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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(2-hydroxyethyl)piperidin-4-yl)-3-methoxybenzamide 1137867-39-0 C28H37F2N7O4
—— 4-(5-cyclopentyl-8-(ethoxycarbonyl)-6,7-dihydro-5H-imidazo[1,5-d]pyrimido[4,5-b][1,4]diazepin-3-ylamino)-3-methoxybenzoic acid 1214265-70-9 C25H28N6O5
—— 8-methyl-3-methylsulfanyl-5,10-dihydro-2,4,5,10-tetraazadibenzo-[a,d]cyclohepten-11-one 942910-90-9 C13H12N4OS
—— 7-methyl-3-methylsulfanyl-5,10-dihydro-2,4,5,10-tetraazadibenzo-[a,d]cyclohepten-11-one 942910-92-1 C13H12N4OS
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-1-yl)benzamide 1137867-48-1 C25H31F2N7O3
—— (R)-4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide 1137868-45-1 C28H37FN8O3
—— 9-cyclopentyl-2-(1-methanesulfonyl-2,3-dihydro-1H-indol-5-ylamino)-5,7,7-trimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 946824-02-8 C24H32N6O3S
—— 4-(9-cyclopentyl-7-ethyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1137868-31-5 C27H36FN7O3
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1137867-70-9 C26H33F2N7O3
—— (S)-4-(9-cyclopentyl-7-ethyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1137868-30-4 C29H40FN7O3
—— 13-chloro-10-methyl-8,9,10,14b-tetrahydro-5<i>H</i>-benzo[5,6][1,4]diazepino[1,7-<i>c</i>]quinazolin-6-one 30631-02-8 C17H16ClN3O
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)benzamide 1137867-85-6 C29H36F5N7O3
—— (S)-4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxypropyl)-3-methoxybenzamide 1137867-96-9 C25H32F2N6O4
—— (R)-4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1137867-73-2 C27H35F2N7O3
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(4-isopropylpiperazin-1-yl)-3-methoxybenzamide 1137868-12-2 C29H40F2N8O3
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperazin-1-yl)benzamide 1137868-10-0 C26H34F2N8O3
—— (S)-4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-3-yl)benzamide 1137868-05-3 C26H33F2N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethyl-N-methylbenzamide 946823-82-1 C25H34N6O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-4-yl)benzamide 946822-85-1 C28H33N7O3
—— 9-cyclopentyl-7,7-difluoro-5-methyl-2-(2-oxoindolin-6-ylamino)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1137867-54-9 C21H22F2N6O2
—— 9-cyclohexyl-2,4-dimethoxy-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1398113-64-8 C16H24N4O3
—— 2-amino-4-methoxy-6-[4-(trifluoromethyl)phenyl]-11H-pyrimido[4,5-b][1,4]benzodiazepine 1096144-92-1 C19H14F3N5O
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide 1137867-69-6 C27H36F2N8O3
—— 2-((R)-2,3-dihydro-1H-inden-1-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-19-4 C24H31N5O
—— 6-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methylpyridine-3-carboxamide 946823-89-8 C22H29N7O2
—— (S)-4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)benzamide 1137868-07-5 C28H37F2N7O3
—— 2-(1H-indazol-5-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-79-6 C22H27N7O
—— 2-(1,6-dihydro-4-methyl-6-oxopyridin-3-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-45-6 C21H28N6O2
—— 3-[3-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzoylamino]-azetidine-1-carboxylic acid tert-butyl ester 946824-07-3 C30H41N7O4
—— N-(4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)acetamide 946823-77-4 C23H30N6O2
—— 7-methyl-3-[methyl(1-methylpiperidin-4-yl)amino]-5,10-dihydro-2,4,5,10-tetraazadibenzo[a,d]cyclohepten-11-one 942910-33-0 C19H24N6O
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-1-yl)benzamide 1137867-97-0 C27H35F2N7O3
—— 4-amino-2-butoxy-8-((1,2,3,4-tetrahydroisoquinolin-6-yl)methyl)-7,8-dihydropteridin-6(5H)-one 1228586-43-3 C20H26N6O2
—— 2-[2-(4-hydroxy-phenyl)-ethylamino]-8-phenyl-7,8-dihydro-5H-pteridin-6-one 908300-88-9 C20H19N5O2
—— 9-cyclopentyl-5,7,7-trimethyl-2-[3-(4-methylpiperazine-1-carbonyl)-phenylamino]-5,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-6-one 946823-70-7 C27H37N7O2
—— (1S,2R,3S,4R)-4-(6-Chloro-8-ethoxy-7,8-dihydro-purin-9-yl)-cyclopentane-1,2,3-triol 142635-47-0 C12H17ClN4O4
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2,2,2-trifluoroethyl)-3-methoxybenzamide 946823-69-4 C25H31F3N6O3
—— 4-(6,7,8,9-tetrahydro-5,7,7-trimethyl-9-((R)-1-methylpyrrolidin-3-yl)-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946822-81-7 C24H33N7O3
—— 11-bromo-6-cyclohexyl-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>a</i>]quinazoline-5,13-dione 71982-02-0 C22H20BrN3O2
—— (rac)-2-chloro-9-cyclopentyl-7-(2-hydroxy-ethyl)-5,7,8,9-tetrahydro-pyrimido[4,5b][1,4]diazepin-6-one 1062244-99-8 C14H19ClN4O2
—— 1417619-61-4 C11H15N3O2
—— N-({(5S)-3-[4-(3-{[tert-butyl(dimethyl)silyl]oxy}-2-oxopiperidin-1-yl)-2-fluorophenyl]-2-oxo-1,3-oxazolidin-5-yl}methyl)-5-chlorothiophene-2-carboxamide 1093628-74-0 C26H33ClFN3O5SSi
—— 2-(1,6-dihydro-6-oxopyridin-3-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-44-5 C20H26N6O2
—— 4-(6,7,8,9-tetrahydro-5,7,7-trimethyl-9-((R)-1-methylpiperidine-3-yl)-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946823-60-5 C25H35N7O3
—— (S)-N,N-dimethyl 3-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,2,4-oxadiazole-5-carboxamide 1092112-27-0 C23H26N8O3
—— 3-[(7R)-8-cyclohexyl-7-methyl-2-[(3-methyl-1H-indazol-5-yl)amino]-6-oxo-7,8-dihydropteridin-5(6H)-yl]benzonitrile 1435458-50-6 C28H28N8O
—— 2-(4-aminophenylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-81-0 C21H28N6O
—— 8-chloro-1-methyl-6-phenyl-4<i>H</i>,6<i>H</i>-benzo[<i>b</i>]imidazo[1,5-<i>d</i>][1,4]diazepin-5-one 67045-89-0 C18H14ClN3O
—— 11-[{4-Methyl-1-piperazinyl)acetyl]-2-phenyl-6-(n-propyl)-5,6-dihydropyrimido[4,5-b][1,5]benzodiazepin-5-one 78438-45-6 C27H30N6O2
—— N-(4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxyphenyl)-2-methoxyacetamide 946823-68-3 C25H34N6O4