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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(1R)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H20N4O2S
6-[(1R)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6S)-2-(2-methoxyethyl)-8-[2-(N-methylanilino)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6S)-2-(2-methoxyethyl)-8-[2-(N-methylanilino)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-[4-(1H-pyrazol-5-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6R)-2-cyclopropyl-8-[4-(1H-pyrazol-5-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(3-hydroxy-2-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O4
(6S)-8-(3-hydroxy-2-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[5-(pyrazol-1-ylmethyl)furan-2-yl]methanone —— C19H26N4O4
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[5-(pyrazol-1-ylmethyl)furan-2-yl]methanone
—— 6-[(6S)-6-hydroxy-1,4-oxazepane-4-carbonyl]-3,4-dihydro-2H-[1]benzothiolo[2,3-c]pyridin-1-one —— C17H18N2O4S
6-[(6S)-6-hydroxy-1,4-oxazepane-4-carbonyl]-3,4-dihydro-2H-[1]benzothiolo[2,3-c]pyridin-1-one
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-hydroxy-2-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O4
(6R)-8-(3-hydroxy-2-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-cyclopropylpropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6R)-8-(3-cyclopropylpropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(6R)-6-hydroxy-1,4-oxazepane-4-carbonyl]-3,4-dihydro-2H-[1]benzothiolo[2,3-c]pyridin-1-one —— C17H18N2O4S
6-[(6R)-6-hydroxy-1,4-oxazepane-4-carbonyl]-3,4-dihydro-2H-[1]benzothiolo[2,3-c]pyridin-1-one
—— 6-oxo-N-[[(2S)-oxolan-2-yl]methyl]-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C15H16N4O3
6-oxo-N-[[(2S)-oxolan-2-yl]methyl]-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[5-(pyrazol-1-ylmethyl)furan-2-yl]methanone —— C19H26N4O4
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[5-(pyrazol-1-ylmethyl)furan-2-yl]methanone
—— (6S)-8-(3-cyclopropylpropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6S)-8-(3-cyclopropylpropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-2-methylquinolin-4-yl)-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methanone —— C22H29N3O2
(6-ethyl-2-methylquinolin-4-yl)-[4-[[(2S)-oxolan-2-yl]methyl]piperazin-1-yl]methanone
—— 6-[2-[(2S)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethylamino]pyridine-2-carbonitrile —— C17H20N6O2
6-[2-[(2S)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethylamino]pyridine-2-carbonitrile
—— (6R)-2-cyclopropyl-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O
(6R)-2-cyclopropyl-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-2-methylquinolin-4-yl)-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methanone —— C22H29N3O2
(6-ethyl-2-methylquinolin-4-yl)-[4-[[(2R)-oxolan-2-yl]methyl]piperazin-1-yl]methanone
—— 6-chloro-N-[(3S,4R)-4-methoxypyrrolidin-3-yl]pyridazin-3-amine —— C9H13ClN4O
6-chloro-N-[(3S,4R)-4-methoxypyrrolidin-3-yl]pyridazin-3-amine
—— 6-oxo-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide —— C15H16N4O3
6-oxo-N-[[(2R)-oxolan-2-yl]methyl]-2-pyridin-2-yl-1H-pyrimidine-5-carboxamide
—— 6-[[(3S,4R)-4-methoxypyrrolidin-3-yl]amino]-2H-1,2,4-triazine-3,5-dione —— C8H13N5O3
6-[[(3S,4R)-4-methoxypyrrolidin-3-yl]amino]-2H-1,2,4-triazine-3,5-dione
—— 6-chloro-N-[(3R,4R)-4-methoxypyrrolidin-3-yl]pyridazin-3-amine —— C9H13ClN4O
6-chloro-N-[(3R,4R)-4-methoxypyrrolidin-3-yl]pyridazin-3-amine
—— 6-[[(3R,4R)-4-methoxypyrrolidin-3-yl]amino]-2H-1,2,4-triazine-3,5-dione —— C8H13N5O3
6-[[(3R,4R)-4-methoxypyrrolidin-3-yl]amino]-2H-1,2,4-triazine-3,5-dione
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(4-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethylamino]pyridine-2-carbonitrile —— C17H20N6O2
6-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethylamino]pyridine-2-carbonitrile
—— (6S)-8-(2-hydroxy-4-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O4
(6S)-8-(2-hydroxy-4-methylbenzoyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R,4R)-4-methoxypyrrolidin-3-yl]amino]pyridine-3-carbonitrile —— C11H14N4O
6-[[(3R,4R)-4-methoxypyrrolidin-3-yl]amino]pyridine-3-carbonitrile
—— (6S)-2-cyclopropyl-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O
(6S)-2-cyclopropyl-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[2-(2-hydroxyethoxy)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6R)-8-[2-(2-hydroxyethoxy)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-(3-methylpyrazol-1-yl)ethyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O
(6S)-8-[2-(3-methylpyrazol-1-yl)ethyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methylamino]methyl]-1,4-oxazepan-6-ol —— C13H19F3N4O2
(6R)-6-[[[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-4-[(3-morpholin-4-ylphenyl)methyl]-1,4-oxazepan-6-ol —— C16H24N2O3
(6S)-4-[(3-morpholin-4-ylphenyl)methyl]-1,4-oxazepan-6-ol
—— 6-[[(3S,4R)-4-methoxypyrrolidin-3-yl]amino]pyridine-3-carbonitrile —— C11H14N4O
6-[[(3S,4R)-4-methoxypyrrolidin-3-yl]amino]pyridine-3-carbonitrile
—— (6R)-8-[2-(3-methylpyrazol-1-yl)ethyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O
(6R)-8-[2-(3-methylpyrazol-1-yl)ethyl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[(3-morpholin-4-ylphenyl)methyl]-1,4-oxazepan-6-ol —— C16H24N2O3
(6R)-4-[(3-morpholin-4-ylphenyl)methyl]-1,4-oxazepan-6-ol
—— (6S)-6-[[[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methylamino]methyl]-1,4-oxazepan-6-ol —— C13H19F3N4O2
(6S)-6-[[[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-8-[2-(2-hydroxyethoxy)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6S)-8-[2-(2-hydroxyethoxy)ethyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N5O2
(6S)-2-(cyclopropylmethyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-pyrrolidin-1-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H33N5O
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-(2-pyrrolidin-1-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-(1-ethyl-5-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6S)-2-butyl-8-(1-ethyl-5-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [6-[[(3R)-3-hydroxypyrrolidin-3-yl]methyl]-2-(methylamino)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]-pyrrolidin-1-ylmethanone —— C18H28N6O2
[6-[[(3R)-3-hydroxypyrrolidin-3-yl]methyl]-2-(methylamino)-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-4-yl]-pyrrolidin-1-ylmethanone
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(2-methyl-5-thiophen-2-ylpyrazol-3-yl)methanone —— C15H19N3O3S
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(2-methyl-5-thiophen-2-ylpyrazol-3-yl)methanone
—— (6R)-2-butyl-8-(6-methyl-2-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O
(6R)-2-butyl-8-(6-methyl-2-propylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[(1,3-benzodioxol-5-ylmethylamino)methyl]-1,4-oxazepan-6-ol —— C14H20N2O4
(6S)-6-[(1,3-benzodioxol-5-ylmethylamino)methyl]-1,4-oxazepan-6-ol
—— (6R)-8-(1-ethylpyrazole-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6R)-8-(1-ethylpyrazole-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N6O2
(6R)-8-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methylbutyl)-8-[3-(5-methyltetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H34N6O
(6R)-2-(3-methylbutyl)-8-[3-(5-methyltetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(1-ethylpyrazole-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6S)-8-(1-ethylpyrazole-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N5O2
(6R)-2-(cyclopropylmethyl)-8-[2-(methylamino)pyrimidine-5-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-ethylpyrimidine-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6R)-8-(2-ethylpyrimidine-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-[(4-methylsulfanylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2S
(6R)-2-(2-methoxyethyl)-8-[(4-methylsulfanylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one