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—— (6R)-8-(6-aminopyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N7O
(6R)-8-(6-aminopyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopentyl-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N3O3
(6S)-2-cyclopentyl-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(3-methylpyrazin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O
(6S)-8-(3-methylpyrazin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[2-(4-phenyl-1,3-thiazol-2-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C17H23N3O2S
(6S)-6-[[2-(4-phenyl-1,3-thiazol-2-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6-chloro-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)-[(2R)-1-methylsulfonylpyrrolidin-2-yl]methanone —— C17H20ClN3O3S
(6-chloro-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)-[(2R)-1-methylsulfonylpyrrolidin-2-yl]methanone
—— (6R)-2-cyclopropyl-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N3O
(6R)-2-cyclopropyl-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6R)-2-(cyclopropylmethyl)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C16H20N4O3
6-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O2
(6R)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-methylpyrazin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N6O
(6R)-8-(3-methylpyrazin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine —— C19H25N5
6-methyl-2-[[(2R)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone —— C13H19N3O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone
—— 6-methyl-2-[[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine —— C19H25N5
6-methyl-2-[[(2S)-2-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-pyrazin-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N6O
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-pyrazin-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[6-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H24F3N3O2
(6S)-2-(2-methoxyethyl)-8-[6-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N5O2
(6S)-2-(cyclopropylmethyl)-8-[2-(1,2,4-triazol-1-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N6O2
(6S)-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-pyrazin-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C19H24N6O
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-pyrazin-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N6O2
(6R)-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-N-[4-[ethyl(propan-2-yl)amino]phenyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide —— C21H25ClN2O3
6-chloro-N-[4-[ethyl(propan-2-yl)amino]phenyl]-3,4-dihydro-2H-1,5-benzodioxepine-8-carboxamide
—— (6R)-2-butyl-8-(3-pyridin-3-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6R)-2-butyl-8-(3-pyridin-3-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopentyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6R)-2-cyclopentyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(5-phenyl-1,2-oxazol-3-yl)methanone —— C20H25N3O4
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(5-phenyl-1,2-oxazol-3-yl)methanone
—— (6S)-2-cyclopentyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6S)-2-cyclopentyl-8-[2-(5-methylpyrazol-1-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-(3-pyridin-3-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6S)-2-butyl-8-(3-pyridin-3-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(5-phenyl-1,2-oxazol-3-yl)methanone —— C20H25N3O4
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(5-phenyl-1,2-oxazol-3-yl)methanone
—— (6R)-2-(cyclopropylmethyl)-8-(2-methoxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N2O3
(6R)-2-(cyclopropylmethyl)-8-(2-methoxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone —— C18H28N4O3
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone
—— 6-[(3R)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C15H15N5O2S
6-[(3R)-3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl-[(1R)-1-phenylethyl]azanium —— C20H22NO2+
(6,7-dimethyl-2-oxochromen-4-yl)methyl-[(1R)-1-phenylethyl]azanium
—— (6,7-dimethyl-2-oxochromen-4-yl)methyl-[(1S)-1-phenylethyl]azanium —— C20H22NO2+
(6,7-dimethyl-2-oxochromen-4-yl)methyl-[(1S)-1-phenylethyl]azanium
—— (6R)-6-[[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C13H21N5O2S
(6R)-6-[[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone —— C18H28N4O3
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone
—— (6R)-2-(2-hydroxyethyl)-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O2
(6R)-2-(2-hydroxyethyl)-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C13H21N5O2S
(6S)-6-[[2-(2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-6-(pyrrolidin-1-ylmethyl)-4-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-1,4-oxazepan-6-ol —— C17H24F3N3O2
(6R)-6-(pyrrolidin-1-ylmethyl)-4-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-1,4-oxazepan-6-ol
—— (6S)-2-(cyclopropylmethyl)-8-(2-methoxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N2O3
(6S)-2-(cyclopropylmethyl)-8-(2-methoxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6R)-2-(2-methoxyethyl)-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-(pyrrolidin-1-ylmethyl)-4-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-1,4-oxazepan-6-ol —— C17H24F3N3O2
(6S)-6-(pyrrolidin-1-ylmethyl)-4-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-1,4-oxazepan-6-ol
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(5-methoxy-1H-indazol-3-yl)methanone —— C14H17N3O4
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(5-methoxy-1H-indazol-3-yl)methanone
—— (6R)-6-[[4-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol —— C16H28N4O2
(6R)-6-[[4-(2-pyrazol-1-ylethyl)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol
—— 6-[[(2R)-2-ethylmorpholin-4-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide —— C20H25N5O3S
6-[[(2R)-2-ethylmorpholin-4-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-4-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,4-oxazepan-6-ol —— C18H28ClN3O2
(6R)-4-[3-[4-(3-chlorophenyl)piperazin-1-yl]propyl]-1,4-oxazepan-6-ol
—— (6R)-8-propylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O3S
(6R)-8-propylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6S)-2-(2-methoxyethyl)-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(5-propylthiophen-3-yl)methanone —— C13H19NO3S
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(5-propylthiophen-3-yl)methanone
—— (6R)-4-[[5-(1-methylbenzimidazol-2-yl)furan-2-yl]methyl]-1,4-oxazepan-6-ol —— C18H21N3O3
(6R)-4-[[5-(1-methylbenzimidazol-2-yl)furan-2-yl]methyl]-1,4-oxazepan-6-ol
—— 6-[[(2S)-2-ethylmorpholin-4-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide —— C20H25N5O3S
6-[[(2S)-2-ethylmorpholin-4-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-8-[2-[(5-amino-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N6O2S
(6R)-8-[2-[(5-amino-1H-1,2,4-triazol-3-yl)sulfanyl]acetyl]-2-butyl-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(5-methoxy-1H-indazol-3-yl)methanone —— C14H17N3O4
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(5-methoxy-1H-indazol-3-yl)methanone