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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— (S)-5-[3-(9-ethylamino-7-methoxy-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-methyl-1,3,4-oxadiazol-2(3H)-one 1092113-00-2 C22H25N7O4
—— (S)-9-ethylamino-5-[3-(5-isopropyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-92-6 C23H27N7O2
—— (S)-9-ethylamino-5-[3-(1-methyl-1H-tetrazol-5-yl)phenyl]-1,2,3,3a,4,5,-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-83-8 C20H23N9O
—— (S)-9-ethylamino-5-[3-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-32-7 C21H23N7O2
—— (S)-9-ethylamino-5-[3-(5-isopropyl-1,2,4-oxadiazol-3-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-20-3 C23H27N7O2
—— (S)-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-(tetrahydro-2H-pyran-4-yl)-1,3,4-oxadiazol-2(3H)-one 1092112-43-0 C24H27N7O4
—— 8-fluoro-3-(pyridin-2-ylethynyl)-7,8,9,10-tetrahydroazepino[2,1-b]quinazolin-12(6H)-one hydrochloride 1312450-92-2 C20H16FN3O*ClH
—— methyl (S)-5-methyl-2-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3-oxazole-4-carboxylate 1092114-55-0 C23H23N5O4S
—— (S)-5-{3-[5-(3-cyanophenyl)-1,3,4-oxadiazol-2-yl]phenyl}-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-95-9 C27H24N8O2
—— (S)-3-methyl-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-thiadiazol-2(3H)-one 1092114-26-5 C20H20N6O2S2
—— 2'-[[5-Methoxy-6-(4-methylimidazol-1-yl)pyridin-3-yl]amino]-8'-methyl-5'-(2,2,2-trifluoroethyl)spiro[cyclopropane-1,7'-pteridine]-6'-one 1452228-15-7 C21H21F3N8O2
—— (S)-5-[3-(5-cyano-1,3-oxazol-2-yl)phenyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-70-3 C22H21N7O2
—— (S)-5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-78-4 C20H20N6OS2
—— (S)-3-methyl-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092112-34-9 C20H21N7O3
—— (S)-7-methoxy-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-72-1 C12H16N4O2S
—— (S)-5-[3-(5-ethyl-1,3,4-oxadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-60-4 C21H22N6O2S
—— (S)-9-ethylamino-5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-12-3 C21H23N7OS
—— (12S,20aS)-2-(tert-butoxycarbonyl)-16-fluoro-8,13-dimethyl-6,9,14-trioxo-1,2,3,4,7,8,9,10,11,12,13,14,20,20a-tetradecahydro-6H-pyrazino[2,1-c][1,4,7,12]benzoxatriazacyclopentadecine-12-carboxylic acid 1264222-15-2 C26H35FN4O8
—— (S)-3-isopropyl-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092114-02-7 C22H24N6O3S
—— (rac)-2-chloro-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-pyridin-4-yl-benzamide 1062243-11-1 C26H28ClN7O2
—— (S)-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-(2-morpholino-2-oxoethyl)-1,3,4-oxadiazol-2(3H)-one 1092112-51-0 C25H28N8O5
—— (S)-5-(1-tert-butoxycarbonyl-5-cyanoindole-3-yl)-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-61-8 C26H29N7O3
—— (S)-5-[3-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-82-0 C22H22N6OS2
—— (S)-3-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,2,4-oxadiazole-5-carboxamide 1092112-30-5 C21H22N8O3
—— (S)-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-3-(tetrahydro-2H-pyran-4-yl)-1,3,4-oxadiazol-2(3H)-one 1092114-06-1 C24H26N6O4S
—— (S)-5-[3-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-31-6 C20H21N7O2
—— (S)-9-ethylamino-5-[3-(1-isopropylpiperidin-4-yloxy)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-94-1 C26H36N6O2
—— 6,7,8,9-Tetrahydro-2-phenyl-5H-pyrimido-[5,4-e][1,4]-diazepin-9-one 195984-68-0 C13H12N4O
—— (S)-5-[3-(5-hydroxymethyl-1,2,4-oxadiazol-3-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-92-2 C20H20N6O3S
—— N-[1-(2-amino-2-methyl-propionyl)-piperidin-4-yl]-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-benzamide 1201691-75-9 C30H40F2N8O4
—— (S)-3-methyl-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-thiadiazol-2(3H)-one 1092112-55-4 C20H21N7O2S
—— (S)-5-[3-(5-ethylamino-1,3,4-oxadiazol-2-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-09-8 C21H24N8O2
—— (S)-5-(3-methylbenzo[d]oxazol-2(3H)-on-5-yl)-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-63-0 C19H19N5O3S
—— (S)-5-cyclopentylmethyl-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-49-3 C17H25N5O
—— (S)-3-ethyl-5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092114-01-6 C21H22N6O3S
—— (S)-3-[3-(9-ethylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-4-methyl-1,2,4-thiadiazol-5(4H)-one 1092112-53-2 C21H23N7O2S
—— (S)-9-ethylamino-5-[3-(5-hydroxymethyl-1,3,4-oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-93-7 C21H23N7O3
—— (S)-3-ethyl-5-[3-(9-methylamino-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-1,3,4-oxadiazol-2(3H)-one 1092112-37-2 C21H23N7O3
—— (S)-9-ethylamino-5-(1-phenylpiperidin-4-yl)methyl-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-78-8 C24H32N6O
—— (S)-5-[3-(2-methyl-2H-tetrazol-5-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-82-7 C19H21N9O
—— (S)-5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-13-4 C20H21N7OS
—— (S)-9-ethylamino-5-[3-(pyridin-4-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10.10b-tetraazabenzo[e]azulen-6-one 1092111-59-5 C23H24N6O
—— (S)-6-(3-cyclopropyl-4-oxo-3,4-dihydroquinazolin-8-yl)-2-ethylamino-6,7,7a,8,9,10-hexahydro-5H-pyrimido[5,4-f]pyrrolo[1,2-a][1,4]diazepin-5-one 1410971-93-5 C23H25N7O2
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-13-9 C27H35N7O3
—— (S)-5-[3-(5-benzyl-1,3,4-oxadiazol-2-yl)phenyl]-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-90-4 C27H27N7O2
—— (S)-5-[3-(5-cyano-1,3-oxazol-2-yl)phenyl]-9-methylthio-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092114-50-5 C21H18N6O2S
—— (S)-5-[3-(5-methoxymethyl-1,3,4-oxadiazol-2-yl)phenyl]-9-methylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-03-2 C21H23N7O3
—— (S)-9-amino-5-[3-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092112-18-9 C19H19N7O2
—— (6aS,8R)-2-chloro-4-ethyl-8-methoxy-5-methyl-6a,7,8,9-tetrahydropyrrolo[2,1-h]pteridin-6-one 1451885-80-5 C13H17ClN4O2
—— (S)-2-{5-[3-(9-methylthio-6-oxo-2,3,3a,4-tetrahydro-1H,6H-5,8,10,10b-tetraazabenzo[e]azulen-5-yl)phenyl]-2-oxo-1,3,4-oxadiazol-3(2H)-yl}acetic acid 1092114-13-0 C21H20N6O5S