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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(((1S,2S)-2-hydroxycyclohexyl)methyl)-3-methoxybenzamide 946825-20-3 C30H42N6O4
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(tetrahydro-2H-pyran-4-yl)benzamide 946824-46-0 C28H36N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(3-(trifluoromethyl)pyridin-4-yl)benzamide 946825-50-9 C29H32F3N7O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclopentyl-3-methoxybenzamide 946823-92-3 C28H38N6O3
—— 4-(9-cyclopentyl-7-fluoro-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1137868-24-6 C26H34FN7O3
—— N-(5-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-methylphenyl)acetamide 946824-26-6 C24H32N6O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methyl-3-(trifluoromethoxy)benzamide 946824-06-2 C24H29F3N6O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-2-yl)benzamide 946825-29-2 C28H33N7O3
—— 2-(3-nitrophenylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-91-2 C21H26N6O3
—— (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2,3-dihydro-1H-inden-1yl)-3-methoxy-benzamide 946825-10-1 C32H38N6O3
—— 4-[(9-cyclopentyl-5,7,7-trimethyl-6-oxo-8H-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-N-[1-(hydroxymethyl)cyclopropyl]-3-methoxybenzamide 946825-82-7 C27H36N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-4-ylmethyl)benzamide 946825-13-4 C29H35N7O3
—— (S)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1137867-44-7 C26H33F2N7O3
—— 2-methyl-6-(1-methyl-2-ethylthio-4-hydroxy-1-butenyl)-5,6-dihydropyrimido<4,5-d>pyrimidine 118743-89-8 C14H20N4OS
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(cyclopentylmethyl)-3-methoxybenzamide 946825-46-3 C29H40N6O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-3-yl)benzamide 946825-06-5 C28H33N7O3
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-(((1S,2S)-2-hydroxycyclohexyl)methyl)-3-methoxybenzamide 946825-68-9 C30H40N6O4
—— (S)-9-ethylamino-5-(2-fluoro-4-methoxybenzyl)-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-16-0 C20H24FN5O2
—— 6-(2-hydroxyphenyl)-8-phenyl-8,9-dihydro-7H-pyrimido[4,5-b][1,4]diazepin-4-ol 135039-30-4 C19H16N4O2
—— N-[3-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-phenyl]-methanesulfonamide 946824-14-2 C22H30N6O3S
—— (S)-5-[5-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)-2-fluorophenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092112-61-2 C21H22FN7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(3,3,3-trifluoro-2-hydroxypropyl)benzamide 946825-90-7 C26H33F3N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((1R,3R)-3-(hydroxymethyl)cyclopentyl)-3-methoxybenzamide 946825-76-9 C29H40N6O4
—— (S)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1157847-22-7 C26H35N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((1R,2R)-2-hydroxycyclopentyl)-3-methoxybenzamide 946825-60-1 C28H38N6O4
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-(3,3-difluorocyclobutyl)-3-methoxybenzamide 946825-85-0 C27H32F2N6O3
—— 5-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)indoline-2,3-dione 946824-03-9 C23H26N6O3
—— (S)-5-[(5-cyanopyridin-2-yl)methyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-21-7 C19H21N7O
—— 3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-5-(trifluoromethyl)-N-methylbenzamide 946824-04-0 C24H29F3N6O2
—— 4-(9-(cyclobutylmethyl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946823-86-5 C24H32N6O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-ethoxy-N-(1-isopropylpiperidin-4-yl)benzamide 946823-99-0 C32H47N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((5-methylisoxazol-3-yl)methyl)benzamide 946825-51-0 C28H35N7O4
—— (S)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-3-ylmethyl)benzamide 1157847-36-3 C26H35N7O3
—— 4-((3aR,10aS)-4-cyclopentyl-9-methyl-10-oxo-1,2,3,3a,4,9,10,10a-octahydro-4,5,7,9-tetraaza-benzo[f]azulen-6-ylamino)-3-methoxy-N-methylbenzamide 946822-76-0 C25H32N6O3
—— 4-(9-(3,3-difluorocyclobutyl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-2H-pyran-4-yl)-3-methoxybenzamide 946824-35-7 C27H34F2N6O4
—— N-(3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)phenyl)-2-methoxyacetamide 946824-11-9 C24H32N6O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-methoxy-ethyl)-benzamide 946824-86-8 C26H36N6O4
—— 9-cyclopentyl-2-[3-(3-cyclopropyl-3-fluoro-azetidine-1-carbonyl)-phenylamino]-5,7,7-trimethyl-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 946824-16-4 C28H35FN6O2
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyridin-3-ylmethyl)benzamide 946824-97-1 C29H35N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-(2-hydroxyethoxy)ethyl)-3-methoxybenzamide 946825-53-2 C27H38N6O5
—— N-(bicyclo[2.2.1]heptan-2-yl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide 946825-11-2 C30H40N6O3
—— (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-hydroxypropan-2-yl)-3-methoxybenzamide 946825-81-6 C26H36N6O4
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3,3,3-trifluoropropyl)-3-methoxybenzamide 946823-95-6 C26H33F3N6O3
—— N-tert-butyl-1-(cyclopropanecarbonyl)-5-oxo-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine-2-carboxamide 1414359-36-6 C18H23N3O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-ethyl-3-methoxybenzamide 946825-25-8 C25H34N6O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N,N-dimethylbenzamide 946825-18-9 C25H34N6O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(3-methoxypropyl)benzamide 946824-88-0 C27H38N6O4
—— 2-(3-(1H-pyrazol-3-yl)phenylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946824-01-7 C24H29N7O
—— 2,2-dioxo-1,3,4,5-tetrahydro-[1,4]thiazepino[3,4-b]quinazolin-7-one 112377-96-5 C12H12N2O3S
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-hydroxy-2,2-dimethylpropyl)-3-methoxybenzamide 946825-12-3 C28H40N6O4