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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxypropyl)-3-methoxybenzamide 946825-87-2 C26H36N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(thiazol-2-yl)benzamide 946825-33-8 C26H31N7O3S
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-propylbenzamide 946825-24-7 C26H36N6O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxyethyl)-3-methoxybenzamide 946825-80-5 C25H34N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-2-ylmethyl)benzamide 946825-71-4 C29H35N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclobutyl-3-methoxybenzamide 946823-58-1 C27H36N6O3
—— 4-(6,7,8,9-tetrahydro-9-((S)-tetrahydrofuran-3-yl)-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946824-52-8 C23H30N6O4
—— 2-amino-4-methoxy-6-(2-fluorophenyl)-11H-pyrimido[4,5-b][1,4]benzodiazepine 1096145-02-6 C18H14FN5O
—— 4-((S)-9-cyclopentyl-6,7,8,9-tetrahydro-5,7-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-2H-pyran-4-yl)-3-methoxybenzamide 946824-40-4 C27H36N6O4
—— spiro[indeno[1',2':5,6]pyrido[2,3-d]pyrimidine-5,3'-indoline]-2,2',4,10(1H,3H,11H)-tetraone 1422371-99-0 C21H12N4O4
—— 3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclopropylbenzamide 946824-23-3 C25H32N6O2
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(pyridin-3-ylmethyl)benzamide 946825-65-6 C29H33N7O3
—— 5-ethoxy-2-hydroxy-4-methyl-11H-pyrimido<4,5-b><1,5>benzodiazepine 131563-02-5 C14H14N4O2
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-(1-hydroxy-2-methylpropan-2-yl)-3-methoxybenzamide 946825-88-3 C27H36N6O4
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-((1R,2R)-2-hydroxycyclopentyl)-3-methoxybenzamide 946825-89-4 C28H36N6O4
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-cyclopropyl-3-methoxybenzamide 946824-48-2 C26H32N6O3
—— 4-(9-(2,2,3,3,3-pentafluoropropyl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946824-24-4 C22H25F5N6O3
—— 4-(9-((2,2-difluorocyclopropyl)methyl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946824-33-5 C23H28F2N6O3
—— 4-Methoxy-5,10-dihydropyrimido<4,5-b>chinolin. 31407-39-3 C12H11N3O
—— (S)-9-ethylamino-5-(thiophene-2-yl)-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-14-8 C16H19N5OS
—— 6-oxo-4-piperidin-1-yl-6,7-dihydro-5H-pyrimido[4,5-b][1,4]thiazine-7-carboxylic acid ethyl ester 54660-35-4 C14H18N4O3S
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(3-(4-methylpiperazin-1-yl)propyl)benzamide 946822-89-5 C31H46N8O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-4-yl)benzamide 946823-65-0 C28H39N7O3
—— Anthyridin-2,6-dithion 33548-27-5 C11H7N3S2
—— 2-methyl-1-(2-piperidin-1-yl-ethyl)-3-<i>o</i>-tolyl-2,3-dihydro-1<i>H</i>-quinazolin-4-one 17617-09-3 C23H29N3O
—— (S)-9-methylamino-5-{3-[4-(morpholine-4-carbonyl)-1,3-oxazol-2-yl]phenyl}-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-76-9 C25H27N7O4
—— 5-[(10-cyclopentyl-9-ethyl-7-methyl-8-oxo-2,4,7,9,10-pentazabicyclo[4.4.0]deca-2,4,11-trien-3-yl)amino]isoindole-1,3-dione 1018317-61-7 C21H23N7O3
—— 4-Piperidino-5-phenyl-5,10-dihydropyrimido<4,5-b>chinolin 31407-41-7 C16H18N4
—— 3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methylbenzamide 946823-07-0 C23H30N6O2
—— 9-amino-4-oxo-2-pyridin-4-yl-5,6,8,9-tetrahydro-4H-1,4a,7-triaza-benzocycloheptene-7-carboxylic acid ethyl ester 1174764-08-9 C16H19N5O3
—— (1R,2S,3S,4R,5S,6S,12R,19R,20R,21S,22R)-4,5,11,11,20,21-hexahydroxy-13,24,25-trioxa-7,9,16,18-tetrazaheptacyclo[12.8.1.13,6.119,22.02,12.07,12.018,23]pentacos-14(23)-ene-8,10,15,17-tetrone 87670-35-7 C18H18N4O13
—— 3,5-Dihydro-2-methyl-4H-pyrimido<4,5-b><1,4>diazepinon-(4) 30215-86-2 C8H8N4O
—— (S)-5-[3-cyano-5-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092114-33-4 C21H19N7O3S
—— (S)-5-[3-bromo-5-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092114-32-3 C20H19BrN6O3S
—— (2S,4R,5aS,9cS)-2-methyl-4-phthalimido-5a-triethylsilyloxy-4,5,5a,9c-tetrahydro-2a,9b-diaza-cyclo-penta[jk]fluorene-1,3-dione 1075239-96-1 C28H31N3O5Si
—— 5-(2-chloro-phenyl)-7-dimethylamino-1-methyl-1,3-dihydro-pyrido[3,2-<i>e</i>][1,4]diazepin-2-one 59451-16-0 C17H17ClN4O
—— 4-amino-8-(1,3-benzodioxol-5-yl)-6-phenyl-8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepine —— C20H17N5O2
—— 2-(2-Bromo-4-isopropyl-phenyl)-4-methyl-6-pentyl-6,7,8,9-tetrahydro-2H-2,3,5,6,9a-pentaaza-benzo[cd]azulen-1-one —— C23H30BrN5O
—— 2-chloro-8-(trifluoromethyl)-6H,11H-benzo[b]pyrimidino[5,4-f]-1,4-diazaperhydroepin-5-one —— C12H6ClF3N4O
—— 4,5,6,7-tetrahydro-2,4-diphenyl-4,7a,12b-triazadibenzo[e,g]azulene-1,3,8-trione —— C27H21N3O3
—— 4,5,6,7-tetrahydro-4-methyl-2-phenyl-4,7a,12b-triazadibenzo[e,g]azulene-1,3,8-trione —— C22H19N3O3
—— N-(4-((8,9-dimethoxy-5-methyl-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H29FN6O5
—— N-(4-((8,9-dimethoxy-11H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H24F2N6O5
—— N-(4-((8,9-dimethoxy-5-methyl-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C31H28F2N6O5
—— N-(4-((8,9-dimethoxy-6-oxo-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H25FN6O6
—— N-(4-fluorophenyl)-N-(4-((8-methoxy-2-methyl-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)cyclopropane-1,1-dicarboxamide —— C30H27FN6O4
—— N-(4-((8,9-dimethoxy-6-oxo-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H24F2N6O6
—— N-(4-fluorophenyl)-N-(4-((8-methoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)cyclopropane-1,1-dicarboxamide —— C29H25FN6O4
—— N-(4-((8,9-dimethoxy-6,11-dihydro-5H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)-3-fluorophenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H26F2N6O5
—— N-(4-((8,9-dimethoxy-11H-benzo[e]pyrimido[5,4-b][1,4]diazepin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide —— C30H25FN6O5