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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6R)-2-(2-methoxyethyl)-8-(5-propyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O4
(6R)-2-(2-methoxyethyl)-8-(5-propyl-1,2-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O2
(6R)-2-cyclopropyl-8-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-(2-aminopyrimidin-4-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C14H23N5O2
(6R)-4-(2-aminopyrimidin-4-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6S)-2-(2-methoxyethyl)-8-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N4O3
(6S)-2-(2-methoxyethyl)-8-[(3-propan-2-yl-1,2,4-oxadiazol-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-ethyl-8-(3-methoxyphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N2O4S
(6S)-2-ethyl-8-(3-methoxyphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-hydroxyethyl)-8-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N2O3
(6R)-2-(2-hydroxyethyl)-8-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-(3-methoxyphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N2O4S
(6R)-2-ethyl-8-(3-methoxyphenyl)sulfonyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[2-[(3-chlorophenyl)methylsulfanyl]ethylamino]methyl]-1,4-oxazepan-6-ol —— C15H23ClN2O2S
(6S)-6-[[2-[(3-chlorophenyl)methylsulfanyl]ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-2-butyl-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O2
(6S)-2-butyl-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(5-propyl-1,2-oxazol-3-yl)methanone —— C17H27N3O4
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(5-propyl-1,2-oxazol-3-yl)methanone
—— (6R)-2-(cyclopropylmethyl)-8-(4-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N2O3
(6R)-2-(cyclopropylmethyl)-8-(4-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-aminopyridin-3-yl)-[(2R)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone —— C17H21N3OS
(6-aminopyridin-3-yl)-[(2R)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone
—— (6S)-6-[[cyclohexyl-[(1-methylpyrazol-4-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol —— C17H30N4O2
(6S)-6-[[cyclohexyl-[(1-methylpyrazol-4-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol
—— 6-chloro-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-2H-chromene-3-carboxamide —— C19H22ClNO4
6-chloro-N-[(4S)-1,9-dioxaspiro[5.5]undecan-4-yl]-2H-chromene-3-carboxamide
—— [(6R)-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methanol —— C14H23N3O2
[(6R)-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methanol
—— (6S)-2-(cyclopropylmethyl)-8-(4-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N2O3
(6S)-2-(cyclopropylmethyl)-8-(4-hydroxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[cyclohexyl-[(1-methylpyrazol-4-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol —— C17H30N4O2
(6R)-6-[[cyclohexyl-[(1-methylpyrazol-4-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol
—— (6S)-2-(2-methoxyethyl)-8-[3-(5-methylpyrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6S)-2-(2-methoxyethyl)-8-[3-(5-methylpyrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-chloro-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-2H-chromene-3-carboxamide —— C19H22ClNO4
6-chloro-N-[(4R)-1,9-dioxaspiro[5.5]undecan-4-yl]-2H-chromene-3-carboxamide
—— (6-aminopyridin-3-yl)-[(2S)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone —— C17H21N3OS
(6-aminopyridin-3-yl)-[(2S)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone
—— 6-[4-[3-[(2S)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]butanoyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one —— C21H28N6O3
6-[4-[3-[(2S)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]butanoyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one
—— (6R)-6-[[2-[(3-chlorophenyl)methylsulfanyl]ethylamino]methyl]-1,4-oxazepan-6-ol —— C15H23ClN2O2S
(6R)-6-[[2-[(3-chlorophenyl)methylsulfanyl]ethylamino]methyl]-1,4-oxazepan-6-ol
—— [(6S)-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methanol —— C14H23N3O2
[(6S)-4-(2-methyl-5-propylpyrimidin-4-yl)-1,4-oxazepan-6-yl]methanol
—— (6S)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6S)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6R)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-ethyl-8-[(4-methylphenyl)methylsulfonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N2O3S
(6R)-2-ethyl-8-[(4-methylphenyl)methylsulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6R)-2-(cyclopropylmethyl)-8-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methylsulfanylpyridin-3-yl)methanone —— C17H25N3O3S
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methylsulfanylpyridin-3-yl)methanone
—— 6-[(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C20H24N6O
6-[(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— 6-[(6S)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C20H26N4O
6-[(6S)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methylsulfanylpyridin-3-yl)methanone —— C17H25N3O3S
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methylsulfanylpyridin-3-yl)methanone
—— (6R)-6-[[2-[2-(methylsulfanylmethyl)-1,3-thiazol-4-yl]ethylamino]methyl]-1,4-oxazepan-6-ol —— C13H23N3O2S2
(6R)-6-[[2-[2-(methylsulfanylmethyl)-1,3-thiazol-4-yl]ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-2-(cyclopropylmethyl)-8-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O2
(6S)-2-(cyclopropylmethyl)-8-[[5-(1H-pyrazol-5-yl)furan-2-yl]methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile —— C20H24N6O
6-[(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-3-carbonitrile
—— (6S)-6-[[2-[2-(methylsulfanylmethyl)-1,3-thiazol-4-yl]ethylamino]methyl]-1,4-oxazepan-6-ol —— C13H23N3O2S2
(6S)-6-[[2-[2-(methylsulfanylmethyl)-1,3-thiazol-4-yl]ethylamino]methyl]-1,4-oxazepan-6-ol
—— 6-[(6R)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile —— C20H26N4O
6-[(6R)-2-cyclopentyl-3-oxo-2,8-diazaspiro[5.5]undecan-8-yl]pyridine-2-carbonitrile
—— (6S)-2-ethyl-8-[(4-methylphenyl)methylsulfonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N2O3S
(6S)-2-ethyl-8-[(4-methylphenyl)methylsulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(3-pyrazol-1-ylphenyl)methanone —— C20H26N4O3
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(3-pyrazol-1-ylphenyl)methanone
—— (6S)-2-(2-hydroxyethyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N2O4
(6S)-2-(2-hydroxyethyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(1R)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-3-methylsulfonylpyrazolo[1,5-a]pyrimidine —— C17H21N5O2S
6-[[(1R)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-3-methylsulfonylpyrazolo[1,5-a]pyrimidine
—— (6S)-8-(2,6-diaminopyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N8O
(6S)-8-(2,6-diaminopyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-N-[(2R)-2-hydroxy-3-piperazin-1-ylpropyl]-2-methylquinoline-4-carboxamide —— C20H28N4O2
6-ethyl-N-[(2R)-2-hydroxy-3-piperazin-1-ylpropyl]-2-methylquinoline-4-carboxamide
—— 6-[[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-3-methylsulfonylpyrazolo[1,5-a]pyrimidine —— C17H21N5O2S
6-[[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]methyl]-3-methylsulfonylpyrazolo[1,5-a]pyrimidine
—— (6R)-2-(2-hydroxyethyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N2O4
(6R)-2-(2-hydroxyethyl)-8-(7-methyl-1-benzofuran-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(2,6-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2
(6S)-8-[(2,6-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(2,6-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2
(6R)-8-[(2,6-dimethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-2-methyl-N-[(3S)-1-methyl-6-oxopiperidin-3-yl]quinoline-4-carboxamide —— C19H23N3O2
6-ethyl-2-methyl-N-[(3S)-1-methyl-6-oxopiperidin-3-yl]quinoline-4-carboxamide
—— (6R)-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O2
(6R)-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[4-(2-pyridin-2-ylethyl)piperazin-1-yl]methyl]-1,4-oxazepan-6-ol —— C17H28N4O2
(6S)-6-[[4-(2-pyridin-2-ylethyl)piperazin-1-yl]methyl]-1,4-oxazepan-6-ol
—— 6-ethyl-N-[(2S)-2-hydroxy-3-piperazin-1-ylpropyl]-2-methylquinoline-4-carboxamide —— C20H28N4O2
6-ethyl-N-[(2S)-2-hydroxy-3-piperazin-1-ylpropyl]-2-methylquinoline-4-carboxamide