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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— (S)-2-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3-oxazole-5-carboxamide 1092112-72-5 C22H23N7O3
—— (S)-9-methylthio-5-[3-(5-trifluoromethyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-67-1 C20H17F3N6O2S
—— (rac)-3-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-pyridin-3-yl-benzamide 1062242-73-2 C26H29N7O2
—— (S)-9-amino-5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-99-3 C19H19N7O2
—— (S)-5-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-31-2 C20H20N6O2S
—— (S)-9-ethylamino-5-[3-(4,5-dimethyl-1,2,4-triazol-3-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-33-8 C22H26N8O
—— (S)-9-ethylamino-5-[3-(5-ethylamino-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-08-7 C22H26N8O2
—— (S)-3-(2-methoxyethyl)-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092114-05-0 C22H24N6O4S
—— (+/-)-9-amino-4-oxo-2-pyrimidin-4-yl-5,6,8,9-tetrahydro-4H-1,4a,7-triaza-benzocycloheptene-7-carboxylic acid ethyl ester hydrobromide 1174764-02-3 BrH*C15H18N6O3
—— 1-Cyclohexyl-4-(4'-methoxy-benzyliden)-3-hydroxy-pyrrolidin 4809-14-7 C18H25NO2
—— (S)-9-ethylamino-5-[3-(5-methoxymethyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-96-0 C22H25N7O3
—— (S)-5-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-98-2 C20H21N7O2
—— (S)-3-(2-methoxyethyl)-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092112-42-9 C22H25N7O4
—— (S)-5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-84-2 C20H20N6O2S
—— (rac)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-ethyl-piperidin-4-yl)-3-methyl-benzamide 1062243-40-6 C29H41N7O2
—— (S)-9-ethylamino-5-[3-(1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-01-0 C20H21N7O2
—— (S)-9-ethylamino-5-[1-(thiazolyl-2-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-76-6 C21H29N7OS
—— (S)-5-[3-(1,2,4-oxadiazol-3-yl)phenyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-28-1 C20H21N7O2
—— (S)-3-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-4-methyl-1,2,4-oxadiazol-5(4H)-one 1092112-36-1 C21H23N7O3
—— (rac)-2-(4-benzyloxy-phenylamino)-9-cyclopentyl-5,7-dimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1062242-82-3 C27H31N5O2
—— (rac)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-dimethylamino-propyl)-benzamide 1062243-34-8 C26H37N7O2
—— (S)-5-[5-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)pyridin-3-yl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092111-89-1 C20H22N8O3
—— 3-[(7R)-2-[(4-fluoro-1H-indazol-5-yl)amino]-7-methyl-6-oxo-8-(tetrahydro-2H-pyran-4-yl)-7,8-dihydropteridin-5(6H)-yl]benzonitrile 1435461-12-3 C26H23FN8O2
—— (S)-5-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092112-35-0 C21H23N7O3
—— (S)-5-[3-(5-methoxymethyl-1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-87-5 C21H22N6O3S
—— (S)-5-[3-(5-methoxymethyl-1,3,4-oxadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-69-3 C21H22N6O3S
—— 9-((5-methylthiazol-2-yl)ethynyl)-3,4-dihydro-1H-pyrazino[2,1-b]quinazolin-6(2H)-one hydrochloride 1312449-82-3 C17H14N4OS*ClH
—— (S)-9-ethylamino-5-[3-(5-hydroxymethyl-1,2,4-oxadiazol-3-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-29-2 C21H23N7O3
—— (S)-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,3,4-oxadiazol-2(3H)-one 1092114-09-4 C25H27N7O4S
—— (rac)-N-[5-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-hydroxy-phenyl]-isonicotinamide 1062242-05-0 C26H29N7O3
—— 1416011-93-2 C20H17N3O2
—— (S)-5-{3-[9-ethylamino-6-oxo-7-(thiazol-2-yl)-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl]phenyl}-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092113-06-8 C24H24N8O3S
—— (S)-5-[3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1234694-03-1 C22H22N6O2S
—— (S)-5-[3-(5-hydroxymethyl-1,3-oxazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-43-6 C21H21N5O3S
—— (S)-9-ethylamino-5-[3-(5-trifluoromethyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-02-1 C21H20F3N7O2
—— (S)-9-ethylamino-5-[3-(5-hydroxymethyl-1,3-oxazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-67-8 C22H24N6O3
—— (S)-9-ethylamino-5-[1-(pyridin-2-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-71-1 C23H31N7O
—— (S)-5-[3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)phenyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-23-6 C23H25N7O2
—— (S)-5-[3-(5-methyl-1,3-oxazol-2-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-66-7 C21H22N6O2
—— (S)-9-methylamino-5-(1-methylindoline-2,3-dion-4-yl)-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-91-8 C20H20N6O3
—— (S)-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-(2-oxopropyl)-1,3,4-oxadiazol-2(3H)-one 1092112-47-4 C22H23N7O4
—— (S)-9-ethylamino-5-[3-(2-methyl-2H-tetrazol-5-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-81-6 C20H23N9O
—— (S)-3-ethyl-5-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092112-38-3 C22H25N7O3
—— (2S)-methyl 2-(6-((((2R,3R,4R)-5-(2-amino-6-methoxy-9H-purin-9-yl)-3,4-dihydroxy-4-methyltetrahydrofuran-2-yl)methoxy)((S)-1-oxo1-(tetrahydro-2H-pyran-4-yloxy)propan-2-ylamino)phosphoryloxy)naphthalen-2-yl)propanoate 1234490-93-7 C34H43N6O12P
—— (S)-5-(5-cyanoindole-3-yl)-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-85-0 C21H21N7O
—— (S)-9-ethylamino-5-[(thiophene-3-yl)methyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-19-3 C17H21N5OS
—— (S)-5-[3-(5-cyclopropyl-1,3,4-oxadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-62-6 C22H22N6O2S
—— (R)-7-ethyl-8-isopropyl-5-methyl-2-(2-oxo-2-(4-fluorophenyl)ethyl)-7,8-dihydropteridin-6(5H)-one 1313516-85-6 C20H23FN4O2
—— (S)-9-ethylamino-5-[1-(pyridin-3-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-79-9 C23H31N7O
—— (S)-9-ethylamino-5-[3-(5-methylthio-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-11-2 C21H23N7O2S