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嘧啶二氮卓类

中文名称 英文名称 CAS号 化学式
—— (R)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-2-fluoro-5-methoxy-N-(piperidin-3-yl)benzamide 1137868-55-3 C26H32F3N7O3
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-(furan-2-ylmethyl)-3-methoxybenzamide 946825-64-5 C28H32N6O4
—— 3-(4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamido)propyl acetate 946825-92-9 C28H38N6O5
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-phenethylbenzamide 946824-99-3 C31H38N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N',N'-dimethylbenzohydrazide 1137869-04-5 C23H29F2N7O3
—— (R)-4-(9-cyclopentyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(piperidin-3-ylmethyl)benzamide 1157847-29-4 C27H37N7O3
—— N-(cyclobutylmethyl)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide 946825-62-3 C28H38N6O3
—— (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-hydroxy-3-methylbutan-2-yl)-3-methoxybenzamide 946825-55-4 C28H40N6O4
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-methoxyethyl)benzamide 946822-71-5 C24H32N6O4
—— 4-(9-cyclopentyl-7-ethyl-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946824-72-2 C24H32N6O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3,3-difluorocyclobutyl)-3-methoxybenzamide 946824-30-2 C27H34F2N6O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(cyclopropylmethyl)-3-methoxybenzamide 946823-94-5 C27H36N6O3
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6', 8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-N-isopropyl-3-methoxybenzamide 946825-79-2 C26H34N6O3
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-(1-methyl-1H-imidazol-5-yl)ethyl)benzamide 946822-88-4 C29H38N8O3
—— 3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(azetidin-3-yl)benzamide 946824-20-0 C25H33N7O2
—— 4-((S)-9-cyclopentyl-7-ethyl-6,7,8,9-tetrahydro-5-methyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclobutyl-3-methoxybenzamide 946823-83-2 C27H36N6O3
—— 4-((S)-9-cyclopentyl-6,7,8,9-tetrahydro-5,7-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclopentyl-3-methoxybenzamide 946824-37-9 C27H36N6O3
—— (S)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(1-methoxypropan-2-yl)benzamide 946825-22-5 C27H38N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((1R,3R)-3-hydroxycyclopentyl)-3-methoxybenzamide 946825-74-7 C28H38N6O4
—— 4-(9-cyclohexyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(2-(pyrrolidin-1-yl)ethyl)benzamide 1137867-90-3 C28H37F2N7O3
—— (R)-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclopropyl-3-methoxybenzamide 946824-60-8 C25H32N6O3
—— (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((1-methylpiperidin-3-yl)methyl)benzamide 1157849-25-6 C30H43N7O3
—— 4-((R)-9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((S)-tetrahydrofuran-3-yl)benzamide 946824-58-4 C26H34N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(5-methyl-1H-pyrazol-3-yl)benzamide 946825-47-4 C27H34N8O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(1-hydroxy-2-methylpropan-2-yl)-3-methoxybenzamide 946825-56-5 C27H38N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(5-methylthiazol-2-yl)benzamide 946825-52-1 C27H33N7O3S
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((2,2-difluorocyclopropyl)methyl)-3-methoxybenzamide 946825-61-2 C27H34F2N6O3
—— (S)-5-(2-chloro-5-methoxyphenyl)-9-ethylamino-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092113-10-4 C19H22ClN5O2
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-tert-butyl-3-methoxybenzamide 946823-93-4 C27H38N6O3
—— 3-(2-(pyrrolidin-1-yl)ethoxy)-4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-methylbenzamide 946823-84-3 C29H41N7O3
—— 4-(9-(3,3-difluorocyclobutyl)-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-methylbenzamide 946824-34-6 C23H28F2N6O3
—— 11-fluoro-6,7-dihydro-benzo[6,7][1,4]diazepino[2,1-<i>a</i>]quinazoline-5,13-dione 71981-85-6 C16H10FN3O2
—— 2-(3-methoxy-5-nitrophenylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946823-46-7 C22H28N6O4
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrrolidin-1-yl)benzamide 946825-05-4 C27H37N7O3
—— 9-ethylamino-5-[3-(5-methyl-[1,3,4]oxadiazol-2-yl)phenyl]-1,2,3,3a,4,5-hexahydro-5,8,10,10b-tetraazabenzo[e]azulen-6-one 1092111-65-3 C21H23N7O2
—— 1097726-80-1 C19H23FN4O5S
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(pyrimidin-4-yl)benzamide 946825-31-6 C27H32N8O3
—— 3-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(tetrahydro-2H-pyran-4-yl)benzamide 946824-05-1 C27H36N6O3
—— (R)-4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-(tetrahydrofuran-3-yl)benzamide 946824-67-5 C27H36N6O4
—— 4-(9'-cyclopentyl-5'-methyl-6'-oxo-5',6',8',9'-tetrahydrospiro[cyclopropane-1,7'-pyrimido[4,5-b][1,4]diazepine]-2'-ylamino)-3-methoxy-N-(pyridin-4-ylmethyl)benzamide 946825-63-4 C29H33N7O3
—— 2-(2-methoxyphenylamino)-5,9-dimethyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one 946824-71-1 C16H19N5O2
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(3-hydroxybutyl)-3-methoxybenzamide 946825-59-8 C27H38N6O4
—— N-(azetidin-3-yl)-4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-5-methoxybenzamide 1137868-63-3 C24H29F2N7O3
—— 5,6-dihydroquinazolino[4,3-b]quinazolin-8-one 109477-69-2 C15H11N3O
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxy-N-((tetrahydro-2H-pyran-4-yl)methyl)benzamide 946824-82-4 C29H40N6O4
—— 4-(9-cyclopentyl-6,7,8,9-tetrahydro-5,7,7-trimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclohexyl-3-methoxybenzamide 946823-96-7 C29H40N6O3
—— (R)-N-cyclopentyl-4-(9-cyclopentyl-5,7-dimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-3-methoxybenzamide 946824-62-0 C27H36N6O3
—— 4-(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-(4-cyclopentylpiperazin-1-yl)-3-methoxybenzamide 1137869-20-5 C30H40F2N8O3
—— 4-(9-cyclopentyl-5,7,7-trimethyl-6-oxo-6,7,8,9-tetrahydro-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-((1-hydroxycyclohexyl)methyl)-3-methoxy-benzamide 946825-03-2 C30H42N6O4
—— 4-((S)-9-cyclopentyl-6,7,8,9-tetrahydro-5,7-dimethyl-6-oxo-5H-pyrimido[4,5-b][1,4]diazepin-2-ylamino)-N-cyclopropyl-3-methoxybenzamide 946824-42-6 C25H32N6O3