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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(6S)-4-[5-methyl-6-(2-methylpyridin-3-yl)oxypyrimidin-4-yl]-1,4-oxazepan-6-yl]methanol —— C17H22N4O3
[(6S)-4-[5-methyl-6-(2-methylpyridin-3-yl)oxypyrimidin-4-yl]-1,4-oxazepan-6-yl]methanol
—— (6R)-8-(2-amino-2-methylpropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N5O
(6R)-8-(2-amino-2-methylpropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[1-(2-fluorophenyl)piperidin-4-yl]-1,4-oxazepan-6-ol —— C16H23FN2O2
(6R)-4-[1-(2-fluorophenyl)piperidin-4-yl]-1,4-oxazepan-6-ol
—— (6S)-2-(3-methoxypropyl)-8-[4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H29N5O2
(6S)-2-(3-methoxypropyl)-8-[4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-hydroxyethyl)-8-[(1-methylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C16H26N4O2
(6R)-2-(2-hydroxyethyl)-8-[(1-methylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-amino-2-methylpropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N5O
(6S)-8-(2-amino-2-methylpropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-(3-phenoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O4
(6S)-2-(2-hydroxyethyl)-8-(3-phenoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-[(1-methylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C16H26N4O2
(6S)-2-(2-hydroxyethyl)-8-[(1-methylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-hydroxyethyl)-8-(3-phenoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O4
(6R)-2-(2-hydroxyethyl)-8-(3-phenoxypropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-(4-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6R)-2-butyl-8-(4-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-cyclopropylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H25N3O3S
(6S)-8-cyclopropylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-[4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H29N5O2
(6R)-2-(3-methoxypropyl)-8-[4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[[4-amino-6-(3-methylanilino)-1,3,5-triazin-2-yl]methyl]-1,4-oxazepan-6-ol —— C16H22N6O2
(6S)-4-[[4-amino-6-(3-methylanilino)-1,3,5-triazin-2-yl]methyl]-1,4-oxazepan-6-ol
—— 6-chloro-N-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridine-3-sulfonamide —— C12H15ClF3N3O2S
6-chloro-N-[[(3S)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridine-3-sulfonamide
—— 6-ethyl-N,2-dimethyl-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide —— C19H21N3OS
6-ethyl-N,2-dimethyl-N-[(1S)-1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C15H17F3N4O3
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— 6-ethyl-N,2-dimethyl-N-[(1R)-1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide —— C19H21N3OS
6-ethyl-N,2-dimethyl-N-[(1R)-1-(1,3-thiazol-5-yl)ethyl]quinoline-4-carboxamide
—— (6S)-2-butyl-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N4OS
(6S)-2-butyl-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4
(6S)-2-(2-hydroxyethyl)-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6S)-8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6R)-2-butyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-N-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridine-3-sulfonamide —— C12H15ClF3N3O2S
6-chloro-N-[[(3R)-1-(2,2,2-trifluoroethyl)pyrrolidin-3-yl]methyl]pyridine-3-sulfonamide
—— (6S)-2-(3-methoxypropyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6S)-2-(3-methoxypropyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6R)-2-(3-methoxypropyl)-8-(3-methoxypyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopentyl-8-(2,3-dihydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N2O4
(6S)-2-cyclopentyl-8-(2,3-dihydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-(2-fluoro-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6R)-2-butyl-8-(2-fluoro-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6S)-2-butyl-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-(4-propan-2-ylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H34N2O2
(6S)-2-butyl-8-(4-propan-2-ylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C17H28N4OS
(6R)-2-butyl-8-[(4-methylthiadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-(2-fluoro-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6S)-2-butyl-8-(2-fluoro-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6R)-8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone —— C15H17F3N4O3
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-2-yl]methanone
—— (6S)-8-ethylsulfonyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H25N3O3S
(6S)-8-ethylsulfonyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-cyclopropylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H25N3O3S
(6R)-8-cyclopropylsulfonyl-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[[4-amino-6-(3-methylanilino)-1,3,5-triazin-2-yl]methyl]-1,4-oxazepan-6-ol —— C16H22N6O2
(6R)-4-[[4-amino-6-(3-methylanilino)-1,3,5-triazin-2-yl]methyl]-1,4-oxazepan-6-ol
—— (6R)-8-ethylsulfonyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H25N3O3S
(6R)-8-ethylsulfonyl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2S)-1-[(5-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C17H21N5
6-methyl-2-[(2S)-1-[(5-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-2-cyclopentyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O
(6S)-2-cyclopentyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C18H19N5O3
6-[(3S)-3-(4-methyl-1H-benzimidazol-2-yl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (6R)-2-cyclopropyl-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26FN3O
(6R)-2-cyclopropyl-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-pentan-3-yl-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-pentan-3-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-hydroxyethyl)-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4
(6R)-2-(2-hydroxyethyl)-8-(2-hydroxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2R)-1-[(5-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C17H21N5
6-methyl-2-[(2R)-1-[(5-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-6-[[2-(3-pyridin-3-yl-1H-1,2,4-triazol-5-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C15H22N6O2
(6S)-6-[[2-(3-pyridin-3-yl-1H-1,2,4-triazol-5-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-6-[(10-methoxy-2,3,4,6-tetrahydro-1,5-benzoxazocin-5-yl)methyl]-1,4-oxazepan-6-ol —— C17H26N2O4
(6R)-6-[(10-methoxy-2,3,4,6-tetrahydro-1,5-benzoxazocin-5-yl)methyl]-1,4-oxazepan-6-ol
—— (6R)-2-cyclopentyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O
(6R)-2-cyclopentyl-8-(2,5,6-trimethylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-3-[(6R)-6-hydroxy-1,4-oxazepane-4-carbonyl]-1,5-dimethylpyridin-2-one —— C15H22N2O4
6-ethyl-3-[(6R)-6-hydroxy-1,4-oxazepane-4-carbonyl]-1,5-dimethylpyridin-2-one
—— 6-ethyl-3-[(6S)-6-hydroxy-1,4-oxazepane-4-carbonyl]-1,5-dimethylpyridin-2-one —— C15H22N2O4
6-ethyl-3-[(6S)-6-hydroxy-1,4-oxazepane-4-carbonyl]-1,5-dimethylpyridin-2-one
—— (6S)-2-cyclopropyl-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H26FN3O
(6S)-2-cyclopropyl-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C17H24N4O4
(6R)-4-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol