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—— (6R)-1-N-(2-methoxyethyl)-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C23H31N5O4
(6R)-1-N-(2-methoxyethyl)-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— (6S)-1-N-(4-ethoxyphenyl)-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide —— C28H33N5O4
(6S)-1-N-(4-ethoxyphenyl)-6-methyl-6-N-[(4-methylphenyl)methyl]-8-oxo-7-propyl-5H-imidazo[1,5-a]pyrazine-1,6-dicarboxamide
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[(2S)-2-phenylpropyl]pyridazin-3-amine —— C20H20ClN3O2S
6-[(4-chlorophenyl)methylsulfonyl]-N-[(2S)-2-phenylpropyl]pyridazin-3-amine
—— 6-[(2S)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione —— C19H18ClN3O4S
6-[(2S)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione
—— 6-[(1R)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione —— C21H23N3O5S
6-[(1R)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione
—— 6-[(1S)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione —— C21H23N3O5S
6-[(1S)-6,7-dimethoxy-1-methyl-3,4-dihydro-1H-isoquinoline-2-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-amine —— C18H23ClN4O2S
6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2R)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-amine
—— 6-[(2R)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione —— C19H18ClN3O4S
6-[(2R)-6-chloro-2-ethyl-2,3-dihydro-1,4-benzoxazine-4-carbonyl]-1,3-dimethylthieno[2,3-d]pyrimidine-2,4-dione
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-amine —— C18H23ClN4O2S
6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2S)-1-ethylpyrrolidin-2-yl]methyl]pyridazin-3-amine
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]pyridazin-3-amine —— C21H29ClN4O2S
6-[(4-chlorophenyl)methylsulfonyl]-N-[3-[(2S)-2-ethylpiperidin-1-yl]propyl]pyridazin-3-amine
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]pyridazin-3-amine —— C21H29ClN4O2S
6-[(4-chlorophenyl)methylsulfonyl]-N-[3-[(2R)-2-ethylpiperidin-1-yl]propyl]pyridazin-3-amine
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[(2R)-2-phenylpropyl]pyridazin-3-amine —— C20H20ClN3O2S
6-[(4-chlorophenyl)methylsulfonyl]-N-[(2R)-2-phenylpropyl]pyridazin-3-amine
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2R)-oxolan-2-yl]methyl]pyridazin-3-amine —— C16H18ClN3O3S
6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2R)-oxolan-2-yl]methyl]pyridazin-3-amine
—— 6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2S)-oxolan-2-yl]methyl]pyridazin-3-amine —— C16H18ClN3O3S
6-[(4-chlorophenyl)methylsulfonyl]-N-[[(2S)-oxolan-2-yl]methyl]pyridazin-3-amine
—— 6-nitro-2-[[(2R)-oxolan-2-yl]methyl]benzo[de]isoquinoline-1,3-dione —— C17H14N2O5
6-nitro-2-[[(2R)-oxolan-2-yl]methyl]benzo[de]isoquinoline-1,3-dione
—— 6-(Benzylthio)-3-(3,4-dimethoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine —— C20H18N4O2S
6-(Benzylthio)-3-(3,4-dimethoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine
—— (6R)-10-bromo-3-ethylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C17H14BrN5OS
(6R)-10-bromo-3-ethylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— (6R)-3-propylsulfanyl-6-pyridin-3-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C18H17N5OS
(6R)-3-propylsulfanyl-6-pyridin-3-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— 6-((3-Fluorobenzyl)thio)-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine —— C19H15FN4OS
6-((3-Fluorobenzyl)thio)-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine
—— (6S)-10-bromo-3-ethylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine —— C17H14BrN5OS
(6S)-10-bromo-3-ethylsulfanyl-6-pyridin-4-yl-6,7-dihydro-[1,2,4]triazino[5,6-d][3,1]benzoxazepine
—— 6-[[(2S)-2-hydroxy-3-[2-(trifluoromethyl)phenoxy]propyl]-methylamino]pyridine-3-carbonitrile —— C17H16F3N3O2
6-[[(2S)-2-hydroxy-3-[2-(trifluoromethyl)phenoxy]propyl]-methylamino]pyridine-3-carbonitrile
—— 6-((4-Fluorobenzyl)thio)-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine —— C19H15FN4OS
6-((4-Fluorobenzyl)thio)-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine
—— 6-Benzylsulfanyl-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine —— C19H16N4OS
6-Benzylsulfanyl-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine
—— 6-((2-Fluorobenzyl)thio)-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine —— C19H15FN4OS
6-((2-Fluorobenzyl)thio)-3-(4-methoxyphenyl)-[1,2,4]triazolo[4,3-b]pyridazine
—— (6S,9R)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H26N2O3
(6S,9R)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9S)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H26N2O3
(6R,9S)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6R,9R)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H26N2O3
(6R,9R)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S,9S)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C28H26N2O3
(6S,9S)-5-(cyclopropanecarbonyl)-6-(furan-2-yl)-9-(4-methylphenyl)-6a,8,9,10-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-2-acetamido-6-methyl-N-naphthalen-1-yl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide —— C22H22N2O2S
(6S)-2-acetamido-6-methyl-N-naphthalen-1-yl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
—— 6-ethyl-3-[(S)-(4-ethylpiperazine-1,4-diium-1-yl)-[1-(2-methoxyethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H33N7O2+2
6-ethyl-3-[(S)-(4-ethylpiperazine-1,4-diium-1-yl)-[1-(2-methoxyethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one —— C23H33N6O+
6-methyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(R)-(4-ethylpiperazin-1-yl)-[1-(2-methoxyethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H31N7O2
6-ethyl-3-[(R)-(4-ethylpiperazin-1-yl)-[1-(2-methoxyethyl)tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-methoxy-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C23H32N6O2
6-methoxy-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C23H32N6O
6-methyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— (6,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(thiophen-2-ylmethyl)azanium —— C17H19N2OS+
(6,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl-(thiophen-2-ylmethyl)azanium
—— 6-methyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C23H32N6O
6-methyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one —— C24H35N6O+
6-ethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-3-[(S)-[(3S)-3-methylpiperidin-1-ium-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C23H31N6O2+
6-methyl-3-[(S)-[(3S)-3-methylpiperidin-1-ium-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-5-[(2Z)-2-(pyridin-4-ylmethylidene)hydrazinyl]-2H-1,2,4-triazin-3-one —— C10H10N6O
6-methyl-5-[(2Z)-2-(pyridin-4-ylmethylidene)hydrazinyl]-2H-1,2,4-triazin-3-one
—— 6,8-dimethyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C24H34N6O
6,8-dimethyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— (6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl-[2-(3-methylphenyl)ethyl]azanium —— C21H25N2O2+
(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl-[2-(3-methylphenyl)ethyl]azanium
—— (6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl-[(4-methoxyphenyl)methyl]azanium —— C20H23N2O3+
(6-ethoxy-2-oxo-1H-quinolin-3-yl)methyl-[(4-methoxyphenyl)methyl]azanium
—— 6,8-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one —— C24H35N6O+
6,8-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one —— C23H33N6O+
6-methyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one
—— 6-ethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C24H34N6O
6-ethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one
—— 6,7-dimethyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one —— C24H35N6O+
6,7-dimethyl-3-[(R)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-ium-1-yl]methyl]-1H-quinolin-2-one
—— 6-methyl-3-[(R)-[(3S)-3-methylpiperidin-1-ium-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C23H31N6O2+
6-methyl-3-[(R)-[(3S)-3-methylpiperidin-1-ium-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (6-methyl-2-oxo-1H-quinolin-3-yl)methyl-(thiophen-2-ylmethyl)azanium —— C16H17N2OS+
(6-methyl-2-oxo-1H-quinolin-3-yl)methyl-(thiophen-2-ylmethyl)azanium
—— 6-methyl-3-[(S)-[(3S)-3-methylpiperidin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C23H30N6O2
6-methyl-3-[(S)-[(3S)-3-methylpiperidin-1-yl]-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— 6,8-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one —— C24H34N6O
6,8-dimethyl-3-[(S)-[1-(2-methylbutan-2-yl)tetrazol-5-yl]-[(3S)-3-methylpiperidin-1-yl]methyl]-1H-quinolin-2-one