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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6aS,7S)-7-[4-(trifluoromethyl)phenyl]-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine —— C24H18F3NS
(6aS,7S)-7-[4-(trifluoromethyl)phenyl]-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine
—— (6aS,7S)-7-thiophen-2-yl-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine —— C21H17NS2
(6aS,7S)-7-thiophen-2-yl-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine
—— 6-[[(3S)-1-(6-methylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C16H17N7S
6-[[(3S)-1-(6-methylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-morpholin-4-yl-N-phenylpyridin-1-ium-3-carboxamide —— C16H18N3O2+
6-morpholin-4-yl-N-phenylpyridin-1-ium-3-carboxamide
—— (6aS,7S)-3-methoxy-7-(4-methylphenyl)-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine —— C25H23NOS
(6aS,7S)-3-methoxy-7-(4-methylphenyl)-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine
—— (6aS,7R)-7-[4-(trifluoromethyl)phenyl]-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine —— C24H18F3NS
(6aS,7R)-7-[4-(trifluoromethyl)phenyl]-5,6,6a,7-tetrahydronaphtho[2,1-c][1,5]benzothiazepine
—— (6aS,7R)-7-[4-(trifluoromethyl)phenyl]-6a,7-dihydro-6H-chromeno[3,4-c][1,5]benzothiazepine —— C23H16F3NOS
(6aS,7R)-7-[4-(trifluoromethyl)phenyl]-6a,7-dihydro-6H-chromeno[3,4-c][1,5]benzothiazepine
—— 6-[[(3R)-1-(1,3-benzoxazol-2-ylmethyl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C19H19N5O
6-[[(3R)-1-(1,3-benzoxazol-2-ylmethyl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— (6aS,7S)-7-[4-(trifluoromethyl)phenyl]-6a,7-dihydro-6H-chromeno[3,4-c][1,5]benzothiazepine —— C23H16F3NOS
(6aS,7S)-7-[4-(trifluoromethyl)phenyl]-6a,7-dihydro-6H-chromeno[3,4-c][1,5]benzothiazepine
—— 6-ethoxy-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-2H-chromene-3-carboxamide —— C19H21N3O3
6-ethoxy-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-2H-chromene-3-carboxamide
—— 6-[[(3R)-1-(3-morpholin-4-yl-3-oxopropyl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C18H25N5O2
6-[[(3R)-1-(3-morpholin-4-yl-3-oxopropyl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— (6S)-6-methyl-N-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-6,7,8,9-tetrahydro-5H-carbazole-1-carboxamide —— C19H20N4O2S
(6S)-6-methyl-N-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-6,7,8,9-tetrahydro-5H-carbazole-1-carboxamide
—— 6-[[(3S)-1-(3-morpholin-4-yl-3-oxopropyl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C18H25N5O2
6-[[(3S)-1-(3-morpholin-4-yl-3-oxopropyl)pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-(dimethylamino)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide —— C15H19N5O
6-(dimethylamino)-N-[(6R)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide
—— 6-ethoxy-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-2H-chromene-3-carboxamide —— C19H21N3O3
6-ethoxy-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]-2H-chromene-3-carboxamide
—— (6R)-6-methyl-N-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-6,7,8,9-tetrahydro-5H-carbazole-1-carboxamide —— C19H20N4O2S
(6R)-6-methyl-N-[2-oxo-2-(1,3-thiazol-2-ylamino)ethyl]-6,7,8,9-tetrahydro-5H-carbazole-1-carboxamide
—— 6-[(1R)-1-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]pyridine-3-carboxamide —— C19H18N4O2
6-[(1R)-1-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]pyridine-3-carboxamide
—— 6-[(1S)-1-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]pyridine-3-carboxamide —— C19H18N4O2
6-[(1S)-1-methyl-1,3,4,9-tetrahydropyrido[3,4-b]indole-2-carbonyl]pyridine-3-carboxamide
—— 6-(dimethylamino)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide —— C15H19N5O
6-(dimethylamino)-N-[(6S)-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-yl]pyridine-3-carboxamide
—— 6-[[(3R)-1-[2-[(2S)-2-methylmorpholin-4-yl]-2-oxoethyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C18H25N5O2
6-[[(3R)-1-[2-[(2S)-2-methylmorpholin-4-yl]-2-oxoethyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-oxo-N-[(2S)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4,5-dihydro-1H-pyridazine-3-carboxamide —— C15H20N4O2S
6-oxo-N-[(2S)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4,5-dihydro-1H-pyridazine-3-carboxamide
—— (6-Chloro-3-ethyl-7-hydroxy-4-methyl-2-oxochromen-8-yl)methyl-diethylazanium —— C17H23ClNO3+
(6-Chloro-3-ethyl-7-hydroxy-4-methyl-2-oxochromen-8-yl)methyl-diethylazanium
—— 6-[[(3R)-1-[2-[(2R)-2-methylmorpholin-4-yl]-2-oxoethyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C18H25N5O2
6-[[(3R)-1-[2-[(2R)-2-methylmorpholin-4-yl]-2-oxoethyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-methyl-4-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C16H23N7
6-methyl-4-[(3R)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[1-[2-[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]hydrazinyl]ethylidene]cyclohexa-2,4-dien-1-one —— C18H16FN3OS
6-[1-[2-[4-(4-fluoro-3-methylphenyl)-1,3-thiazol-2-yl]hydrazinyl]ethylidene]cyclohexa-2,4-dien-1-one
—— 6-[4-[(2R)-2-(2,2,2-trifluoroethoxy)propanoyl]piperazin-1-yl]pyridine-3-carbonitrile —— C15H17F3N4O2
6-[4-[(2R)-2-(2,2,2-trifluoroethoxy)propanoyl]piperazin-1-yl]pyridine-3-carbonitrile
—— 6-[4-[(2S)-2-(2,2,2-trifluoroethoxy)propanoyl]piperazin-1-yl]pyridine-3-carbonitrile —— C15H17F3N4O2
6-[4-[(2S)-2-(2,2,2-trifluoroethoxy)propanoyl]piperazin-1-yl]pyridine-3-carbonitrile
—— 6-oxo-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4,5-dihydro-1H-pyridazine-3-carboxamide —— C15H20N4O2S
6-oxo-N-[(2R)-2-pyrrolidin-1-yl-2-thiophen-2-ylethyl]-4,5-dihydro-1H-pyridazine-3-carboxamide
—— (6S)-N-[[5-(dimethylamino)-1,3-dimethylpyrazol-4-yl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-amine —— C15H24N6
(6S)-N-[[5-(dimethylamino)-1,3-dimethylpyrazol-4-yl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-amine
—— (6S)-N-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-amine —— C14H21N5O
(6S)-N-[(5-methoxy-1,3-dimethylpyrazol-4-yl)methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-amine
—— (6R)-N-[[5-(dimethylamino)-1,3-dimethylpyrazol-4-yl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-amine —— C15H24N6
(6R)-N-[[5-(dimethylamino)-1,3-dimethylpyrazol-4-yl]methyl]-5,6,7,8-tetrahydroimidazo[1,2-a]pyridin-6-amine
—— 6-chloro-2-methyl-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]pyrimidin-4-amine —— C16H19ClN4
6-chloro-2-methyl-N-[[(3R)-1-phenylpyrrolidin-3-yl]methyl]pyrimidin-4-amine
—— 6-methyl-4-[(3S)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C16H23N7
6-methyl-4-[(3S)-3-(4-methyl-1,2,4-triazol-3-yl)piperidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-chloro-2-methyl-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]pyrimidin-4-amine —— C16H19ClN4
6-chloro-2-methyl-N-[[(3S)-1-phenylpyrrolidin-3-yl]methyl]pyrimidin-4-amine
—— 6-[[(3S)-1-[(1-methyl-2-oxopyridin-4-yl)methyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C18H21N5O
6-[[(3S)-1-[(1-methyl-2-oxopyridin-4-yl)methyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-[[(3R)-1-[(3R,5R)-5-methyl-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C16H20N4O2
6-[[(3R)-1-[(3R,5R)-5-methyl-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-[[(3R)-1-[(3R,5S)-5-methyl-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C16H20N4O2
6-[[(3R)-1-[(3R,5S)-5-methyl-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-[[(3R)-1-quinazolin-4-ylpyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C19H18N6
6-[[(3R)-1-quinazolin-4-ylpyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-[[(3R)-1-[(1-methyl-2-oxopyridin-4-yl)methyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C18H21N5O
6-[[(3R)-1-[(1-methyl-2-oxopyridin-4-yl)methyl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-[[(3S)-1-[(3R)-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C15H18N4O2
6-[[(3S)-1-[(3R)-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— (6R)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one —— C21H21NO2S
(6R)-6-(4-hydroxyphenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[c][1,5]benzothiazepin-7-one
—— (6R)-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C19H16FNOS
(6R)-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6S,9R)-6-methyl-9-phenyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one —— C17H15F3N4O
(6S,9R)-6-methyl-9-phenyl-2-(trifluoromethyl)-5,6,7,9-tetrahydro-4H-[1,2,4]triazolo[5,1-b]quinazolin-8-one
—— 6-methyl-4-[(2R)-2-(2-methylphenyl)pyrrolidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H24N4
6-methyl-4-[(2R)-2-(2-methylphenyl)pyrrolidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— 6-[[(3S)-1-quinazolin-4-ylpyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C19H18N6
6-[[(3S)-1-quinazolin-4-ylpyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile
—— 6-(butanoylamino)-N-[(2R)-butan-2-yl]-12,12-dimethyl-11-oxa-4-thia-2-azatricyclo[7.4.0.03,7]trideca-1,3(7),5,8-tetraene-5-carboxamide —— C21H29N3O3S
6-(butanoylamino)-N-[(2R)-butan-2-yl]-12,12-dimethyl-11-oxa-4-thia-2-azatricyclo[7.4.0.03,7]trideca-1,3(7),5,8-tetraene-5-carboxamide
—— 6-methyl-4-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine —— C19H24N4
6-methyl-4-[(2S)-2-(2-methylphenyl)pyrrolidin-1-yl]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidine
—— (6S)-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one —— C19H16FNOS
(6S)-6-(4-fluorophenyl)-8,9,10,11-tetrahydro-6H-benzo[c][1,5]benzothiazepin-7-one
—— (6S,7R)-7-(4-carboxybutanoylamino)-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C13H16N2O6S
(6S,7R)-7-(4-carboxybutanoylamino)-3-methyl-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 6-[[(3R)-1-[(3S,5R)-5-methyl-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile —— C16H20N4O2
6-[[(3R)-1-[(3S,5R)-5-methyl-2-oxooxolan-3-yl]pyrrolidin-3-yl]methylamino]pyridine-3-carbonitrile