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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— (S)-6-(3-(2-fluoroethyl)-2-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410972-32-5 C22H24FN7O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-morpholinoethyl)benzamide 946822-94-2 C29H41N7O4
—— 4-[4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoylamino]-piperidine-1-carboxylic acid tert-butyl ester 946823-59-2 C33H47N7O5
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-dimethylamino-ethyl)-3-methoxy-benzamide 1201691-11-3 C24H31F2N7O3
—— 7-chloro-2-(trifluoromethyl)-6,11-dihydro-5H-benzo[b]pyrido[2,3-e][1,4]diazepin-5-one 1039715-36-0 C13H7ClF3N3O
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methyl-benzoic acid 1062245-22-0 C23H29N5O3
—— 2-(2-methyl-2H-indazol-7-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-54-7 C23H29N7O
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1201691-10-2 C25H30F2N6O4
—— 9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-2-(phenylamino)-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-53-6 C21H27N5O
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-3-methoxy-benzamide 1137867-71-0 C29H39F2N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946822-77-1 C24H32N6O3
—— 4-(-9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(2-fluoroethyl)piperidin-4-yl)-3-methoxybenzamide 946823-39-8 C30H42FN7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-tert-butylpiperidin-4-yl)-3-methoxybenzamide 946823-33-2 C32H47N7O3
—— 12-methoxy-5b,6,7,8-tetrahydrobenzo[6,7]pyrrolo[2',1':3,4][1,4]diazepino[2,1-b]quinazoline-10,16-dione 1239969-54-0 C20H17N3O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxyphenyl-(4-tert-butoxycarbonylpiperazin-1-yl)methanone 946822-67-9 C30H41N7O5
—— (S)-2-{5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-2-oxo-1,3,4-oxadiazol-3(2H)-yl}methyl acetate 1092114-12-9 C22H22N6O5S
—— 9-cyclopentyl-2-[4-((S)-3-fluoro-pyrrolidine-1-carbonyl)-2-methoxyphenylamino]-5,7,7-trimethyl-5,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-6-one 946822-93-1 C27H35FN6O3
—— methyl 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoate 1282611-90-8 C24H31N5O4
—— 101389-64-4 C25H18N4O2
—— 4-[(9-cyclopentyl-6,7,8,9-tetrahydro-5-methyl-6-oxospiro[5H-pyrimido[4,5-b][1,4]diazepine-7,1'-cyclopropan]-2-yl)amino]-N-(tetrahydropyran-4-yl)benzamide 1062242-46-9 C27H34N6O3
—— (S)-9-ethylamino-5-(3-methoxyphenyl)-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-57-3 C19H23N5O2
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methyl-benzamide 1201693-14-2 C22H26F2N6O2
—— 4-(9-cyclopentyl-5-ethyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl-amino)-N-(3-dimethyl-amino-propyl)-benzamide 1201692-23-0 C26H35F2N7O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((S)-1-isopropylpyrrolidin-3-yl)-3-methoxybenzamide 946823-35-4 C30H43N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethoxy-N-(1-methylpiperidin-4-yl)benzamide 946823-36-5 C30H43N7O3
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzamide 1201691-15-7 C19H20F2N6O2
—— (+/-)-6-fluoro-4H-benzo[1,3]dioxine-8-carboxylic acid (7-isopropyl-4-oxo-2-pyridin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-amide hydrochloride 1175078-17-7 C25H26FN5O4*ClH
—— 4-[(9-cyclopentyl-6,7,8,9-tetrahydro-5-methyl-6-oxospiro[5H-pyrimido[4,5-b][1,4]diazepine-7,1'-cyclopropan]-2-yl)amino]-benzoic acid 1062245-53-7 C22H25N5O3
—— 4-(9-cyclobutyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-dimethylamino-propyl)-benzamide 1201691-23-7 C24H31F2N7O2
—— 4-benzyl-1,4-diazepano<2,1-b>quinazolin-11(11aH)-one 126411-74-3 C19H19N3O
—— (S)-6-(3-ethyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-11-9 C21H22N6O2S
—— 4-[(2-cyclopentyl-4,4,6-trimethyl-5-oxo-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-10-yl)amino]-3-methoxy-N-(2-pyrrolidin-1-ylethyl)benzamide 946822-95-3 C29H41N7O3
—— (rac)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-methyl-piperidin-4-yl)-benzamide 1062240-90-7 C27H37N7O2
—— 1,3-Dimethyl-11H-pyrimido<4,5-b><1,4>benzodiazepin-2,4,6-(1H,3H,5H)-trion 18830-60-9 C13H12N4O3
—— 6-(4-nitrophenyl)-8-phenyl-1,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-4-one 135039-35-9 C19H15N5O3
—— 9-methoxy-10-methyl-6-(4-chlorophenyl)-6,7,10,12-tetrahydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepine-5,11-dione 1072880-15-9 C22H17ClN4O3
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzamide 1201693-13-1 C21H24F2N6O2
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzoic acid 1201693-12-0 C21H23F2N5O3
—— 911494-10-5 C16H24N4O6
—— (S)-6-(6-aminopyridin-2-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-21-1 C16H18N6OS
—— (rac)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-yl amino)-3-methoxy-benzoic acid 946822-70-4 C22H27N5O4
—— N-(8-benzyl-2-{[(4-fluorobenzyl)amino]carbonyl}-3-hydroxy-4-oxo-4,6,7,8,9,10-hexahydropyrimido[1,2-d][1,4]diazepin-10-yl)-N,N',N'-trimethylethanediamide trifluoroacetate 911492-58-5 C2HF3O2*C28H31FN6O5
—— N-(4-fluorobenzyl)-3-hydroxy-8-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrazino[1,2-a]pyrimidine-2-carboxamide trifluoroacetate 911492-41-6 C2HF3O2*C16H17FN4O3
—— (S)-7-chloro-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-37-5 C11H13ClN4OS
—— (rac)-2-chloro-9-cyclopentyl-7-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062243-94-0 C13H17ClN4O
—— 5'-methyl-3'-(phenylmethyl)spiro[cyclopentane-1,7'(8'H)-[3H]imidazo[2,1-b]purin]-4(5'H)-one 140378-61-6 C19H21N5O
—— 2-chloro-9-cyclobutyl-7,7-difluoro-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1201693-59-5 C11H11ClF2N4O
—— (S)-3-(5,13-dioxo-5,6,7,13-tetrahydro-6,8,13a-triazabenzo[3,4]cyclohepta[1,2-b]naphthalen-7-yl)-N-methylpropanamide 1620751-50-9 C20H18N4O3
—— (S)-7-[3-oxo-3-(pyrrolidin-1-yl)propyl]-6,7-dihydro-6,8,13atriazabenzo[3,4]cyclohepta[1,2-b]naphthalene-5,13-dione 1620751-53-2 C23H22N4O3
—— 4-[(9-cyclopentyl-6,7,8,9-tetrahydro-5-methyl-6-oxospiro[5H-pyrimido[4,5-b][1,4]diazepine-7,1'-cyclopropan]-2-yl)amino]-N-(1-methyl-4-piperidinyl)benzamide 1062242-43-6 C28H37N7O2