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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2S)-4-(furan-2-yl)butan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H30N4O3
N-[(2S)-4-(furan-2-yl)butan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[2-(3-fluorophenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H27FN4O2
N-[2-(3-fluorophenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-methyl-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C21H28N4O4S
N-[(3S)-1,1-dioxothiolan-3-yl]-N-methyl-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[(4-fluorophenyl)methyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C23H25FN4O2
N-[(4-fluorophenyl)methyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 8-(Azepane-1-carbonyl)-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C22H30N4O2
8-(Azepane-1-carbonyl)-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 11-oxo-N-(2-phenylethyl)-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H28N4O2
11-oxo-N-(2-phenylethyl)-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-methyl-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C22H30N4O4S
N-methyl-N-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-methyl-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C22H30N4O4S
N-methyl-N-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 11-oxo-3-propan-2-yl-N-prop-2-enyl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C19H24N4O2
11-oxo-3-propan-2-yl-N-prop-2-enyl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[2-(4-methoxyphenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H30N4O3
N-[2-(4-methoxyphenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 8-[2,2-Bis(prop-2-enyl)azetidine-1-carbonyl]-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C25H32N4O2
8-[2,2-Bis(prop-2-enyl)azetidine-1-carbonyl]-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 8-(Morpholine-4-carbonyl)-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C20H26N4O3
8-(Morpholine-4-carbonyl)-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— N-[(2R)-4-(furan-2-yl)butan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H30N4O3
N-[(2R)-4-(furan-2-yl)butan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C21H28N4O4S
N-[(3R)-1,1-dioxothiolan-3-yl]-N-methyl-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 11-Oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-9-carboxylic acid —— C16H19N3O3
11-Oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-9-carboxylic acid
—— 3-benzyl-N-(2-methylpropyl)-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H28N4O2
3-benzyl-N-(2-methylpropyl)-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[(2S)-3-methylbutan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C21H30N4O2
N-[(2S)-3-methylbutan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-benzyl-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H30N4O3
3-benzyl-N-[(2S)-1-hydroxy-3-methylbutan-2-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[(2R)-3-methylbutan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C21H30N4O2
N-[(2R)-3-methylbutan-2-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-benzyl-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H30N4O3
3-benzyl-N-[(2R)-1-hydroxy-3-methylbutan-2-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 4-Thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C10H11N3OS
4-Thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-(Pyridin-2-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C16H16N4OS
12-(Pyridin-2-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 3-(Thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C17H17N3OS
3-(Thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[(3,4-Difluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H17F2N3O
3-[(3,4-Difluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[(4-Fluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H18FN3O
3-[(4-Fluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[(2,6-Difluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H17F2N3O
3-[(2,6-Difluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[(2,5-Difluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H17F2N3O
3-[(2,5-Difluorophenyl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-Benzyl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H19N3O
3-Benzyl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-benzyl-11-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H28N4O3
3-benzyl-11-oxo-N-[[(2R)-oxolan-2-yl]methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-Benzyl-9-fluoro-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H18FN3O
3-Benzyl-9-fluoro-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-benzyl-N-(2-hydroxyethyl)-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C22H24N4O3
3-benzyl-N-(2-hydroxyethyl)-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-Benzyl-8-(thiomorpholine-4-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C24H26N4O2S
3-Benzyl-8-(thiomorpholine-4-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-benzyl-N-[(3R)-oxan-3-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H28N4O3
3-benzyl-N-[(3R)-oxan-3-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-Benzyl-8-(morpholine-4-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C24H26N4O3
3-Benzyl-8-(morpholine-4-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-benzyl-N-[(3S)-oxan-3-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H28N4O3
3-benzyl-N-[(3S)-oxan-3-yl]-11-oxo-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 12-[(2-Chlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H16ClN3OS
12-[(2-Chlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[[2-(Trifluoromethyl)phenyl]methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C18H16F3N3OS
12-[[2-(Trifluoromethyl)phenyl]methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 9-Fluoro-3-(thiophen-3-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C17H16FN3OS
9-Fluoro-3-(thiophen-3-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 12-(Thiophen-2-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C15H15N3OS2
12-(Thiophen-2-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 9-Fluoro-3-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C17H16FN3OS
9-Fluoro-3-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 12-(Pyridin-3-ylmethyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C16H16N4OS
12-(Pyridin-3-ylmethyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(3,4-Dichlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15Cl2N3OS
12-[(3,4-Dichlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,4-Difluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15F2N3OS
12-[(2,4-Difluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,4-Dichlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15Cl2N3OS
12-[(2,4-Dichlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,5-Difluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15F2N3OS
12-[(2,5-Difluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2-Chloro-6-fluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15ClFN3OS
12-[(2-Chloro-6-fluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,6-Dichlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15Cl2N3OS
12-[(2,6-Dichlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,3-Difluorophenyl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C17H15F2N3OS
12-[(2,3-Difluorophenyl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(4-Chloro-3-fluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15ClFN3OS
12-[(4-Chloro-3-fluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,3-Difluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H15F2N3OS
12-[(2,3-Difluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one