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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— 4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(4-cyclopentylpiperazin-1-yl)-3-methoxybenzamide 1157847-63-6 C33H48N8O3
—— 4-(9-cyclopentyl-7-hydroxy-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-82-2 C28H39N7O4
—— (R)-4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylpiperidin-3-yl)benzamide 1157848-16-2 C29H39N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-morpholinobenzamide 1157847-51-2 C27H37N7O4
—— (S)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-2-ylmethyl)benzamide 1157847-27-2 C26H35N7O3
—— 4-((S)-7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-pyrrolidin-3-yl)benzamide 1157848-47-9 C28H37N7O3
—— 9-cyclopentyl-5-methyl-2-(pyridin-2-ylamino)-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157848-95-7 C18H22N6O
—— 4-(9-cyclohexyl-7-cyclopropyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-06-0 C31H43N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-(2-(dimethylamino)acetyl)piperidin-4-yl)-3-methoxybenzamide 1157849-17-6 C32H46N8O4
—— N-(1-acetylazetidin-3-yl)-4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide 1137868-02-0 C27H33F2N7O4
—— (R)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-2-ylmethyl)benzamide 1157847-32-9 C27H37N7O3
—— 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-70-8 C29H39N7O3
—— 9-cyclopentyl-2-(5-fluoro-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-03-0 C20H24FN5O2
—— 2-chloro-9-cyclopentyl-7-hydroxy-7-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-44-9 C13H17ClN4O2
—— 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(2-hydroxy-ethyl)-3-methoxy-benzamide 1137208-70-8 C23H30N6O4
—— 4-((S)-7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-pyrrolidin-3-yl)benzamide 1157848-48-0 C28H37N7O3
—— 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-69-5 C31H43N7O3
—— (R)-4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-3-yl)benzamide 1157847-60-3 C28H39N7O3
—— (S)-4-(7-allyl-9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1157848-67-3 C31H43N7O3
—— 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-piperidin-3-yl)benzamide 1157848-37-7 C30H41N7O3
—— 9-cyclopentyl-2-(2-methoxy-4-(4-methylpiperazine-1-carbonyl)phenylamino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-09-6 C26H35N7O3
—— 4-(9-cyclopentyl-5,7-dimethyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-92-4 C28H37N7O3
—— 4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-23-1 C28H37N7O3
—— diethyl 2-(2-(benzylamino)-4,4-dimethyl-6-oxocyclohex-1-en-1-yl)-1H-benzo[d]imidazole-1,3(2H)-dicarboxylate 1467055-75-9 C28H33N3O5
—— (S)-4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157847-91-0 C29H41N7O3
—— 4-(9-cyclohexyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(4-methylpiperazin-1-yl)benzamide 1157847-58-9 C29H42N8O3
—— 4-((S)-7-allyl-9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-1-methylpiperidin-3-yl)benzamide 1157848-44-6 C30H41N7O3
—— 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-1-methylpiperidin-3-yl)benzamide 1157848-72-0 C31H43N7O3
—— 4-(9-cyclohexyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-1-methylpyrrolidin-3-yl)benzamide 1157848-12-8 C28H39N7O3
—— 2-chloro-9-cyclopentyl-7-methoxy-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-45-0 C15H21ClN4O2
—— 6-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)nicotinamide 1157849-02-9 C19H23N7O2
—— (R)-4-(9-cyclohexyl-7-ethyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157847-92-1 C29H41N7O3
—— 7-(tert-butyldimethylsilyloxy)-2-chloro-9-cyclopentyl-5,7-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 1157849-47-2 C20H33ClN4O2Si
—— 4-(7-allyl-9-cyclohexyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-1-methylpiperidin-3-yl)benzamide 1157848-73-1 C31H43N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methyl-piperidin-4-ylmethyl)-benzamide 1137209-35-8 C30H43N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-hydroxybenzoic acid 1157847-66-9 C22H27N5O4
—— 6-Methyl-2-phenyl-11-[2-(piperazino)propionyl]-5,6-dihydropyrimido[4,5-b][1,5]benzodiazepin-5-one 78438-58-1 C25H26N6O2
—— (S)-9-ethylamino-5-[(furan-3-yl)methyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-20-6 C17H21N5O2
—— 4-(4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamido)-N-ethylpiperidine-1-carboxamide 1157849-18-7 C31H44N8O4
—— (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-yl)benzamide 1157847-48-7 C28H39N7O3
—— (S)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-2-ylmethyl)benzamide 1157847-31-8 C27H37N7O3
—— 4-(9'-cyclohexyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[5,4-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(1-methyl-4-piperidyl)benzamide 1001345-32-9 C30H41N7O3
—— 9-cyclopentyl-5-methyl-2-phenylamino-5,7,8,9-tetrahydro-pyrimido[4,5-b][1,4]diazepin-6-one 1137207-00-1 C19H23N5O
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-(methylsulfonyl)piperidin-4-yl)benzamide 1137869-19-2 C27H35F2N7O5S
—— 4-(9-cyclopentyl-7-fluoro-5-methyl-6-oxo-7-vinyl-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((R)-piperidin-3-yl)benzamide 1137868-38-2 C28H36FN7O3
—— 5-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)picolinamide 1157849-01-8 C19H23N7O2
—— 4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-4-ylmethyl)benzamide 1157847-26-1 C27H37N7O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-(difluoromethoxy)-N-(1-methylpiperidin-4-yl)benzamide 1157847-72-7 C29H39F2N7O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-fluoro-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide 1137868-60-0 C27H34F3N7O3
—— 4-(9-cyclohexyl-7-(2-fluoroallyl)-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methylazetidin-3-yl)benzamide 1157848-78-6 C29H38FN7O3