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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-8-(2-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6S)-8-(2-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[2-(4-fluorophenoxy)ethyl]-1,4-oxazepan-6-ol —— C13H18FNO3
(6S)-4-[2-(4-fluorophenoxy)ethyl]-1,4-oxazepan-6-ol
—— (6S)-2-(cyclopropylmethyl)-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O
(6S)-2-(cyclopropylmethyl)-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methoxypyridin-4-yl)methanone —— C17H25N3O4
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methoxypyridin-4-yl)methanone
—— (6S)-3-oxo-N-propan-2-yl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C19H28N4O2
(6S)-3-oxo-N-propan-2-yl-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-7-ylmethanone —— C13H15N3O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-7-ylmethanone
—— [(6S)-4-[(4-chloro-1-methylindazol-3-yl)methyl]-1,4-oxazepan-6-yl]methanol —— C15H20ClN3O2
[(6S)-4-[(4-chloro-1-methylindazol-3-yl)methyl]-1,4-oxazepan-6-yl]methanol
—— 6-[(1R)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one —— C18H20N4O2S
6-[(1R)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[5-(imidazol-1-ylmethyl)furan-2-yl]methanone —— C19H26N4O4
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[5-(imidazol-1-ylmethyl)furan-2-yl]methanone
—— 6-[(2R)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C16H19N3O3S
6-[(2R)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (6R)-8-(3-imidazol-1-ylpropanoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6R)-8-(3-imidazol-1-ylpropanoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[6-(2-hydroxyethylamino)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N5O2
(6R)-2-(cyclopropylmethyl)-8-[6-(2-hydroxyethylamino)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[4-[3-[(2S)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]butanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one —— C21H26N6O3
6-[4-[3-[(2S)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]butanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one
—— (6S)-8-(3-imidazol-1-ylpropanoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6S)-8-(3-imidazol-1-ylpropanoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-chloro-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)-[(2S)-1-methylsulfonylpyrrolidin-2-yl]methanone —— C17H20ClN3O3S
(6-chloro-1,3,4,5-tetrahydropyrido[4,3-b]indol-2-yl)-[(2S)-1-methylsulfonylpyrrolidin-2-yl]methanone
—— (6R)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H26ClFN2O
(6R)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6R)-8-(2-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O2
(6R)-8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-Amino-3-methyl-1-(2-methylpropyl)-5-(2-pyrimidin-2-ylsulfanylacetyl)pyrimidine-2,4-dione —— C15H19N5O3S
6-Amino-3-methyl-1-(2-methylpropyl)-5-(2-pyrimidin-2-ylsulfanylacetyl)pyrimidine-2,4-dione
—— (6S)-8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O2
(6S)-8-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-2-cyclopentyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6R)-2-(3-methoxypropyl)-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O2
(6S)-2-(cyclopropylmethyl)-8-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6S)-2-(cyclopropylmethyl)-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-4-[(4-chloro-1-methylindazol-3-yl)methyl]-1,4-oxazepan-6-yl]methanol —— C15H20ClN3O2
[(6R)-4-[(4-chloro-1-methylindazol-3-yl)methyl]-1,4-oxazepan-6-yl]methanol
—— 6-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C16H19N3O3S
6-[(2S)-2-(2-thiophen-2-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— (6S)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H26ClFN2O
(6S)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-7-ylmethanone —— C13H15N3O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-7-ylmethanone
—— 6-ethyl-N,2-dimethyl-N-[3-[(2R)-oxolan-2-yl]propyl]quinoline-4-carboxamide —— C21H28N2O2
6-ethyl-N,2-dimethyl-N-[3-[(2R)-oxolan-2-yl]propyl]quinoline-4-carboxamide
—— 6-ethyl-N-[(1S)-2-hydroxy-1-(thian-4-yl)ethyl]-2-methylquinoline-4-carboxamide —— C20H26N2O2S
6-ethyl-N-[(1S)-2-hydroxy-1-(thian-4-yl)ethyl]-2-methylquinoline-4-carboxamide
—— (6S)-2-cyclopropyl-8-[[2-(2-hydroxyethoxy)phenyl]methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6S)-2-cyclopropyl-8-[[2-(2-hydroxyethoxy)phenyl]methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methoxypyridin-4-yl)methanone —— C17H25N3O4
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methoxypyridin-4-yl)methanone
—— (6R)-8-[(2,3-dichlorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24Cl2N2O2
(6R)-8-[(2,3-dichlorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H27N3O
(6S)-2-cyclopropyl-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone —— C13H19N3O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydropyrazolo[1,5-a]pyridin-3-yl)methanone
—— (6S)-8-(6-aminopyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N7O
(6S)-8-(6-aminopyrimidin-4-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one —— C18H20N4O2S
6-[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-3,5-dimethylthieno[2,3-d]pyrimidin-4-one
—— (6R)-4-[2-(2-ethylphenoxy)ethyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C20H32N2O3
(6R)-4-[2-(2-ethylphenoxy)ethyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— 6-[4-[3-[(2R)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]butanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one —— C21H26N6O3
6-[4-[3-[(2R)-1-methoxypropan-2-yl]imidazo[4,5-b]pyridin-2-yl]butanoyl]-2-methyl-5,7-dihydro-3H-pyrrolo[3,4-d]pyrimidin-4-one
—— 6-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C16H20N4O3
6-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6S)-2-(3-methoxypropyl)-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6S)-2-(3-methoxypropyl)-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-[6-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H24F3N3O2
(6R)-2-(2-methoxyethyl)-8-[6-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(2,3-dichlorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24Cl2N2O2
(6S)-8-[(2,3-dichlorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[2-(4-phenyl-1,3-thiazol-2-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C17H23N3O2S
(6R)-6-[[2-(4-phenyl-1,3-thiazol-2-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O
(6R)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O
(6S)-8-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[6-(2-hydroxyethylamino)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N5O2
(6S)-2-(cyclopropylmethyl)-8-[6-(2-hydroxyethylamino)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6R)-2-(cyclopropylmethyl)-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O2
(6S)-2-(cyclopropylmethyl)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopentyl-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N3O3
(6R)-2-cyclopentyl-8-(2-methoxypyridine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O2
(6R)-2-(cyclopropylmethyl)-8-[2-[methyl(pyridin-4-ylmethyl)amino]acetyl]-2,8-diazaspiro[5.5]undecan-3-one