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—— (E)-3-[4-[[1-[[1-[(2S,6S)-2,6-dimethylcyclohexyl]-2-(2-furyl)benzimidazole-5-carbonyl]amino]cyclopentanecarbonyl]amino]phenyl]prop-2-enoic acid —— C35H38N4O5
(E)-3-[4-[[1-[[1-[(2S,6S)-2,6-dimethylcyclohexyl]-2-(2-furyl)benzimidazole-5-carbonyl]amino]cyclopentanecarbonyl]amino]phenyl]prop-2-enoic acid
—— (E)-N-{5-[(cyclohexylmethyl)amino]-1,3,4-thiadiazol-2-yl}-3-phenyl-2-propenamide —— C18H22N4OS
(E)-N-{5-[(cyclohexylmethyl)amino]-1,3,4-thiadiazol-2-yl}-3-phenyl-2-propenamide
—— (E)-N-[(1S)-1-[[3-(2,4-dinitrophenyl)imidazol-4-yl]methyl]-2-[2-(2-hydroxybenzoyl)hydrazino]-2-oxo-ethyl]-3-(3-thioxocyclohexa-1,5-dien-1-yl)prop-2-enamide —— C28H23N7O8S
(E)-N-[(1S)-1-[[3-(2,4-dinitrophenyl)imidazol-4-yl]methyl]-2-[2-(2-hydroxybenzoyl)hydrazino]-2-oxo-ethyl]-3-(3-thioxocyclohexa-1,5-dien-1-yl)prop-2-enamide
—— ethyl 4-bromo-2-methylquinoline-6-carboxylate —— C13H12BrNO2
ethyl 4-bromo-2-methylquinoline-6-carboxylate
—— (E)-N-[5-[(4-chlorophenyl)sulfamoyl]-1-naphthyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide —— C25H19ClN2O5S
(E)-N-[5-[(4-chlorophenyl)sulfamoyl]-1-naphthyl]-3-(3,4-dihydroxyphenyl)prop-2-enamide
—— ethyl (E,4S)-7-amino-4-[[(2R)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-ethylsulfanyl-propanoyl]amino]-7-oxo-hept-2-enoate —— C28H42N4O7S
ethyl (E,4S)-7-amino-4-[[(2R)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]-3-ethylsulfanyl-propanoyl]amino]-7-oxo-hept-2-enoate
—— ethyl (2S)-2-[(S)-[(4R)-3-methyl-5-oxo-1-phenyl-4H-pyrazol-4-yl]-phenylmethyl]-3-oxobutanoate —— C23H24N2O4
ethyl (2S)-2-[(S)-[(4R)-3-methyl-5-oxo-1-phenyl-4H-pyrazol-4-yl]-phenylmethyl]-3-oxobutanoate
—— (E)-3-(2-chlorophenyl)-N-[5-(neopentylamino)-1,3,4-thiadiazol-2-yl]-2-propenamide —— C16H19ClN4OS
(E)-3-(2-chlorophenyl)-N-[5-(neopentylamino)-1,3,4-thiadiazol-2-yl]-2-propenamide
—— (E)-N-(5-{[4-(aminosulfonyl)phenethyl]amino}-1,3,4-thiadiazol-2-yl)-3-(2-chlorophenyl)-2-propenamide —— C19H18ClN5O3S2
(E)-N-(5-{[4-(aminosulfonyl)phenethyl]amino}-1,3,4-thiadiazol-2-yl)-3-(2-chlorophenyl)-2-propenamide
—— Ethyl 4-((5-(2-hydroxy-3-methoxybenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)methylene)-5-oxo-1-phenyl-4,5-dihydro-1H-pyrazole-3-carboxylate —— C24H19N3O6S2
Ethyl 4-((5-(2-hydroxy-3-methoxybenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)methylene)-5-oxo-1-phenyl-4,5-dihydro-1H-pyrazole-3-carboxylate
—— (E)-3-(3,4-dihydroxyphenyl)prop-2-enoic acid; 3,4,5-trihydroxybenzoic acid —— C16H14O9
(E)-3-(3,4-dihydroxyphenyl)prop-2-enoic acid; 3,4,5-trihydroxybenzoic acid
—— (E)-3-{3-[2-((S)-4,4-Difluoro-2-{[(2S,4S)-1-((S)-2-isobutoxycarbonylamino-3-methyl-butyryl)-4-phenyl-pyrrolidine-2-carbonyl]-amino}-butyrylamino)-ethyl]-4-fluoro-phenyl}-acrylic acid —— C36H45F3N4O7
(E)-3-{3-[2-((S)-4,4-Difluoro-2-{[(2S,4S)-1-((S)-2-isobutoxycarbonylamino-3-methyl-butyryl)-4-phenyl-pyrrolidine-2-carbonyl]-amino}-butyrylamino)-ethyl]-4-fluoro-phenyl}-acrylic acid
—— (E)-N-{5-[(1,3-benzodioxol-5-ylmethyl)amino]-1,3,4-thiadiazol-2-yl}-9-octadecenamide —— C28H42N4O3S
(E)-N-{5-[(1,3-benzodioxol-5-ylmethyl)amino]-1,3,4-thiadiazol-2-yl}-9-octadecenamide
—— (E)-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-[(3,4-dihydroxyphenyl)methyl]-2-[2-(2-hydroxybenzoyl)hydrazino]-2-oxo-ethyl]prop-2-enamide —— C25H23N3O8
(E)-3-(3,4-dihydroxyphenyl)-N-[(1S)-1-[(3,4-dihydroxyphenyl)methyl]-2-[2-(2-hydroxybenzoyl)hydrazino]-2-oxo-ethyl]prop-2-enamide
—— (E)-3-(2,6-Dimethoxy-phenyl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide —— C20H20N2O5S
(E)-3-(2,6-Dimethoxy-phenyl)-N-[(S)-1-(5-methyl-4-oxo-4H-thieno[2,3-d][1,3]oxazin-2-yl)-ethyl]-acrylamide
—— ethyl (4R)-4-pyridin-2-yl-4,5-dihydro-1H-pyrazole-3-carboxylate —— C11H13N3O2
ethyl (4R)-4-pyridin-2-yl-4,5-dihydro-1H-pyrazole-3-carboxylate
—— (E)-1-[(1S,2S)-2-[(S)-hydroxy-[(2R)-6-oxo-2,3-dihydropyran-2-yl]methyl]cyclopropyl]-6-(4-methoxyphenyl)-2-methyl-hex-5-ene-1,4-dione —— C23H26O6
(E)-1-[(1S,2S)-2-[(S)-hydroxy-[(2R)-6-oxo-2,3-dihydropyran-2-yl]methyl]cyclopropyl]-6-(4-methoxyphenyl)-2-methyl-hex-5-ene-1,4-dione
—— (E)-3-(2-chlorophenyl)-N-[5-(cyclobutylamino)-1,3,4-thiadiazol-2-yl]-2-propenamide —— C15H15ClN4OS
(E)-3-(2-chlorophenyl)-N-[5-(cyclobutylamino)-1,3,4-thiadiazol-2-yl]-2-propenamide
—— (E)-3-(2-chlorophenyl)-N-{5-[(2,2-diphenylethyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide —— C25H21ClN4OS
(E)-3-(2-chlorophenyl)-N-{5-[(2,2-diphenylethyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide
—— ethyl (2S)-2,4-dimethyl-3H-pyrido[3,2-b][1,4]oxazine-2-carboxylate —— C12H16N2O3
ethyl (2S)-2,4-dimethyl-3H-pyrido[3,2-b][1,4]oxazine-2-carboxylate
—— (E)-3-(3,4-dihydroxyphenyl)-N-[5-[(3-nitrophenyl)sulfamoyl]-1-naphthyl]prop-2-enamide —— C25H19N3O7S
(E)-3-(3,4-dihydroxyphenyl)-N-[5-[(3-nitrophenyl)sulfamoyl]-1-naphthyl]prop-2-enamide
—— (E)-3-(2-chlorophenyl)-N-[(3Z)-1-hydroxy-3-[hydroxy(phenyl)methylene]-2-oxo-indolin-6-yl]prop-2-enamide —— C24H17ClN2O4
(E)-3-(2-chlorophenyl)-N-[(3Z)-1-hydroxy-3-[hydroxy(phenyl)methylene]-2-oxo-indolin-6-yl]prop-2-enamide
—— Ethyl 3-(4-(bis(2-cyanoethyl)amino)-2-methylphenyl)-2-(cinnamoylamino)acrylate —— C27H28N4O3
Ethyl 3-(4-(bis(2-cyanoethyl)amino)-2-methylphenyl)-2-(cinnamoylamino)acrylate
—— (E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-isobutyrylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester —— C28H42N4O6
(E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-isobutyrylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester
—— (E)-N-(5-{[2-(1-methyl-2-pyrrolidinyl)ethyl]amino}-1,3,4-thiadiazol-2-yl)-9-octadecenamide —— C27H49N5OS
(E)-N-(5-{[2-(1-methyl-2-pyrrolidinyl)ethyl]amino}-1,3,4-thiadiazol-2-yl)-9-octadecenamide
—— ethyl (3S,4R)-1-[(2-chlorophenyl)methyl]-4-(2-cyanophenyl)pyrrolidine-3-carboxylate —— C21H21ClN2O2
ethyl (3S,4R)-1-[(2-chlorophenyl)methyl]-4-(2-cyanophenyl)pyrrolidine-3-carboxylate
—— (E)-N-{5-[(3-pyridinylmethyl)amino]-1,3,4-thiadiazol-2-yl}-9-octadecenamide —— C26H41N5OS
(E)-N-{5-[(3-pyridinylmethyl)amino]-1,3,4-thiadiazol-2-yl}-9-octadecenamide
—— ethyl (3R)-1-[2-(4-fluorophenyl)ethyl]-2,4-dioxopiperidine-3-carboxylate —— C16H18FNO4
ethyl (3R)-1-[2-(4-fluorophenyl)ethyl]-2,4-dioxopiperidine-3-carboxylate
—— ethyl (E,4S)-4-[[(2S)-3-(4-acetoxyphenyl)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]propanoyl]amino]-7-amino-7-oxo-hept-2-enoate —— C34H44N4O9
ethyl (E,4S)-4-[[(2S)-3-(4-acetoxyphenyl)-2-[[(2S)-2-(benzyloxycarbonylamino)-4-methyl-pentanoyl]amino]propanoyl]amino]-7-amino-7-oxo-hept-2-enoate
—— ethyl (4aS)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate —— C21H27NO5
ethyl (4aS)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate
—— (E)-3-phenyl-N-{5-[(4-phenylbutyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide —— C21H22N4OS
(E)-3-phenyl-N-{5-[(4-phenylbutyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide
—— ethyl (4aR)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate —— C21H27NO5
ethyl (4aR)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate
—— (E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-cyclohexyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester —— C31H46N4O7
(E)-(S)-6-Carbamoyl-4-[(S)-2-((S)-2-cyclohexyloxycarbonylamino-4-methyl-pentanoylamino)-3-phenyl-propionylamino]-hex-2-enoic acid ethyl ester
—— ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-4-methyl-2-(4-pyridylmethoxycarbonylamino)pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate —— C31H41N5O7
ethyl (E,4S)-7-amino-4-[[(2S)-2-[[(2S)-4-methyl-2-(4-pyridylmethoxycarbonylamino)pentanoyl]amino]-3-phenyl-propanoyl]amino]-7-oxo-hept-2-enoate
—— (E)-N-{5-[(2-anilinoethyl)amino]-1,3,4-thiadiazol-2-yl}-3-(2-chlorophenyl)-2-propenamide —— C19H18ClN5OS
(E)-N-{5-[(2-anilinoethyl)amino]-1,3,4-thiadiazol-2-yl}-3-(2-chlorophenyl)-2-propenamide
—— (E)-3-(2-chlorophenyl)-N-{5-[(1-naphthylmethyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide —— C22H17ClN4OS
(E)-3-(2-chlorophenyl)-N-{5-[(1-naphthylmethyl)amino]-1,3,4-thiadiazol-2-yl}-2-propenamide
—— (E)-N-(5-{[3-(cyclohexylamino)propyl]amino}-1,3,4-thiadiazol-2-yl)-3-phenyl-2-propenamide —— C20H27N5OS
(E)-N-(5-{[3-(cyclohexylamino)propyl]amino}-1,3,4-thiadiazol-2-yl)-3-phenyl-2-propenamide
—— ethyl (3S)-1-[2-(4-fluorophenyl)ethyl]-2,4-dioxopiperidine-3-carboxylate —— C16H18FNO4
ethyl (3S)-1-[2-(4-fluorophenyl)ethyl]-2,4-dioxopiperidine-3-carboxylate
—— (E)-(S)-4-((2R,5S)-2-Benzyl-5-benzylsulfanylcarbonylamino-6-methyl-4-oxo-heptanoylamino)-6-carbamoyl-hex-2-enoic acid ethyl ester —— C32H41N3O6S
(E)-(S)-4-((2R,5S)-2-Benzyl-5-benzylsulfanylcarbonylamino-6-methyl-4-oxo-heptanoylamino)-6-carbamoyl-hex-2-enoic acid ethyl ester
—— ethyl (4aR)-2-oxo-1-piperidin-4-yl-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate —— C17H26N2O3
ethyl (4aR)-2-oxo-1-piperidin-4-yl-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate
—— ethyl (3R,4R)-4-aminooxolane-3-carboxylate —— C7H13NO3
ethyl (3R,4R)-4-aminooxolane-3-carboxylate
—— ethyl (4S)-4-pyridin-2-yl-4,5-dihydro-1H-pyrazole-3-carboxylate —— C11H13N3O2
ethyl (4S)-4-pyridin-2-yl-4,5-dihydro-1H-pyrazole-3-carboxylate
—— ethyl (4aS)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-3,4,5,6-tetrahydrocyclopenta[b]pyridine-4a-carboxylate —— C20H25NO5
ethyl (4aS)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-3,4,5,6-tetrahydrocyclopenta[b]pyridine-4a-carboxylate
—— Ethyl 1-[(4-chlorophenyl)methyl]-4-sulfanylidenequinoline-3-carboxylate —— C19H16ClNO2S
Ethyl 1-[(4-chlorophenyl)methyl]-4-sulfanylidenequinoline-3-carboxylate
—— ethyl (3S,4S)-1-[(2-chlorophenyl)methyl]-4-(2-cyanophenyl)pyrrolidine-3-carboxylate —— C21H21ClN2O2
ethyl (3S,4S)-1-[(2-chlorophenyl)methyl]-4-(2-cyanophenyl)pyrrolidine-3-carboxylate
—— ethyl (2R)-2,4-dimethyl-3H-pyrido[3,2-b][1,4]oxazine-2-carboxylate —— C12H16N2O3
ethyl (2R)-2,4-dimethyl-3H-pyrido[3,2-b][1,4]oxazine-2-carboxylate
—— ethyl (2E)-2-[(3-chlorophenyl)methylene]-3-oxo-butanoate —— C13H13ClO3
ethyl (2E)-2-[(3-chlorophenyl)methylene]-3-oxo-butanoate
—— ethyl (4aS)-2-oxo-1-piperidin-4-yl-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate —— C17H26N2O3
ethyl (4aS)-2-oxo-1-piperidin-4-yl-4,5,6,7-tetrahydro-3H-quinoline-4a-carboxylate
—— ethyl (4aR)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-3,4,5,6-tetrahydrocyclopenta[b]pyridine-4a-carboxylate —— C20H25NO5
ethyl (4aR)-1-[(3,4-dimethoxyphenyl)methyl]-2-oxo-3,4,5,6-tetrahydrocyclopenta[b]pyridine-4a-carboxylate
—— ethyl (E)-2-(diethylamino)-3-(3-methoxyphenyl)prop-2-enoate —— C16H23NO3
ethyl (E)-2-(diethylamino)-3-(3-methoxyphenyl)prop-2-enoate