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—— (E)-3-(5-bromofuran-2-yl)-N-[(2S,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide —— C12H16BrNO3S
(E)-3-(5-bromofuran-2-yl)-N-[(2S,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide
—— (E)-3-(5-chlorothiophen-2-yl)-N-[(2S,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide —— C12H16ClNO2S2
(E)-3-(5-chlorothiophen-2-yl)-N-[(2S,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide
—— (E)-N-[(2R,3R)-4-hydroxy-3-methylsulfanylbutan-2-yl]-3-quinolin-2-ylprop-2-enamide —— C17H20N2O2S
(E)-N-[(2R,3R)-4-hydroxy-3-methylsulfanylbutan-2-yl]-3-quinolin-2-ylprop-2-enamide
—— (E)-3-(2-cyanophenyl)-N-[(2S,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide —— C15H18N2O2S
(E)-3-(2-cyanophenyl)-N-[(2S,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide
—— (E)-3-(5-chlorothiophen-2-yl)-N-[(2R,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide —— C12H16ClNO2S2
(E)-3-(5-chlorothiophen-2-yl)-N-[(2R,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide
—— (E)-N-[(2R,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]-3-(2-methyl-1,3-thiazol-5-yl)prop-2-enamide —— C12H18N2O2S2
(E)-N-[(2R,3S)-4-hydroxy-3-methylsulfanylbutan-2-yl]-3-(2-methyl-1,3-thiazol-5-yl)prop-2-enamide
—— (E)-3-(2-cyanophenyl)-N-[(2S,3R)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide —— C15H18N2O2S
(E)-3-(2-cyanophenyl)-N-[(2S,3R)-4-hydroxy-3-methylsulfanylbutan-2-yl]prop-2-enamide
—— Ethyl 4-methyl-2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]quinoline-3-carboxylate —— C19H22N4O2S
Ethyl 4-methyl-2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]quinoline-3-carboxylate
—— Ethyl 2-[[2-[[2-(4-methylphenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]amino]-2-oxoacetyl]amino]acetate —— C18H20N4O4S
Ethyl 2-[[2-[[2-(4-methylphenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]amino]-2-oxoacetyl]amino]acetate
—— (E)-N-[[(3S,9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]oxazin-3-yl]methyl]-3-cyclopropylbut-2-enamide —— C16H26N2O2
(E)-N-[[(3S,9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]oxazin-3-yl]methyl]-3-cyclopropylbut-2-enamide
—— (E)-N-[[(3R,9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]oxazin-3-yl]methyl]-3-cyclopropylbut-2-enamide —— C16H26N2O2
(E)-N-[[(3R,9aR)-1,3,4,6,7,8,9,9a-octahydropyrido[2,1-c][1,4]oxazin-3-yl]methyl]-3-cyclopropylbut-2-enamide
—— Ethyl 5-ethyl-4-methyl-2-[[2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]thiophene-3-carboxylate —— C17H24N4O3S2
Ethyl 5-ethyl-4-methyl-2-[[2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]thiophene-3-carboxylate
—— ethyl (3S)-4-[[5-(difluoromethylsulfanylmethyl)furan-2-carbonyl]amino]-3-methylbutanoate —— C14H19F2NO4S
ethyl (3S)-4-[[5-(difluoromethylsulfanylmethyl)furan-2-carbonyl]amino]-3-methylbutanoate
—— Ethyl 4-cyclopropyl-2-[[2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]thiophene-3-carboxylate —— C17H22N4O3S2
Ethyl 4-cyclopropyl-2-[[2-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanyl]acetyl]amino]thiophene-3-carboxylate
—— ethyl (3R)-4-[[4-(cyclopropylamino)-5-nitropyrimidin-2-yl]amino]-3-methylbutanoate —— C14H21N5O4
ethyl (3R)-4-[[4-(cyclopropylamino)-5-nitropyrimidin-2-yl]amino]-3-methylbutanoate
—— ethyl (3R)-4-[[5-(difluoromethylsulfanylmethyl)furan-2-carbonyl]amino]-3-methylbutanoate —— C14H19F2NO4S
ethyl (3R)-4-[[5-(difluoromethylsulfanylmethyl)furan-2-carbonyl]amino]-3-methylbutanoate
—— ethyl (4S)-4-[[3-[(6-methylimidazo[1,2-a]pyridin-2-yl)methoxy]benzoyl]amino]pentanoate —— C23H27N3O4
ethyl (4S)-4-[[3-[(6-methylimidazo[1,2-a]pyridin-2-yl)methoxy]benzoyl]amino]pentanoate
—— (E)-2-cyano-3-(2-fluorophenyl)-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide —— C17H19FN2O
(E)-2-cyano-3-(2-fluorophenyl)-N-[(1R,2S)-2-methylcyclohexyl]prop-2-enamide
—— (E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide —— C17H21N3O3
(E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide
—— (E)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-propan-2-ylphenyl)prop-2-en-1-one —— C20H20O3
(E)-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(4-propan-2-ylphenyl)prop-2-en-1-one
—— (E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide —— C17H21N3O3
(E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1S,2R)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide
—— Ethyl 2-[[2-(3-chloro-2-methylanilino)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C20H23ClN2O3S
Ethyl 2-[[2-(3-chloro-2-methylanilino)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (2S)-2-[5-(4-methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoate —— C18H18N2O3S2
ethyl (2S)-2-[5-(4-methoxyphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoate
—— ethyl (3S)-4-[[4-(cyclopropylamino)-5-nitropyrimidin-2-yl]amino]-3-methylbutanoate —— C14H21N5O4
ethyl (3S)-4-[[4-(cyclopropylamino)-5-nitropyrimidin-2-yl]amino]-3-methylbutanoate
—— Ethyl 3-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-1-benzofuran-2-carboxylate —— C17H19N3O3S
Ethyl 3-[(4-propan-2-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-1-benzofuran-2-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-1-[(2R,5S)-5-(hydroxymethyl)-2-methylpiperidin-1-yl]prop-2-en-1-one —— C17H21NO4
(E)-3-(1,3-benzodioxol-5-yl)-1-[(2R,5S)-5-(hydroxymethyl)-2-methylpiperidin-1-yl]prop-2-en-1-one
—— ethyl 4-[2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C20H23N5O3S
ethyl 4-[2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-3-(5-bromo-2-fluorophenyl)-N-[(1S)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]prop-2-enamide —— C15H15BrFN3O2
(E)-3-(5-bromo-2-fluorophenyl)-N-[(1S)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]prop-2-enamide
—— ethyl (4S)-4-[[5-chloro-1-(4-chlorophenyl)-6-oxopyridazin-4-yl]amino]pentanoate —— C17H19Cl2N3O3
ethyl (4S)-4-[[5-chloro-1-(4-chlorophenyl)-6-oxopyridazin-4-yl]amino]pentanoate
—— Ethyl 2-[[2-(dibutylamino)acetyl]amino]-5-phenylthiophene-3-carboxylate —— C23H32N2O3S
Ethyl 2-[[2-(dibutylamino)acetyl]amino]-5-phenylthiophene-3-carboxylate
—— ethyl (3S)-4-(1,3-benzothiazol-2-ylamino)-3-methylbutanoate —— C14H18N2O2S
ethyl (3S)-4-(1,3-benzothiazol-2-ylamino)-3-methylbutanoate
—— ethyl (4R)-4-[[3-[(6-methylimidazo[1,2-a]pyridin-2-yl)methoxy]benzoyl]amino]pentanoate —— C23H27N3O4
ethyl (4R)-4-[[3-[(6-methylimidazo[1,2-a]pyridin-2-yl)methoxy]benzoyl]amino]pentanoate
—— Ethyl 2-[[2-[bis(2-methoxyethyl)amino]acetyl]amino]-4-phenylthiophene-3-carboxylate —— C21H28N2O5S
Ethyl 2-[[2-[bis(2-methoxyethyl)amino]acetyl]amino]-4-phenylthiophene-3-carboxylate
—— ethyl (3R)-4-(1,3-benzothiazol-2-ylamino)-3-methylbutanoate —— C14H18N2O2S
ethyl (3R)-4-(1,3-benzothiazol-2-ylamino)-3-methylbutanoate
—— (E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide —— C17H21N3O3
(E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide
—— Ethyl 2-[[2-[methyl-(1-methylpiperidin-4-yl)amino]acetyl]amino]-4-phenylthiophene-3-carboxylate —— C22H29N3O3S
Ethyl 2-[[2-[methyl-(1-methylpiperidin-4-yl)amino]acetyl]amino]-4-phenylthiophene-3-carboxylate
—— Ethyl 2-[[2-[[2-(4-fluorophenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]amino]-2-oxoacetyl]amino]acetate —— C17H17FN4O4S
Ethyl 2-[[2-[[2-(4-fluorophenyl)-4,6-dihydrothieno[3,4-c]pyrazol-3-yl]amino]-2-oxoacetyl]amino]acetate
—— (E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide —— C17H21N3O3
(E)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]-3-[5-[(1S,2S)-2-methylcyclopropyl]furan-2-yl]prop-2-enamide
—— ethyl (4R)-4-[[5-chloro-1-(4-chlorophenyl)-6-oxopyridazin-4-yl]amino]pentanoate —— C17H19Cl2N3O3
ethyl (4R)-4-[[5-chloro-1-(4-chlorophenyl)-6-oxopyridazin-4-yl]amino]pentanoate
—— ethyl (3S)-1-[2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]piperidine-3-carboxylate —— C19H25N5O3S
ethyl (3S)-1-[2-[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylacetyl]piperidine-3-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-1-[(2R,5R)-5-(hydroxymethyl)-2-methylpiperidin-1-yl]prop-2-en-1-one —— C17H21NO4
(E)-3-(1,3-benzodioxol-5-yl)-1-[(2R,5R)-5-(hydroxymethyl)-2-methylpiperidin-1-yl]prop-2-en-1-one
—— (E)-3-(5-bromo-2-fluorophenyl)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]prop-2-enamide —— C15H15BrFN3O2
(E)-3-(5-bromo-2-fluorophenyl)-N-[(1R)-2-hydroxy-1-(1-methylpyrazol-4-yl)ethyl]prop-2-enamide
—— Ethyl 2-[[2-(3-chloro-4-methylanilino)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C20H23ClN2O3S
Ethyl 2-[[2-(3-chloro-4-methylanilino)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 1-[4-[(2R)-2-(3-hydroxypropyl)pyrrolidine-1-carbonyl]phenyl]-5-methylpyrazole-4-carboxylate —— C21H27N3O4
ethyl 1-[4-[(2R)-2-(3-hydroxypropyl)pyrrolidine-1-carbonyl]phenyl]-5-methylpyrazole-4-carboxylate
—— Ethyl 2-(3-(p-tolylthio)propanamido)benzo[b]thiophene-3-carboxylate —— C21H21NO3S2
Ethyl 2-(3-(p-tolylthio)propanamido)benzo[b]thiophene-3-carboxylate
—— Ethyl 2-(4-(ethylsulfonyl)benzamido)benzo[b]thiophene-3-carboxylate —— C20H19NO5S2
Ethyl 2-(4-(ethylsulfonyl)benzamido)benzo[b]thiophene-3-carboxylate
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-[(1S)-1-(3-fluorophenyl)-2-hydroxyethyl]-N-methylprop-2-enamide —— C19H19F2NO3
(E)-3-(3-fluoro-4-methoxyphenyl)-N-[(1S)-1-(3-fluorophenyl)-2-hydroxyethyl]-N-methylprop-2-enamide
—— ethyl (4R)-6-[[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C19H24N6O3S
ethyl (4R)-6-[[1-(2,4-dimethylphenyl)tetrazol-5-yl]sulfanylmethyl]-4-ethyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (6R)-2-[[2-(4-chloro-2-methylanilino)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H25ClN2O3S
ethyl (6R)-2-[[2-(4-chloro-2-methylanilino)acetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-[[2-[cyclohexyl(methyl)amino]acetyl]amino]-4-(4-methylphenyl)thiophene-3-carboxylate —— C23H30N2O3S
Ethyl 2-[[2-[cyclohexyl(methyl)amino]acetyl]amino]-4-(4-methylphenyl)thiophene-3-carboxylate