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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 9,11-diamino-6-(4-chlorophenyl)-6,7-dihydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepin-5(5aH)-one 1101201-55-1 C20H15ClN6O
—— N-[(2S)-7,15-dioxo-6,14,22-triazapentacyclo[12.8.0.02,6.08,13.016,21]docosa-1(22),8,10,12,16(21),17,19-heptaen-18-yl]acetamide 1359681-85-8 C21H18N4O3
—— 2-chloro-9-cyclopentyl-5,7-dimethyl-7-vinyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-48-3 C16H21ClN4O
—— (S)-2-(ethylamino)-6-(3-methyl-4-oxo-4,7-dihydro-3H-pyrrolo[2,3-d]pyrimidin-5-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410973-54-4 C19H22N8O2
—— 10-nitro-7,9-diphenyl-1,2,3,4,5,7,8,9-octahydropyrimido[1,6-a][1,3]diazepine 1350750-95-6 C20H22N4O2
—— 11-amino-6-phenyl-6,7-dihydroindeno[1,2-e]pyrimido[4,5-b][1,4]diazepin-5(5aH)-one 1101201-49-3 C20H15N5O
—— (S)-2-(ethylamino)-6-(3-(2-methoxyethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-72-0 C23H27N7O3
—— (S)-6-(3-(2-methoxyethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-2-(methylamino)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-69-5 C22H25N7O3
—— (S)-6-(3-(2-methoxyethyl)-4-oxo-3,4-dihydroquinazolin-8-yl)-2-(methylthio)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-42-6 C22H24N6O3S
—— (7aS,9S)-9-methoxy-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-97-1 C21H22N6O3S
—— (7aS,9S)-9-hydroxy-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-methylthio-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410975-95-9 C20H20N6O3S
—— 8-amino-3-carbethoxy-1,5-dimethyl-1H-pyrimido<4,5-c>-1,2-diazepin-6(7H)-one 80081-85-2 C12H15N5O3
—— 8-amino-5-carbethoxy-1,3-dimethyl-1H-pyrimido<4,5-c>-1,2-diazepin-6(7H)-one 80081-89-6 C12H15N5O3
—— 4-[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-fluoro-5-methoxy-benzoyl-amino]-piperidin-1-carboxylic acid tert-butyl ester 1137869-89-6 C31H40F3N7O5
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1,2,2,6,6-pentamethyl-piperidin-4-yl)-benzamide 1201691-72-6 C31H43F2N7O3
—— (2S)-19-fluoro-6,14,22-triazapentacyclo[12.8.0.02,6.08,13.016,21]docosa-1(22),8,10,12,16(21),17,19-heptaene-7,15-dione 1359681-76-7 C19H14FN3O2
—— 10-Chloro-2,6-dimethyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 946826-03-5 C9H11ClN4O
—— 3-{[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoylamino]-methyl}-azetidine-1-carboxylic acid tert-butyl ester 1201691-78-2 C30H39F2N7O5
—— 2-chloro-9-cyclohexyl-7,7-difluoro-8,9-dihydro-5H-pyrimido[5,4-b][1,4]diazepin-6(7H)-one 1137869-50-1 C13H15ClF2N4O
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1137867-68-5 C28H37F2N7O3
—— 2-chloro-9-cyclohexyl-7,7-difluoro-5-methyl-8,9-dihydro-5H-pyrimido[5,4-b][1,4]diazepin-6(7H)-one 1137869-51-2 C14H17ClF2N4O
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoic acid 1137867-67-4 C22H25F2N5O4
—— 2-[1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridin-3-yl]-6-methyl-8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepin-4-amine 1361569-00-7 C21H19FN8
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-fluoro-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-90-1 C25H29F3N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methyl-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-58-1 C26H32F2N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethyl-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-66-1 C27H34F2N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-pyran-4-yl)-3-trifluoromethyl-benzamide 1201692-74-1 C26H29F5N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-82-1 C27H34F2N6O4
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2,5-difluoro-N-(tetrahydro-pyran-4-yl)-benzamide 1201693-00-6 C25H28F4N6O3
—— 1-Oxo-1H,8H-4,7a,12b-triaza-dibenzo[e,g]azulene-2-carboxylic acid ethyl ester 99390-30-4 C18H15N3O3
—— 6-Methyl-4H,9H-2-oxa-1,4a,8,9-tetraaza-benzo[f]azulene-5,10-dione 190070-43-0 C10H8N4O3
—— 8-amino-1,3,5-trimethyl-1H-pyrimido<4,5-c>-1,2-diazepin-6(7H)-one 70311-77-2 C10H13N5O
—— 4-[9-cyclopentyl-7,7-difluoro-6-oxo-5-(2,2,2-trifluoro-ethyl)-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino]-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1201692-31-0 C28H34F5N7O3
—— (rac)-4-(9-allyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1062242-52-7 C26H35N7O3
—— 4-(9-cyclopentyl-7-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1137206-31-5 C27H37N7O3
—— (rac)-3-methoxy-4-(8-methyl-9-oxo-1,3,5,8-tetraaza-tricyclo[8.3.1.0(2,7)]tetradeca-2,4,6-trien-4-ylamino)-N-(1-methyl-piperidin-4-yl)-benzamide 1062242-58-3 C25H33N7O3
—— 10-chloro-6-methyl-2-(2-methylpropyl)-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-09-3 C12H17ClN4O
—— (rac)-2-chloro-9-cyclohexyl-7-methyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-15-8 C14H19ClN4O
—— (rac)-4-[5,7-dimethyl-9-(3-methyl-butyl)-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino]-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1062241-42-2 C28H41N7O3
—— 10-chloro-2-cyclopentyl-4-ethyl-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 946826-63-7 C15H21ClN4O
—— (rac)-9-allyl-2-chloro-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-65-1 C12H15ClN4O
—— 2-benzyl-10-chloro-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-24-2 C15H15ClN4O
—— (rac)-4-(9-cyclobutyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1062242-16-3 C27H37N7O3
—— (rac)-2-chloro-5,7-dimethyl-9-(3-methyl-butyl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-46-5 C14H21ClN4O
—— (rac)-2-chloro-9-cyclopentylmethyl-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-21-9 C15H21ClN4O
—— 10-chloro-2-(1-methoxypropan-2-yl)-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-36-6 C12H17ClN4O2
—— (rac)-2-chloro-9-cyclobutyl-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062245-11-7 C13H17ClN4O
—— (rac)-9-benzyl-2-chloro-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-66-9 C16H17ClN4O
—— (rac)-2-chloro-5,7-dimethyl-9-(tetrahydro-pyran-4-yl)-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062244-86-3 C14H19ClN4O2
—— 10-chloro-2-(2-methoxyethyl)-6-methyl-2,6,9,11-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-5-one 1001346-33-3 C11H15ClN4O2