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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[(2,3-Difluorophenyl)methyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C21H21F2N3O3
3-[(2,3-Difluorophenyl)methyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[(4-Fluorophenyl)methyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C21H22FN3O3
3-[(4-Fluorophenyl)methyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[3-(Diethylamino)-2,2-dimethylpropyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C23H36N4O3
3-[3-(Diethylamino)-2,2-dimethylpropyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 12-benzyl-4-methyl-2-oxo-N-propyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide —— C22H26N4O2S
12-benzyl-4-methyl-2-oxo-N-propyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide
—— N-[2-(4-fluorophenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H27FN4O2
N-[2-(4-fluorophenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-benzyl-11-oxo-N-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C23H26N4O2
3-benzyl-11-oxo-N-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-Propan-2-yl-8-(pyrrolidine-1-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C20H26N4O2
3-Propan-2-yl-8-(pyrrolidine-1-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 11-oxo-3-propan-2-yl-N-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C21H24N4O2S
11-oxo-3-propan-2-yl-N-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[2-(4-fluorophenoxy)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C24H27FN4O3
N-[2-(4-fluorophenoxy)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 12-(Thiophen-3-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C15H15N3OS2
12-(Thiophen-3-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 3-benzyl-11-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H28N4O3
3-benzyl-11-oxo-N-[[(2S)-oxolan-2-yl]methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-Benzyl-8-(pyrrolidine-1-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C24H26N4O2
3-Benzyl-8-(pyrrolidine-1-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-benzyl-11-oxo-N-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H24N4O2S
3-benzyl-11-oxo-N-(thiophen-2-ylmethyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 8-(Azepane-1-carbonyl)-3-benzyl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C26H30N4O2
8-(Azepane-1-carbonyl)-3-benzyl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 12-[(2-Fluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H16FN3OS
12-[(2-Fluorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(4-Chlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H16ClN3OS
12-[(4-Chlorophenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(3,4-Difluorophenyl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C17H15F2N3OS
12-[(3,4-Difluorophenyl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 6-Methyl-12-(pyridin-2-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C17H18N4OS
6-Methyl-12-(pyridin-2-ylmethyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 5-Methyl-12-[(6-methylpyridin-2-yl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C18H20N4OS
5-Methyl-12-[(6-methylpyridin-2-yl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— N-[2-(3-methylphenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H30N4O2
N-[2-(3-methylphenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— diethyl (6S)-2-amino-6-methyl-4-oxo-5,9-dihydro-3H-pyrimido[4,5-b][1,4]diazepine-6,8-dicarboxylate —— C14H19N5O5
diethyl (6S)-2-amino-6-methyl-4-oxo-5,9-dihydro-3H-pyrimido[4,5-b][1,4]diazepine-6,8-dicarboxylate
—— 12-(2-Methoxyacetyl)-4-methyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C14H17N3O3S
12-(2-Methoxyacetyl)-4-methyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-(4-Chloro-1-methylpyrazole-3-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C15H14ClN5O2S
12-(4-Chloro-1-methylpyrazole-3-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(3R)-1-[(2R)-1-methoxypropan-2-yl]-5-oxopyrrolidine-3-carbonyl]-4-methyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C20H26N4O4S
12-[(3R)-1-[(2R)-1-methoxypropan-2-yl]-5-oxopyrrolidine-3-carbonyl]-4-methyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 4-Methyl-12-(2-methylpropanoyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C15H19N3O2S
4-Methyl-12-(2-methylpropanoyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-(3-Methoxypropanoyl)-5-methyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C15H19N3O3S
12-(3-Methoxypropanoyl)-5-methyl-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 5-Methyl-12-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C17H18N4O2S2
5-Methyl-12-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 4-methyl-12-[(2S)-2-methyl-3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C21H27N5O2S
4-methyl-12-[(2S)-2-methyl-3-(3,4,5-trimethylpyrazol-1-yl)propanoyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 5-Methyl-12-(2-methylpyridine-3-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C18H18N4O2S
5-Methyl-12-(2-methylpyridine-3-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-(2-Methylpyridine-3-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C17H16N4O2S
12-(2-Methylpyridine-3-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(2R)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C19H22ClN5O2S
12-[(2R)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(2,4-Dimethoxyphenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C19H21N3O3S
12-[(2,4-Dimethoxyphenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-(Pyridine-3-carbonyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C16H14N4O2S
12-(Pyridine-3-carbonyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-(1-Ethyl-3,5-dimethylpyrazole-4-carbonyl)-6-methyl-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C19H23N5O2S
12-(1-Ethyl-3,5-dimethylpyrazole-4-carbonyl)-6-methyl-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(4-Ethoxyphenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C19H21N3O2S
12-[(4-Ethoxyphenyl)methyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 4-Methyl-12-(3-methyl-1,2-oxazole-5-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C16H16N4O3S
4-Methyl-12-(3-methyl-1,2-oxazole-5-carbonyl)-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(2R)-butan-2-yl]-N,N-diethyl-4-methyl-2-oxo-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide —— C20H30N4O2S
12-[(2R)-butan-2-yl]-N,N-diethyl-4-methyl-2-oxo-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-triene-5-carboxamide
—— 12-[3-(3,5-Dimethylpyrazol-1-yl)propanoyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C18H21N5O2S
12-[3-(3,5-Dimethylpyrazol-1-yl)propanoyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C18H22N4O4S
12-[(3S)-1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— 12-(3,4-Dimethoxybenzoyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C19H19N3O4S
12-(3,4-Dimethoxybenzoyl)-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 6-methyl-12-[(2R)-2-methyl-3-(2-methylimidazol-1-yl)propanoyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one —— C19H23N5O2S
6-methyl-12-[(2R)-2-methyl-3-(2-methylimidazol-1-yl)propanoyl]-4-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),5,8-trien-2-one
—— 12-[(2,3-Dimethylimidazol-4-yl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one —— C16H19N5OS
12-[(2,3-Dimethylimidazol-4-yl)methyl]-6-thia-1,8,12-triazatricyclo[7.5.0.03,7]tetradeca-3(7),4,8-trien-2-one
—— N-[(1S)-1-(2-methoxyphenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C25H30N4O3
N-[(1S)-1-(2-methoxyphenyl)ethyl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-cycloheptyl-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C23H32N4O2
N-cycloheptyl-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— N-[(3R)-oxan-3-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide —— C21H28N4O3
N-[(3R)-oxan-3-yl]-11-oxo-3-propan-2-yl-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazoline-8-carboxamide
—— 3-[2-(4-Oxoquinazolin-3-yl)acetyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C22H19N5O3
3-[2-(4-Oxoquinazolin-3-yl)acetyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 8,9-Dimethoxy-3-[(1-methylpyrazol-4-yl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H23N5O3
8,9-Dimethoxy-3-[(1-methylpyrazol-4-yl)methyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[2-(Benzotriazol-1-yl)acetyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C20H18N6O2
3-[2-(Benzotriazol-1-yl)acetyl]-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-(Pyrazolo[1,5-a]pyrimidine-3-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C19H16N6O2
3-(Pyrazolo[1,5-a]pyrimidine-3-carbonyl)-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one
—— 3-[(1,5-Dimethylpyrazol-4-yl)methyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one —— C20H25N5O3
3-[(1,5-Dimethylpyrazol-4-yl)methyl]-8,9-dimethoxy-1,2,4,5-tetrahydro-[1,4]diazepino[7,1-b]quinazolin-11-one