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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-cyclopentyl-5-ethyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-42-3 C27H34F2N6O4
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methyl-benzamide 1201692-34-3 C21H24F2N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-5-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1201692-46-7 C29H39F2N7O3
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-5-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methyl-benzamide 1201692-45-6 C24H30F2N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201692-33-2 C20H22F2N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzamide 1201692-13-8 C19H20F2N6O2
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-5-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-48-9 C28H36F2N6O4
—— 4-(9-cyclopentyl-5-ethyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methyl-benzamide 1201692-39-8 C23H28F2N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-5-propyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-benzamide 1201692-26-3 C22H26F2N6O2
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-yl)-benzamide 1201692-18-3 C26H33F2N7O3
—— 4-(9-cyclopentyl-5-ethyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methyl-benzamide 1201692-21-8 C22H26F2N6O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-fluoro-5-methoxy-N-methyl-benzamide 1201692-51-4 C22H25F3N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydro-pyran-4-yl)-benzamide 1201692-36-5 C25H30F2N6O4
—— 8-methoxy-3-[methyl-(1-methylpiperidin-4-yl)amino]-5,10-dihydro-2,4,5,10-tetraazadibenzo[a,d]cyclohepten-11-one 942910-38-5 C19H24N6O2
—— (S)-5-[3-(7-cyclopropylamino-9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092114-85-6 C23H25N7O3S
—— tert-butyl 4-[[4-[(6-cyclopentyl-2-methyl-3-oxo-2,6,8,10-tetrazabicyclo[5.4.0]undeca-7,9,11-trien-9-yl)amino]-3-methoxy-benzoyl]amino]piperidine-1-carboxylate 946822-64-6 C31H43N7O5
—— (S)-5-[3-(7-chloro-9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092114-81-2 C20H19ClN6O3S
—— (S)-5-[3-(7,9-bis(Methylamino)-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092113-01-3 C21H24N8O3
—— (S)-5-[3-(7-methylamino-9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092114-82-3 C21H23N7O3S
—— (E)-benzomalvin B 157047-97-7 C24H17N3O2
—— (S)-5-[3-(1-Acetylpiperidin-4-yloxy)phenyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-95-2 C25H32N6O3
—— (S)-2-methylamino-6-(4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410970-92-1 C19H19N7O2
—— (S)-6-(2,3-dimethyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl)-2-methylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-07-1 C21H23N7O2
—— (S)-9-Ethylamino-5-[3-(1-methylpiperidin-4-yloxy)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-93-0 C24H32N6O2
—— (S)-9-ethylamino-5-[3-(piperidin-4-yloxy)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-92-9 C23H30N6O2
—— 4-methyl-1,4-diazepano<2,1-b>quinazolin-11(11aH)-one 126411-73-2 C13H15N3O
—— (+/-)-4-Amino-5-chloro-2-methoxy-N-(4-oxo-2-pyrimidin-4-yl-4,5,6,7,8,9-hexahydro-1,4a,7-triaza-benzocyclohepten-9-yl)-benzamide 1174763-68-8 C20H20ClN7O3
—— 2'-chloro-9'-cyclopentyl-5'-methyl-8',9'-dihydrospiro[cyclobutane-1,7'-pyrimido[4,5-b][1,4]diazepin]-6'(5'H)-one 946826-25-1 C16H21ClN4O
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-fluoro-benzoic acid 1137870-06-4 C20H20F3N5O3
—— (S)-2-amino-6-(3-methyl-4-oxo-3,4-dihydroquinazolin-8-yl)-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-91-3 C19H19N7O2
—— 4-{3-[4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzoylamino]-propyl}-piperazine-1-carboxylic acid tert-butyl ester 1201691-81-7 C33H46F2N8O5
—— 6-(4-Methoxyphenyl)-8-phenyl-3,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-4-one 135039-32-6 C20H18N4O2
—— 2,4-diphenyl-6-hydroxy-2,3-dihydropyrimido<5,6-b>-1H-1,5-diazepine 135039-26-8 C19H16N4O
—— 8-(4-bromophenyl)-6-phenyl-8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepin-4-ol 135039-28-0 C19H15BrN4O
—— 6-(4-Bromophenyl)-8-phenyl-3,7,8,9-tetrahydropyrimido[4,5-b][1,4]diazepin-4-one 135039-34-8 C19H15BrN4O
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2,5-difluoro-benzoic acid 1201692-97-8 C20H19F4N5O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-dimethylamino-2,2-dimethyl-propyl)-3-methoxy-benzamide 1201691-52-2 C28H39F2N7O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-[2-(4-methyl-piperazin-1-yl)-ethyl]-benzamide 1201691-42-0 C28H38F2N8O3
—— 6,7,8,9-tetrahydro-5H-pyrimido<4,5-b><1,4>diazepine-6,8-dione 154124-55-7 C7H6N4O2
—— (S)-9-Ethylamino-5-[1-(5-aminocarbonylpyridin-2-yl)piperidin-4-yl]methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-73-3 C24H32N8O2
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-dimethylamino-ethyl)-2-fluoro-5-methoxy-benzamide 1201692-54-7 C25H32F3N7O3
—— 1,5,9,13-Tetrazatetracyclo[7.7.2.05,17.013,18]octadecane 74199-15-8 C14H26N4
—— perhydro-3a,5a,8a,11a-tetraazacyclohepta[d,e,f]phenanthrene 74199-13-6 C13H24N4
—— 1,5,9,12-Tetrazatetracyclo[7.6.2.05,17.012,16]heptadecane 201605-50-7 C13H24N4
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethyl-benzoic acid 1137870-11-1 C22H25F2N5O3
—— (S)-5-[3-(5-isopropyl-1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-86-4 C22H24N6O2S
—— 9-Benzyl-2,4-dimethoxy-7-(2-methoxy-2-oxoethyl)-5-methyl-8,9-dihydro-7H-pyrimido[4,5-e][1,4]diazepin-6-ium-6-olate 348636-03-3 C20H24N4O5
—— 9-Benzyl-2,4-dimethoxy-7-(2-methoxy-2-oxoethyl)-8,9-dihydro-7H-pyrimido[4,5-e][1,4]diazepin-6-ium-6-olate 348636-02-2 C19H22N4O5
—— 9-chloro-7-(2-fluorophenyl)-1,2,4,5-tetrahydro-2-methyl-3H-pyrimido<1,6-a><1,4>benzodiazepin-3-one 112634-56-7 C19H17ClFN3O
—— 1-chloro-7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraazadibenzo[a,d]cycloheptene 870258-04-1 C13H13ClN4O2