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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-(cyclopropylmethyl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946823-20-7 C23H30N6O3
—— 2-(1H-indazol-6-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-08-1 C22H27N7O
—— 2-(2-methoxyphenylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-66-1 C22H29N5O2
—— 2,2-difluoro-9-(pyridin-2-ylethynyl)-2,3,5,6,14,14a-hexahydropyrrolo[2',1:3,4][1,4]diazepino[7,1-b]quinazolin-12(1H)-one 1416011-13-6 C22H18F2N4O
—— 8-ethyl-3-(pyridin-2-ylethynyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1416010-93-9 C22H21N3O
—— (S)-3-(2,2-difluoroethyl)-5-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092112-45-2 C22H23F2N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclopropyl-3-methoxybenzamide 946823-57-0 C26H34N6O3
—— 4-((R)-9-cyclopentyl-6,7,8,9-tetrahydro-5,7-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946822-79-3 C23H30N6O3
—— 4-(9-cyclopropyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946822-91-9 C22H28N6O3
—— 9-ethynyl-2-methyl-3,4-dihydro-1H-pyrazino[2,1-b]quinazolin-6(2H)-one 1312454-95-7 C14H13N3O
—— 9-methylthio-6-(4-trifluoromethylphenyl)-6,7,10,12-tetrahydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-dione 1072879-99-2 C22H15F3N4O2S
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclobutane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 946823-26-3 C30H41N7O3
—— 2-(1H-indazol-4-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-43-4 C22H27N7O
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-(azetidin-1-yl)ethyl)-3-methoxybenzamide 946822-99-7 C28H39N7O3
—— 4-(4-benzyloxypyrimidin-2-yl)-3-hydroxy-1-isopropyl-1,5-dihydropyrrol-2-one 500368-34-3 C18H19N3O3
—— 8-hydroxy-3-(pyridin-3-ylethynyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312539-22-2 C20H17N3O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-(1-methyl-1H-imidazo-4-yl)ethyl)benzamide 946822-92-0 C29H38N8O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(cyclopropylmethyl)piperidin-4-yl)-3-methoxybenzamide 946823-21-8 C32H45N7O3
—— 3-methoxy-N-(1-methyl-piperidin-4-yl)-4-[6-oxo-9-(tetrahydro-pyran-4-yl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino]-benzamide 1137206-44-0 C26H35N7O4
—— 3-ethynyl-8-methyl-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one 1312455-39-2 C16H16N2O
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-isopropoxy-N-methylbenzamide 946823-11-6 C26H36N6O3
—— 2-chloro-9-(1-ethyl-propyl)-5-ethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1137213-32-1 C14H21ClN4O
—— 3-[(1-acetyl-2,3-dihydroindol-7-yl)amino]-10-cyclopentyl-9-ethyl-7-methyl-2,4,7,9,10-pentazabicyclo[4.4.0]deca-1,3,5-trien-8-one 1018317-32-2 C23H29N7O2
—— 4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1137868-36-0 C27H34FN7O3
—— 4-(9-cyclopentyl-7-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-methyl-piperidin-4-yl)-benzamide 1137206-33-7 C26H35N7O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)-benzamide 946823-30-9 C33H49N7O3
—— 9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-2-(phenethylamino)-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-17-2 C23H31N5O
—— ethyl 3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)benzoate 1092111-63-1 C21H25N5O3
—— 4-[9-(1-ethyl-propyl)-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino]-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1137206-35-9 C26H37N7O3
—— 1-hydroxymethyl-6-phenyl-8-trifluoromethyl-4<i>H</i>,6<i>H</i>-benzo[<i>b</i>][1,2,4]triazolo[4,3-<i>d</i>][1,4]diazepin-5-one 54705-85-0 C18H13F3N4O2
—— 11-amino-6-(4-nitrophenyl)-6,7-dihydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepin-5(5aH)-one 1101201-44-8 C20H14N6O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(isobutyl)piperidin-4-yl)-3-methoxybenzamide 946823-32-1 C32H47N7O3
—— 9-methylthio-6-(4-methylphenyl)-6,7,10,12-tetrahydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-dione 1072879-97-0 C22H18N4O2S
—— (S)-5-(2,4-difluorobenzyl)-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-48-2 C19H21F2N5O
—— (+/-)-4-Chloro-2-methoxy-N-(4-oxo-2-pyrimidin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-benzamide hydrochloride 1174763-90-6 C20H19ClN6O3*ClH
—— 10-methyl-9-methylthio-6-(4-fluorophenyl)-6,7,10,12-tetrahydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-dione 1072880-09-1 C22H17FN4O2S
—— 4-(9-cyclohexyl-8-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1137206-56-4 C28H39N7O3
—— 9-cyclopentyl-2-(4-((3-hydroxypropyl)(methyl)amino)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1234479-83-4 C24H34N6O3
—— 2-(1H-indazo-7-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-51-4 C22H27N7O
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzoic acid 946822-62-4 C20H23N5O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-propylpiperidin-4-yl)benzamide 946823-31-0 C31H45N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(cyclopropylmethyl)azetidin-3-yl)-3-methoxybenzamide 946823-15-0 C30H41N7O3
—— (S)-9-ethylamino-5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-17-8 C21H23N7O2
—— 8-benzyl-N-(4-fluorobenzyl)-3-hydroxy-4-oxo-4,6,7,8,9,10-hexahydropyrimido[1,2-d][1,4]diazepine-2-carboxamide trifluoroacetate 911493-60-2 C2HF3O2*C23H23FN4O3
—— (S)-5-cyclopentylmethyl-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-47-1 C18H27N5O
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-((S)-3-fluoropyrrolidin-1-yl)ethyl)-3-methoxybenzamide 946822-98-6 C29H40FN7O3
—— methyl 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxyphenylcarbamate 946823-67-2 C24H32N6O4
—— Circumdatin A 223130-52-7 C21H19N3O5
—— 4-((R)-9-cyclopentyl-6,7,8,9-tetrahydro-5,8-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946823-23-0 C23H30N6O3
—— 2-(4-(1H-1,2,4-triazol-1-yl)phenylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-10-5 C23H28N8O