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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-dimethylamino-ethyl)-3-trifluoromethyl-benzamide 1201692-75-2 C25H30F5N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2,5-difluoro-N-methyl-benzamide 1201693-03-9 C21H22F4N6O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-3-fluoro-benzamide 1201692-89-8 C27H34F3N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-dimethylamino-propyl)-3-trifluoromethyl-benzamide 1201692-76-3 C26H32F5N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-3-methyl-benzamide 1201692-57-0 C28H37F2N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-dimethylamino-ethyl)-3-methyl-benzamide 1201692-59-2 C25H33F2N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methyl-benzamide 1201692-64-9 C21H24F2N6O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2,5-difluoro-N-piperidin-4-yl-benzamide 1201693-05-1 C25H29F4N7O2
—— 4-[[7,7-difluoro-5-methyl-6-oxo-9-(2-phenylethyl)-8H-pyrimido[4,5-b][1,4]diazepin-2-yl]amino]-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1201693-30-2 C30H35F2N7O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-fluoro-N-methyl-benzamide 1201692-93-4 C21H23F3N6O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-dimethylamino-propyl)-2,5-difluoro-benzamide 1201693-02-8 C25H31F4N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-2,3-difluoro-benzamide 1201693-09-5 C27H33F4N7O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethyl-N-methyl-benzamide 1201692-69-4 C23H28F2N6O2
—— 10-chloro-6-methyl-2-(oxan-4-yl)-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001345-65-8 C13H17ClN4O2
—— (+/-)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclobutane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide 1137209-65-4 C31H41N7O3
—— 9-benzyl-2-chloro-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-34-1 C14H13ClN4O
—— 2-(methylthio)-6,11-dihydro-5H-benzo[b]pyrimido[4,5-e][1,4]diazepin-5-one 1313713-95-9 C12H10N4OS
—— (R)-2'-chloro-9'-(3,3-difluorocyclopentyl)-5'-methyl-8',9'-dihydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepin]-6'(5'H)-one 1117936-75-0 C15H17ClF2N4O
—— (R)-2-chloro-9-(3,3-difluorocyclopentyl)-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1117936-71-6 C15H19ClF2N4O
—— (R)-N-cyclopropyl-4-(9'-(3,3-difluorocyclopentyl)-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxybenzamide 1117936-49-8 C26H30F2N6O3
—— 4-amino-2-(butylamino)-9-(3-(pyrrolidin-1-ylmethyl)benzyl)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1228586-17-1 C23H33N7O
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2,3-difluoro-benzoic acid 1253115-61-5 C20H19F4N5O3
—— 8-methoxy-3-methylsulfanyl-5,10-dihydro-2,4,5,10-tetraazadibenzo[a,d]-cyclohepten-11-one 942910-88-5 C13H12N4O2S
—— (S)-5-[3-(4-cyano-1,3-oxazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-53-8 C21H18N6O2S
—— (S)-9-methylthio-5-[3-(5-trifluoromethyl-1,2,4-oxadiazol-3-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1234694-01-9 C20H17F3N6O2S
—— (S)-9-methylthio-5-[3-(2H-tetrazol-5-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-56-1 C18H18N8OS
—— (S)-5-[3-(1-methyl-1H-tetrazol-5-yl)phenyl]-9-methylthio-1,2,3,3a.4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-58-3 C19H20N8OS
—— (S)-5-[3-(1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-90-0 C19H18N6O2S
—— (S)-5-[3-(2-methyl-2H-tetrazol-5-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-57-2 C19H20N8OS
—— (R)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide 1137212-41-9 C30H39N7O3
—— (+/-)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide 1137209-31-4 C30H41N7O3
—— (S)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide 1137212-43-1 C30H39N7O3
—— (+/-)-9-(4-Chloro-2-methoxy-benzoylamino)-4-oxo-2-pyrimidin-4-yl-5,6,8,9-tetrahydro-4H-1,4a,7-triaza-benzocycloheptene-7-carboxylic acid ethyl ester 1174763-40-6 C23H23ClN6O5
—— 2-hydroxycircumdatin C 1184940-80-4 C17H13N3O4
—— mono<2,3,9,9a-tetrahydro-2-(2-methylpropyl)-3-oxo-9-<(5,6,7,13-tetrahydro-5,13-dioxoquinazolino<3,2-a><1,4>benzodiazepin-7-yl)methyl>1H-imidazo<1,2-a>indol-9-yl>butanedioic acid ester 102996-22-5 C35H33N5O7
—— 1-[4-(2,4-diamino-8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepin-6-yl)phenyl]-3-phenylurea 1029135-19-0 C20H20N8O
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-piperazin-1-yl-ethyl)-benzamide 1201691-44-2 C27H36F2N8O3
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-piperidin-4-yl-benzamide 1201691-17-9 C24H29F2N7O2
—— N-(2-amino-ethyl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-43-1 C23H29F2N7O3
—— N-(3-amino-propyl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-63-5 C24H31F2N7O3
—— 6-Methylsulfanyl-10-phenyl-2,5,7,9-tetrazatetracyclo[9.7.0.03,8.013,18]octadeca-1(11),3(8),6,13,15,17-hexaene-4,12-dione 1072879-96-9 C21H16N4O2S
—— 11-acetyl-10-(2,4-dichloro-phenyl)-4-hydroxy-7,7-dimethyl-5,6,7,8,10,11-hexahydro-1,3,5,11-tetraaza-dibenzo[a,d]cyclohepten-9-one 1047618-82-5 C21H20Cl2N4O3
—— 11-acetyl-10-(2,4-dichloro-phenyl)-7,7-dimethyl-5,6,7,8,10,11-hexahydro-1,3,5,11-tetraaza-dibenzo[a,d]cyclohepten-9-one 1047618-85-8 C21H20Cl2N4O2
—— 2H-[1,4]diazepino[2,1-b]quinazoline-3,7(1H,4H,5H)-dione 173915-18-9 C12H11N3O2
—— (+/-)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(quinuclidin-3-yl)benzamide 1137209-12-1 C30H39N7O3
—— 4-[(2S,9S,9aS)-9-((S)-5,13-Dioxo-5,6,7,13-tetrahydro-6,8,13a-triaza-benzo[3,4]cyclohepta[1,2-b]naphthalen-7-ylmethyl)-9-hydroxy-2-isobutyl-3-oxo-2,3,9,9a-tetrahydro-imidazo[1,2-a]indol-1-yl]-4-oxo-butyric acid 102996-15-6 C35H33N5O7
—— (S)-7-((2S,9S,9aS)-1-Acetyl-9-hydroxy-2-isobutyl-3-oxo-2,3,9,9a-tetrahydro-1H-imidazo[1,2-a]indol-9-ylmethyl)-6,7-dihydro-6,8,13a-triaza-benzo[3,4]cyclohepta[1,2-b]naphthalene-5,13-dione 102743-49-7 C33H31N5O5
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-05-5 C20H22F2N6O3
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-piperidin-4-yl-benzamide 1201691-08-8 C25H31F2N7O3
—— 8-(1,3-benzodioxol-5-yl)-6-(4-chlorophenyl)-8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepine-2,4-diamine 1402415-29-5 C20H17ClN6O2