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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-8-[(2-aminopyridin-3-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O
(6R)-8-[(2-aminopyridin-3-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-pyrimidin-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C16H24N4O2
(6R)-2-(2-methoxyethyl)-8-pyrimidin-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-4-[[2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-1,4-oxazepan-6-yl]methanol —— C21H35N3O2
[(6S)-4-[[2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-1,4-oxazepan-6-yl]methanol
—— (6S)-8-[(2-aminopyridin-3-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O
(6S)-8-[(2-aminopyridin-3-yl)methyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(1-propan-2-ylpyrrol-2-yl)methanone —— C18H29N3O3
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(1-propan-2-ylpyrrol-2-yl)methanone
—— 6-methyl-4-[(2S)-2-methyl-4-(2-methylphenyl)-5-oxopiperazine-1-carbonyl]-1H-quinolin-2-one —— C23H23N3O3
6-methyl-4-[(2S)-2-methyl-4-(2-methylphenyl)-5-oxopiperazine-1-carbonyl]-1H-quinolin-2-one
—— 6-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C19H25N7
6-[(3S)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— [(6R)-4-[[2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-1,4-oxazepan-6-yl]methanol —— C21H35N3O2
[(6R)-4-[[2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-1,4-oxazepan-6-yl]methanol
—— 6-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile —— C19H25N7
6-[(3R)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-1,2,4-triazol-3-yl]piperidin-1-yl]pyridine-3-carbonitrile
—— (6R)-2-(2-methoxyethyl)-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O3
(6R)-2-(2-methoxyethyl)-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(1,3-Benzothiazol-2-ylamino)-1-(4-phenylpiperazin-1-yl)hexan-1-one —— C23H28N4OS
6-(1,3-Benzothiazol-2-ylamino)-1-(4-phenylpiperazin-1-yl)hexan-1-one
—— 6-Nitro-4-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,4-benzoxazin-3-one —— C20H20N4O5
6-Nitro-4-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-1,4-benzoxazin-3-one
—— 6-[(Z)-[[2-[(3S)-1,1-dioxothiolan-3-yl]acetyl]hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid —— C16H20N2O7S
6-[(Z)-[[2-[(3S)-1,1-dioxothiolan-3-yl]acetyl]hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid
—— 6-[(Z)-[[2-[(3R)-1,1-dioxothiolan-3-yl]acetyl]hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid —— C16H20N2O7S
6-[(Z)-[[2-[(3R)-1,1-dioxothiolan-3-yl]acetyl]hydrazinylidene]methyl]-2,3-dimethoxybenzoic acid
—— 6-[(Z)-[[2-[(3S)-1,1-dioxothiolan-3-yl]acetyl]hydrazinylidene]methyl]-2,3-dimethoxybenzoate —— C16H19N2O7S-
6-[(Z)-[[2-[(3S)-1,1-dioxothiolan-3-yl]acetyl]hydrazinylidene]methyl]-2,3-dimethoxybenzoate
—— (6S)-8-(3-fluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H23FN2O3
(6S)-8-(3-fluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(benzenesulfonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O3S
(6R)-8-(benzenesulfonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N6O2
(6R)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-acetylpyridin-2-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O3
(6S)-8-(5-acetylpyridin-2-yl)-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6S)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N6O
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6R)-8-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-pyrimidin-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C16H24N4O2
(6S)-2-(2-methoxyethyl)-8-pyrimidin-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(benzenesulfonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O3S
(6S)-8-(benzenesulfonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-thieno[3,2-d]pyrimidin-4-yl-1,4-oxazepan-6-ol —— C11H13N3O2S
(6R)-4-thieno[3,2-d]pyrimidin-4-yl-1,4-oxazepan-6-ol
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(1-propan-2-ylpyrrol-2-yl)methanone —— C18H29N3O3
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(1-propan-2-ylpyrrol-2-yl)methanone
—— (6R)-4-[1-(1,3-benzodioxol-5-yl)piperidin-4-yl]-1,4-oxazepan-6-ol —— C17H24N2O4
(6R)-4-[1-(1,3-benzodioxol-5-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
—— (6S)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N6O2
(6S)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-[(5-methoxy-2H-indazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6R)-2-cyclopropyl-8-[(5-methoxy-2H-indazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-ethylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H25N3O3S
(6R)-8-ethylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-(3,4-dimethylphenoxy)ethyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N2O3
(6S)-8-[2-(3,4-dimethylphenoxy)ethyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-amino-7H-purin-6-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N7O2
(6S)-8-(2-amino-7H-purin-6-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28FN5O2
(6S)-8-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[1-(1,3-benzodioxol-5-yl)piperidin-4-yl]-1,4-oxazepan-6-ol —— C17H24N2O4
(6S)-4-[1-(1,3-benzodioxol-5-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
—— (6R)-2-(3-methylbutyl)-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N3O2
(6R)-2-(3-methylbutyl)-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(2R)-2-[5-(methylcarbamoyl)thiophen-2-yl]pyrrolidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C17H20N4O3S
6-[[(2R)-2-[5-(methylcarbamoyl)thiophen-2-yl]pyrrolidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-2-cyclopentyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N5O
(6R)-2-cyclopentyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-[(5-methoxy-2H-indazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6S)-2-cyclopropyl-8-[(5-methoxy-2H-indazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methylbutyl)-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H31N3O2
(6S)-2-(3-methylbutyl)-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-propan-2-yl-3-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-1H-pyridin-2-one —— C20H26N2O2S
6-propan-2-yl-3-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-1H-pyridin-2-one
—— (6S)-8-(4-aminopyrimidin-2-yl)-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N5O
(6S)-8-(4-aminopyrimidin-2-yl)-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-amino-7H-purin-6-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N7O2
(6R)-8-(2-amino-7H-purin-6-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[(4-pyrazol-1-ylphenyl)methylamino]methyl]-1,4-oxazepan-6-ol —— C16H22N4O2
(6R)-6-[[(4-pyrazol-1-ylphenyl)methylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-2-butyl-8-(4-chloro-1-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27ClN4O2
(6R)-2-butyl-8-(4-chloro-1-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2,6-difluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H22F2N2O3
(6S)-8-(2,6-difluorobenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-methylsulfanylpyrimidin-4-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C17H26N4OS
(6S)-8-(2-methylsulfanylpyrimidin-4-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— [6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone —— C20H22N4O3
[6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidin-3-yl]-[(2S)-2-(3-methoxyphenyl)pyrrolidin-1-yl]methanone
—— 6-fluoro-2-[(2R)-1-(1H-imidazol-5-ylmethyl)pyrrolidin-2-yl]-1H-benzimidazole —— C15H16FN5
6-fluoro-2-[(2R)-1-(1H-imidazol-5-ylmethyl)pyrrolidin-2-yl]-1H-benzimidazole
—— 6-fluoro-2-[(2S)-1-(1H-imidazol-5-ylmethyl)pyrrolidin-2-yl]-1H-benzimidazole —— C15H16FN5
6-fluoro-2-[(2S)-1-(1H-imidazol-5-ylmethyl)pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-6-[[(4-pyrazol-1-ylphenyl)methylamino]methyl]-1,4-oxazepan-6-ol —— C16H22N4O2
(6S)-6-[[(4-pyrazol-1-ylphenyl)methylamino]methyl]-1,4-oxazepan-6-ol