| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | (rac)-4-(9-cyclohexyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid methyl ester | 1062245-69-5 | C24H31N5O4 |
| —— | 6,11-dihydro-6-methyl-5H-pyrimido[4,5-b][1,5]benzodiazepin-5-one | 78438-72-9 | C12H10N4O |
| —— | N-(1-(azetidine-3-carbonyl)piperidin-4-yl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1157849-21-2 | C32H44N8O4 |
| —— | 9-allyl-2-chloro-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 946826-41-1 | C13H17ClN4O |
| —— | (S)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(tetrahydrofuran-3-yl)benzamide | 946824-50-6 | C27H34N6O4 |
| —— | 1416011-92-1 | C20H17N3O2 | |
| —— | (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((1-methylpyrrolidin-3-yl)methyl)benzamide | 1157849-23-4 | C29H41N7O3 |
| —— | 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-2H-pyran-4-yl)benzamide | 1157847-16-9 | C26H34N6O4 |
| —— | (S)-3-(2-fluoroethyl)-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one | 1092112-44-1 | C21H22FN7O3 |
| —— | 1044271-83-1 | C21H27N5O3S | |
| —— | 5-cyclopropyl-8-fluoro-1-(pyrazine-2-carbonyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one | 1307894-72-9 | C18H17FN4O2 |
| —— | 5-[3-(2-chloropyridin-4-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092113-45-5 | C22H20ClN5OS |
| —— | (S)-N-(2-fluoroethyl)-2-{5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-2-oxo-1,3,4-oxadiazol-3(2H)-yl}acetamide | 1092567-01-5 | C23H24FN7O4S |
| —— | 4-[(9-cyclopentyl-5,8-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-N-methylbenzamide | 1157846-87-1 | C23H30N6O3 |
| —— | (S)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-ylmethyl)benzamide | 1157847-30-7 | C27H37N7O3 |
| —— | auranthic acid ethyl ester | 1233669-28-7 | C20H17N3O4 |
| —— | 4-(9-((R)-3,3-difluorocyclopentyl)-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b] [1,4]diazepin-2-ylamino)-N-((1R,3R)-3-fluorocyclopentyl)-3-methoxybenzamide | 1117936-47-6 | C28H35F3N6O3 |
| —— | 1433992-36-9 | C23H17F4N5O3S | |
| —— | 4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-01-5 | C31H45N7O3 |
| —— | 4-chloro-5-phenyl-11H-pyrimido<4,5-b><1,5>benzodiazepine | 134031-30-4 | C17H11ClN4 |
| —— | (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-phenylethyl)benzamide | 946825-39-4 | C31H38N6O3 |
| —— | (+/-)-N-(7-benzyl-4-oxo-2-pyrimidin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-2-methoxy-nicotinamide hydrochloride | 1175078-15-5 | C26H25N7O3*ClH |
| —— | 1233669-24-3 | C22H19N3O5 | |
| —— | 1-Morpholinoacetyl-2-carboxy-4-<pyridyl-(4)-methylamino>-1,2,3,4-tetrahydro-5H-1,4-benzodiazepin-5-on | 19050-59-0 | C22H25N5O5 |
| —— | 4-carboxy-2-(4-chloro-2-fluoro-3-methoxyphenyl)-6,7-dimethyl-5,6,7,8-tetrahydropteridine | 1292287-88-7 | C16H16ClFN4O3 |
| —— | (S)-3-(2-fluoroethyl)-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one | 1092114-07-2 | C21H21FN6O3S |
| —— | N-(2-aminoethyl)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1157847-17-0 | C23H31N7O3 |
| —— | 2-chloro-9-cyclobutyl-7,7-difluoro-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1201693-60-8 | C12H13ClF2N4O |
| —— | N-(1-acetyl-piperidin-4-yl)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide | 1137209-53-0 | C28H37N7O4 |
| —— | 4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide | 1157847-89-6 | C30H44N8O3 |
| —— | 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-methanesulfonyl-piperidin-4-yl)-3-methoxy-benzamide | 1137209-51-8 | C27H37N7O5S |
| —— | (rac)-2-chloro-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-methyl-piperidin-4-yl)-benzamide | 1062243-06-4 | C27H36ClN7O2 |
| —— | 8-chloro-5-cyclopropyl-1-(pyrazine-2-carbonyl)-2,3,5,6-tetrahydrobenzo[b][1,5]diazocin-4(1H)-one | 1307894-75-2 | C18H17ClN4O2 |
| —— | (S)-5-[3-(7-chloro-9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one | 1092113-02-4 | C21H22ClN7O3 |
| —— | (rac)-3-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-pyridin-4-yl-benzamide | 1062243-25-7 | C26H29N7O2 |
| —— | 7-(4-chloro-7-(4-methoxybenzyl)-6,7-dihydro-5H-pyrrolo[2,3-d]pyrimidin-2-ylamino)-1-ethyl-6-methoxy-4,5-dihydro-1H-benzo[b]azepin-2(3H)-one | 1312163-68-0 | C27H30ClN5O3 |
| —— | 1233669-22-1 | C19H14ClN3O2 | |
| —— | (rac)-4-(9-cyclohexyl-7-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide | 1062241-18-2 | C28H39N7O3 |
| —— | (S)-9-ethylamino-5-[(pyridin-4-yl)methyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092113-17-1 | C18H22N6O |
| —— | 8-chloro-6-cyclohexylidene-1,2,6,7-tetrahydro-7,9,11,11b-tetraaza-dibenzo[c,d,h]azulene | 889654-92-6 | C18H19ClN4 |
| —— | 4-(9-cyclopentyl-5-methyl-6-oxo-7-(prop-2-ynyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-piperidin-3-yl)benzamide | 1157848-55-9 | C29H37N7O3 |
| —— | (S)-3-(2,2-difluoroethyl)-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one | 1092114-08-3 | C21H20F2N6O3S |
| —— | 6-(4-methylphenyl)-8-phenyl-1,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-4-one | 135039-31-5 | C20H18N4O |
| —— | 3-[(1S,2S)-2-hydroxycyclohexyl]-10-methyl-6-{[2-(trifluoromethyl)pyridin-4-yl]methyl}-9,10-dihydropyrido[3,2-h]quinazolin-4(3H)-one | 1413974-68-1 | C25H25F3N4O2 |
| —— | methyl (S)-2-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3-oxazole-4-carboxylate | 1092112-68-9 | C23H24N6O4 |
| —— | (rac)-3-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-4-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide | 1062242-79-8 | C27H36N6O4 |
| —— | (+/-)-6-fluoro-4H-benzo[1,3]dioxine-8-carboxylic acid (7-benzyl-4-oxo-2-pyridin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-amide hydrochloride | 1175078-18-8 | C29H26FN5O4*ClH |
| —— | 2-(benzylamino)-8,9-dihydro-3-methyl-6-(4-nitrophenyl)-3Hpyrimido[4,5-b][1,4]diazepin-4(7H)-one | 1607450-27-0 | C21H20N6O3 |
| —— | 1-(Morpholinoacetyl)-2-carboxy-4-<pyridyl-(3)-methylamino>-1,2,3,4-tetrahydro-5H-1,4-benzodiazepin-5-on | 19050-58-9 | C22H25N5O5 |
| —— | (S)-5-[3-(4-methyl-5-thioxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092112-58-7 | C20H21N7O2S |