| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 4-chloro-6-(2-hydroxyethyl)-9-methyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one | 1228425-69-1 | C10H13ClN4O2 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(4-(2-hydroxyethyl)piperazin-1-yl)-3-methoxybenzamide | 1137869-13-6 | C27H36F2N8O4 |
| —— | 4-(6,7,8,9-tetrahydro-5,7,7-trimethyl-9-neopentyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide | 946824-32-4 | C24H34N6O3 |
| —— | (R)-4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxypropyl)-3-methoxybenzamide | 1137867-95-8 | C25H32F2N6O4 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-ethyl-3-methoxybenzamide | 1137869-01-2 | C23H28F2N6O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethylazetidin-3-yl)-3-methoxybenzamide | 1137868-64-4 | C26H33F2N7O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-isopropylazetidin-3-yl)-3-methoxybenzamide | 1137868-65-5 | C27H35F2N7O3 |
| —— | (S)-3-methyl-5-[2-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one | 1092114-29-8 | C20H20N6O3S |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-methoxypyridin-3-yl)benzamide | 946825-42-9 | C29H35N7O4 |
| —— | (Z)-4-(7-(but-2-enyl)-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1157848-63-9 | C31H43N7O3 |
| —— | 9-cyclohexyl-7,7-difluoro-2-(2-methoxy-4-(4-methylpiperazine-1-carbonyl)-phenylamino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137867-91-4 | C27H35F2N7O3 |
| —— | N-(cyclohexylmethyl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 946824-84-6 | C30H42N6O3 |
| —— | 4-[(5-cyclopentyl-4-ethyl-2-methyI-3-oxo-2,4,5,7,9-pentazabicyclo[4.4.0]deca-6,8,10-trien-8-yl)amino]-3-methoxy-N-(2-pyrrolidin-1-ylethyl)benzamide | 1018317-73-1 | C27H38N8O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1137868-74-6 | C27H37F2N7O2 |
| —— | 9-cyclopentyl-2-(2-methoxy-4-(3-methoxyazetidine-1-carbonyl)phenylamino)-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 946825-27-0 | C27H36N6O4 |
| —— | 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclobutane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-methylbenzamide | 946823-22-9 | C25H32N6O3 |
| —— | 4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-1-methylpyrrolidin-3-yl)benzamide | 1157847-90-9 | C30H43N7O3 |
| —— | 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((S)-1-(cyclopropylmethyl)pyrrolidin-3-yl)-3-methoxybenzamide | 946823-37-6 | C31H43N7O3 |
| —— | 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((S)-tetrahydrofuran-3-yl)-3-methoxybenzamide | 946824-36-8 | C27H36N6O4 |
| —— | 5-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-methylpiperidin-4-yl)picolinamide | 1137868-82-6 | C25H32F2N8O2 |
| —— | 2,3,4,5-tetrahydro-2-chloroacetyl-1,4-diazepino<2,1-b>quinazolin-7(1H)-one | 166770-96-3 | C14H14ClN3O2 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((tetrahydrofuran-2-yl)methyl)benzamide | 946824-80-2 | C28H38N6O4 |
| —— | benzyl 4-(4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamido)piperazine-1-carboxylate | 1137869-53-4 | C34H40F2N8O5 |
| —— | 4-(6,7,8,9-tetrahydro-9-((R)-tetrahydrofuran-3-yl)-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide | 946824-54-0 | C23H30N6O4 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-fluoro-5-methoxy-N-(1-methylpiperidin-4-yl)benzamide | 1137868-58-6 | C27H34F3N7O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-morpholinobenzamide | 1137869-10-3 | C25H31F2N7O4 |
| —— | 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-pyrrolidin-3-yl)benzamide | 1157848-38-8 | C29H39N7O3 |
| —— | 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-((1R,3R)-3-hydroxycyclopentyl)-3-methoxybenzamide | 946825-95-2 | C28H36N6O4 |
| —— | 4-(9-cyclobutyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide | 946824-31-3 | C23H30N6O3 |
| —— | 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-oxoazepan-3-yl)benzamide | 1137869-14-7 | C27H33F2N7O4 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(hydroxymethyl)cyclopentyl)-3-methoxybenzamide | 946825-70-3 | C29H40N6O4 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(furan-2-ylmethyl)-3-methoxybenzamide | 946824-78-8 | C28H34N6O4 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-isopropyl-3-methoxybenzamide | 946825-54-3 | C26H36N6O3 |
| —— | 3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-methoxyethyl)benzamide | 946824-08-4 | C25H34N6O3 |
| —— | N-(3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-4-methoxyphenyl)acetamide | 946824-22-2 | C24H32N6O3 |
| —— | 2-(4-aminophenylamino)-9-cyclopentyl-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1157849-06-3 | C19H24N6O |
| —— | 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-2H-pyran-4-yl)-3-methoxybenzamide | 946823-97-8 | C28H38N6O4 |
| —— | 9-cyclopentyl-2-(4-(5,5-dimethyl-4,5-dihydro-1H-imidazol-2-yl)-2-methoxyphenylamino)-5,7,7-trimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 946825-73-6 | C27H37N7O2 |
| —— | 6-(2-methoxy-ethyl)-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>a</i>]quinazoline-5,13-dione | 71981-90-3 | C19H17N3O3 |
| —— | 9-cyclopentyl-2-(4-(4-(cyclopropylmethyl)piperazine-1-carbonyl)-2-methoxyphenylamino)-7,7-difluoro-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137868-70-2 | C29H37F2N7O3 |
| —— | 4-chloro-9-methyl-6-o-tolyl-8,9-dihydro-5H-pyrimido[4,5-e][1,4]diazepin-7(6H)-one | 1228425-51-1 | C15H15ClN4O |
| —— | 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1,3-dihydroxy-2-methylpropan-2-yl)-3-methoxybenzamide | 946824-00-6 | C27H38N6O5 |
| —— | 9-benzyl-2-chloro-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 946826-02-4 | C17H19ClN4O |
| —— | (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2,3-dihydroxypropyl)-3-methoxybenzamide | 946825-58-7 | C26H36N6O5 |
| —— | 9-cyclopentyl-2-(4-(4-(cyclopropylmethyl)piperazine-1-carbonyl)-5-fluoro-2-methoxyphenylamino)-7,7-difluoro-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one | 1137868-71-3 | C29H36F3N7O3 |
| —— | 6-[2-(2-amino-6-chloro-4H-quinazolin-3-yl)ethylamino]-3-[(4-fluorophenyl)methyl]-1-[[4-(trifluoromethoxy)phenyl]methyl]-1,3,5-triazine-2,4-dione | 1148127-94-9 | C28H24ClF4N7O3 |
| —— | 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((1R,3R)-3-(hydroxycyclopentyl)methyl)-3-methoxybenzamide | 946825-75-8 | C29H40N6O4 |
| —— | N-(3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)cyclobutanecarboxamide | 946824-15-3 | C26H34N6O2 |
| —— | (R)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-2H-pyran-4-yl)benzamide | 946824-56-2 | C27H36N6O4 |
| —— | N-(2-chloropyridin-4-yl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide | 946825-41-8 | C28H32ClN7O3 |