4-Oxo-4-(pyrrolidin-1-ylamino)butanoic acid | 23744-05-0

• 分子结构分类: 有机化合物 - 脂质和类脂质分子 - 脂肪酰基
• 英文名称: 4-Oxo-4-(pyrrolidin-1-ylamino)butanoic acid
• CAS: 23744-05-0
• 化学式: C₈H₁₄N₂O₃
• 分子量: 186.21
• InChiKey: QXFBANIPKREOBY-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  -2.6
• 重原子数：
  13
• 可旋转键数：
  4
• 环数：
  1.0
• sp3杂化的碳原子比例：
  0.75
• 拓扑面积：
  69.6
• 氢给体数：
  2
• 氢受体数：
  4

文献信息

• MULTICOMPARTMENT GRANULATE FORMULATIONS FOR ACTIVE SUBSTANCES
  申请人：Letmathe Claudia

  公开号：US20090317468A1

  公开（公告）日：2009-12-24

  The invention relates to molded article that contains active substances and comprises at least two compartments that have a different material composition. Each compartment is independently provided with at least one active substance that is contained in a matrix. Each matrix encompasses at least one filler at a concentration of ≧20 percent by weight to ≦100 percent by weight relative to the total weight of the respective matrix. The invention further relates to a method for producing such molded articles as well as the use thereof.

  该发明涉及一种含有活性物质的成型制品，包括至少两个具有不同材料组成的隔间。每个隔间都独立地装有至少一种活性物质，该活性物质含在一个基质中。每个基质包含至少一种填料，其浓度相对于各自基质的总重量为≧20%至≦100%。该发明还涉及一种生产这种成型制品的方法以及其用途。
• [EN] COMPOUNDS HAVING PROLYL OLIGOPEPTIDASE INHIBITORY ACTIVITY, METHODS FOR THEIR PREPARATION AND THEIR USE<br/>[FR] COMPOSES INHIBITEURS DE LA PROLYL OLIGOPEPTIDASE, PROCEDES DE PREPARATION ET UTILISATION
  申请人：ORION CORP

  公开号：WO2003004468A1

  公开（公告）日：2003-01-16

  Compounds of the formula (I), wherein the symbol aa means a residue of an α-amino acid. The invention is also directed to a method for the preparation of the compounds of formula (I), as well as their use as prolyl oligopeptide inhibitors, for example for the treatment of Alzheimer's disease.

  公式（I）的化合物，其中符号aa表示α-氨基酸的残基。本发明还涉及一种制备公式（I）化合物的方法，以及它们作为脯氨酰寡肽抑制剂的用途，例如用于治疗阿尔茨海默病。
• Compounds having prolyl oligopeptidase inhibitory activity, methods for their preparation and their use
  申请人：Gynther Jukka

  公开号：US20050020677A1

  公开（公告）日：2005-01-27

  Compounds of the formula (I), wherein the symbol aa means a residue of an α-amino acid. The invention is also directed to a method for the preparation of the compounds of formula (I), as well as their use as prolyl oligopeptide inhibitors, for example for the treatment of Alzheimer's disease.

  式(I)的化合物，其中符号aa表示α-氨基酸残基。本发明还涉及一种制备式(I)化合物的方法，以及它们作为脯氨酰寡肽酶抑制剂的用途，例如用于治疗阿尔茨海默病。
• Cyanbenzofuran derivatives, processes for their preparation and their use in herbicidal compositions; cyanobenzene, benzodioxepine, benzodioxaphosphepine and benzodioxathiepine derivatives
  申请人：FBC LIMITED

  公开号：EP0007719A2

  公开（公告）日：1980-02-06

  The invention provides herbicidally-active 2,3-dihydro-5-cyano-benzofurans of the formula: (wherein: R' and R2 together represent =O or R' represents hydrogen and R2 represents hydrogen, hydroxy, alkoxy, acyloxy, alkoxycarbonyloxy, alkylthiocarbonyloxy, halogen, isothiocyanato, amino, alkylamino, dialkylamino, arylamino, acylamino, alkoxycarbonylamino, alkyhhiocarbonylamino. N-bonded heterocyclyl, cyano or alkylthio; R3 and R4 together represent alkylene or each represent hydrogen or alkyl; and R5, R6 and R7, which may be the same or different, each represent hydrogen, halogen, alkyl, alkoxy, acyl or cyano), processes for their preparation and herbicidal compositions containing them.

  本发明提供了具有除草活性的 2,3-二氢-5-氰基苯并呋喃，其化学式为 其中R'和R2一起代表＝O或R'代表氢，R2代表氢、羟基、烷氧基、酰氧基、烷氧基羰氧基、烷硫基羰氧基、卤素、异硫氰基、氨基、烷基氨基、二烷基氨基、芳基氨基、酰氨基、烷氧基羰基氨基、烷硫基羰基氨基。R3和R4共同代表亚烷基或各自代表氢或烷基；R5、R6和R7可以相同或不同，各自代表氢、卤素、烷基、烷氧基、酰基或氰基），以及它们的制备方法和含有它们的除草组合物。
• Pesticidal compositions
  申请人：SYNGENTA PARTICIPATIONS AG

  公开号：US10674728B2

  公开（公告）日：2020-06-09

  The present invention relates to pesticidal compositions. In particular it relates to composition comprising a compound of formula (I) and a further active ingredient. Such compositions are useful for the control of pests and/or for improving the yield of crop plants.

  本发明涉及杀虫剂组合物。特别是涉及由式（I）化合物和另一种活性成分组成的组合物。这种组合物可用于防治害虫和/或提高作物产量。