| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | (S)-4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-3-yl)benzamide | 1157847-61-4 | C28H39N7O3 |
| —— | 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-2-ylmethyl)benzamide | 1157847-33-0 | C27H31N7O3 |
| —— | (R)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-86-6 | C30H41N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-(difluoromethoxy)benzoic acid | 1157847-71-6 | C23H27F2N5O4 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-fluoroethyl)-3-methoxybenzamide | 946825-91-8 | C25H33FN6O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((1R,2R)-2-hydroxycyclohexyl)-3-methoxybenzamide | 946825-84-9 | C29H40N6O4 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(4-(dimethylamino)cyclohexyl)-3-methoxybenzamide | 1137869-12-5 | C29H39F2N7O3 |
| —— | (S)-9-methylamino-5-(2-methylisoindoline-1,3-dion-5-yl)-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one | 1092112-87-2 | C20H20N6O3 |
| —— | (R)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxypropyl)-3-methoxybenzamide | 1137869-06-7 | C24H30F2N6O4 |
| —— | 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-pyrrolidin-3-yl)benzamide | 1157848-39-9 | C29H39N7O3 |
| —— | methyl (3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)carbamate | 946824-19-7 | C23H30N6O3 |
| —— | 2-(benzylamino)-8,9-dihydro-3-methyl-6-phenyl-3H-pyrimido[4,5-b][1,4]diazepin-4(7H)-one | 1607450-30-5 | C21H21N5O |
| —— | 4-(9-((R)-1-(cyclopropylmethyl)pyrrolidin-3-yl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide | 946823-28-5 | C27H37N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-methylpiperidin-4-yl)-3-propoxybenzamide | 1157847-68-1 | C31H45N7O3 |
| —— | N-(azetidin-3-yl)-4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1157847-64-7 | C27H37N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(4-(2-hydroxyethyl)piperazin-1-yl)-3-methoxybenzamide | 1157847-52-3 | C29H42N8O4 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-methyl-N-(1-methylpiperidin-4-yl)benzamide | 1137868-80-4 | C27H35F2N7O2 |
| —— | (S)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide | 1157848-17-3 | C28H37N7O3 |
| —— | 4-(9-cyclobutyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide | 1157848-04-8 | C26H35N7O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethylazetidin-3-yl)-2-fluoro-5-methoxybenzamide | 1137868-67-7 | C26H32F3N7O3 |
| —— | N-(3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)-3,3,3-trifluoropropanamide | 946824-09-5 | C24H29F3N6O2 |
| —— | N-cyclopentyl-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxybenzamide | 946824-44-8 | C28H36N6O3 |
| —— | 9-cyclopentyl-2-(2-methoxy-4-(morpholine-4-carbonyl)phenylamino)-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 946824-89-1 | C27H36N6O4 |
| —— | (R)-N-cyclobutyl-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 946824-65-3 | C26H34N6O3 |
| —— | 4-(7-allyl-9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-66-2 | C31H43N7O3 |
| —— | (R)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide | 1137867-42-5 | C26H33F2N7O3 |
| —— | 1,3-Dimethyl-5,8-dibenzyl-5,6,7,8-tetrahydro-lumazin | 31595-79-6 | C22H24N4O2 |
| —— | 4-(7-(2-amino-2-oxoethyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-31-1 | C29H40N8O4 |
| —— | 11-bromo-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>a</i>]quinazoline-5,13-dione | 72004-69-4 | C16H10BrN3O2 |
| —— | 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-(3-hydroxypropyl)-3-methoxybenzamide | 946825-78-1 | C26H34N6O4 |
| —— | (rac)-4-(9-cyclohexyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide | 1062241-21-7 | C29H41N7O3 |
| —— | 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-methylbenzamide | 946823-24-1 | C24H30N6O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(((1S,2R)-2-hydroxycyclohexyl)methyl)-3-methoxybenzamide | 946825-45-2 | C30H42N6O4 |
| —— | (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)benzamide | 1157847-46-5 | C29H41N7O3 |
| —— | 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N',N'-dimethylbenzohydrazide | 1137867-94-7 | C24H31F2N7O3 |
| —— | 7,8,9,10-tetrahydro-10-benzyloxy-9-heptyl-[1,4]diazepino[1,2,3-g,h]purine | 608523-33-7 | C22H29N5O |
| —— | (S)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide | 1157849-15-4 | C28H37N7O3 |
| —— | 4-(7-(cyanomethyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzoic acid | 1157848-29-7 | C23H26N6O4 |
| —— | 4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157847-86-3 | C31H45N7O3 |
| —— | (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)benzamide | 1157847-47-6 | C29H41N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrazin-2-yl)benzamide | 946825-35-0 | C27H32N8O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-fluoro-N-(1-(2-hydroxyethyl)piperidin-4-yl)-5-methoxybenzamide | 1137868-53-1 | C28H36F3N7O4 |
| —— | 2-nitro-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>a</i>]quinazoline-5,13-dione | 71981-89-0 | C16H10N4O4 |
| —— | 11-chloro-5,13-dioxo-7,13-dihydro-5<i>H</i>-benzo[6,7][1,4]diazepino[2,1-<i>a</i>]quinazoline-6-carboxylic acid ethyl ester | 71981-94-7 | C19H14ClN3O4 |
| —— | 3-((3-fluorophenyl)ethynyl)-8-methoxy-6,7,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one | 1312450-49-9 | C22H19FN2O2 |
| —— | N-(3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-4-methylphenyl)acetamide | 946824-27-7 | C24H32N6O2 |
| —— | N-(1-(2-amino-2-oxoethyl)piperidin-4-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 1137868-50-8 | C28H36F2N8O4 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1137868-81-5 | C27H35F2N7O3 |
| —— | (S)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxypropyl)-3-methoxybenzamide | 1137869-05-6 | C24H30F2N6O4 |
| —— | 8-fluoro-3-(pyridin-2-ylethynyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one | 1312457-52-5 | C20H16FN3O |