-chloro-10-(4-fluorophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 11-butyl-4-chloro-10-(2,4-dichlorophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one 1246291-50-8 C21H21Cl3N4O
11-butyl-4-chloro-10-(2,4-dichlorophenyl)-7,8,10,11-tetrahydro-5H-benzo[e]pyrimido[4,5-b][1,4]diazepin-9(6H)-one
—— 2,8-Dichloro-11H-pyrimido<4,5-b><1,4>-benzodiazepin-6(5H)-on 66427-85-8 C11H6Cl2N4O
2,8-Dichloro-11H-pyrimido<4,5-b><1,4>-benzodiazepin-6(5H)-on
—— 10-chloro-6-methyl-2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-26-4 C13H14ClN5OS
10-chloro-6-methyl-2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one
—— 8-(4-Nitrophenyl)-6-phenyl-3,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-4-one 135039-29-1 C19H15N5O3
8-(4-Nitrophenyl)-6-phenyl-3,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-4-one
—— 2-amino-4-methoxy-5,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-6-one 1403677-09-7 C8H11N5O2
2-amino-4-methoxy-5,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-6-one
—— 6-[(2,4-dimethoxyphenyl)methyl]-7H-quinazolino[3,2-a][1,4]benzodiazepine-5,13-dione 623586-36-7 C25H21N3O4
6-[(2,4-dimethoxyphenyl)methyl]-7H-quinazolino[3,2-a][1,4]benzodiazepine-5,13-dione
—— 5-benzyl-1-chloro-N-(4-chlorophenyl)-6,7-dihydro-5H-pyrimido[4,5-b]pyrrolo[1,2-d][1,4]diazepin-7-amine 1256908-00-5 C23H19Cl2N5
5-benzyl-1-chloro-N-(4-chlorophenyl)-6,7-dihydro-5H-pyrimido[4,5-b]pyrrolo[1,2-d][1,4]diazepin-7-amine
—— 4-chloro-9-methyl-6-p-tolyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one 1228425-49-7 C15H15ClN4O
4-chloro-9-methyl-6-p-tolyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one
—— 4-chloro-6-cyclopentyl-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one 1228425-35-1 C13H17ClN4O
4-chloro-6-cyclopentyl-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one
—— 4-chloro-6-(4-methoxyphenyl)-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one 1228425-47-5 C15H15ClN4O2
4-chloro-6-(4-methoxyphenyl)-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one
—— 6-benzyl-4-chloro-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one 1228425-29-3 C15H15ClN4O
6-benzyl-4-chloro-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one
—— (2S)-7,15-dioxo-6,14,22-triazapentacyclo[12.8.0.02,6.08,13.016,21]docosa-1(22),8,10,12,16(21),17,19-heptaene-18-carbonitrile 1359681-82-5 C20H14N4O2
(2S)-7,15-dioxo-6,14,22-triazapentacyclo[12.8.0.02,6.08,13.016,21]docosa-1(22),8,10,12,16(21),17,19-heptaene-18-carbonitrile
—— 4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1062241-63-7 C20H24N6O3
4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide
—— 4-(9-cyclohexyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1062241-48-8 C27H37N7O3
4-(9-cyclohexyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide
—— 4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-imidazol-1-yl-propyl)-3-methoxy-benzamide 1062241-69-3 C26H32N8O3
4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-imidazol-1-yl-propyl)-3-methoxy-benzamide
—— 4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N,N-dimethyl-benzamide 1062241-66-0 C22H28N6O3
4-(9-cyclobutyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N,N-dimethyl-benzamide
—— 4-(9-cyclohexyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1062241-60-4 C26H34N6O4
4-(9-cyclohexyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide
—— 4-(9-cyclohexyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-propyl-benzamide 1062241-51-3 C24H32N6O3
4-(9-cyclohexyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-propyl-benzamide
—— (S)-5-[3-(5-mercapto-1,3,4-oxadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-76-2 C19H18N6O2S2
(S)-5-[3-(5-mercapto-1,3,4-oxadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one
—— 2-chloro-9-cyclohexyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1001347-58-5 C13H17ClN4O
2-chloro-9-cyclohexyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one
—— (S)-9-methylthio-5-[3-(1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-65-9 C19H18N6O2S
(S)-9-methylthio-5-[3-(1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one
—— (S)-9-methylthio-5-[3-(5-methylthio-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-77-3 C20H20N6O2S2
(S)-9-methylthio-5-[3-(5-methylthio-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one
—— 6-(3-morpholin-4-yl-propyl)-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>b</i>]quinazoline-5,13-dione 65641-88-5 C23H24N4O3
6-(3-morpholin-4-yl-propyl)-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>b</i>]quinazoline-5,13-dione
—— (S)-6-(3-methyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-2-(methylthio)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-58-4 C18H19N7O2S
(S)-6-(3-methyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-2-(methylthio)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(3-methyl-4-oxo-7-tosyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-2-(methylthio)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-55-1 C25H25N7O4S2
(S)-6-(3-methyl-4-oxo-7-tosyl-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-2-(methylthio)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— (S)-6-(3-methyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-2-(methylamino)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410973-51-1 C18H20N8O2
(S)-6-(3-methyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-2-(methylamino)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one
—— 2,6-dimethyl-4-methylthio-2,6,7,9-tetrahydro-8H-pyrazolo[5,4,3-de]pyrimido[4,5-e][1,4]diazepin-8-one 1114784-96-1 C10H12N6OS
2,6-dimethyl-4-methylthio-2,6,7,9-tetrahydro-8H-pyrazolo[5,4,3-de]pyrimido[4,5-e][1,4]diazepin-8-one
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-{3-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-propyl}-3-methoxy-benzamide 1201691-83-9 C30H42F2N8O4
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-{3-[4-(2-hydroxy-ethyl)-piperazin-1-yl]-propyl}-3-methoxy-benzamide
—— N-((S)-1-benzyl-pyrrolidin-3-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-86-2 C32H37F2N7O3
N-((S)-1-benzyl-pyrrolidin-3-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-pyridin-2-yl-ethyl)-benzamide 1201691-98-6 C28H31F2N7O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-pyridin-2-yl-ethyl)-benzamide
—— 4-[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoylamino]-piperidine-1-carboxylic acid tert-butyl ester 1201691-61-3 C31H41F2N7O5
4-[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoylamino]-piperidine-1-carboxylic acid tert-butyl ester
—— (4-(9-cyclopentyl-7,7-difluoro-5-methyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxyphenyl)methanol 1137868-73-5 C21H27F2N5O2
(4-(9-cyclopentyl-7,7-difluoro-5-methyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxyphenyl)methanol
—— 4-{3-[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoylamino]-2-hydroxy-propyl}-piperazine-1-carboxylic acid tert-butyl ester 1201692-01-4 C33H46F2N8O6
4-{3-[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoylamino]-2-hydroxy-propyl}-piperazine-1-carboxylic acid tert-butyl ester
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-[2-(1H-indol-3-yl)-ethyl]-3-methoxy-benzamide 1201691-45-3 C31H33F2N7O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-[2-(1H-indol-3-yl)-ethyl]-3-methoxy-benzamide
—— N-((R)-1-benzyl-pyrrolidin-3-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-87-3 C32H37F2N7O3
N-((R)-1-benzyl-pyrrolidin-3-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide
—— N-[(1S,2R)-(2-carbamoyl-cyclopentyl)]-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-40-8 C27H33F2N7O4
N-[(1S,2R)-(2-carbamoyl-cyclopentyl)]-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-3-methoxy-benzamide 1137867-41-4 C28H37F2N7O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-3-methoxy-benzamide
—— (R)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-oxo-piperidin-4-yl)-benzamide 1201691-76-0 C26H31F2N7O4
(R)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-oxo-piperidin-4-yl)-benzamide
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-isopropylamino-propyl)-3-methoxy-benzamide 1201691-41-9 C27H37F2N7O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-isopropylamino-propyl)-3-methoxy-benzamide
—— (S)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide 1137869-21-6 C28H35F2N7O3
(S)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-[3-(2-methyl-piperidin-1-yl)-propyl]-benzamide 1201691-93-1 C30H41F2N7O3
4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-[3-(2-methyl-piperidin-1-yl)-propyl]-benzamide
—— N-(1-acetyl-piperidin-4-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1137869-18-1 C28H35F2N7O4
N-(1-acetyl-piperidin-4-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide