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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-2-cyclopropyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N5O
(6S)-2-cyclopropyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(4-aminopyrimidin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H25N7O
(6S)-8-(4-aminopyrimidin-2-yl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26ClFN2O2
(6R)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[(2-methoxy-4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N2O3
(6S)-2-(2-methoxyethyl)-8-[(2-methoxy-4-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-4-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-1,4-oxazepan-6-yl]methanol —— C17H23N3O3
[(6R)-4-[[1-(4-methoxyphenyl)imidazol-2-yl]methyl]-1,4-oxazepan-6-yl]methanol
—— (6S)-2-(2-hydroxyethyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6S)-2-(2-hydroxyethyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-4,5,6,7-tetrahydroindazol-3-yl)methanone —— C15H23N3O3
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-4,5,6,7-tetrahydroindazol-3-yl)methanone
—— (6R)-2-(2-hydroxyethyl)-8-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N4O3
(6R)-2-(2-hydroxyethyl)-8-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(4-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24N2O4
(6R)-8-(4-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-(pyrimidin-2-ylsulfanylmethyl)furan-2-yl]methanone —— C16H19N3O4S
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-(pyrimidin-2-ylsulfanylmethyl)furan-2-yl]methanone
—— (6S)-2-(2-hydroxyethyl)-8-[2-(4-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4
(6S)-2-(2-hydroxyethyl)-8-[2-(4-hydroxyphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methylbutyl)-8-(2-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O2
(6S)-2-(3-methylbutyl)-8-(2-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone —— C17H26N2O4
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone
—— 6-chloro-2-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzothiazole —— C15H15ClN4S
6-chloro-2-[(3R)-3-(1H-imidazol-2-yl)piperidin-1-yl]-1,3-benzothiazole
—— 6-[(3S)-3-(imidazol-1-ylmethyl)piperidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one —— C17H19N5O2S
6-[(3S)-3-(imidazol-1-ylmethyl)piperidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one
—— (6S)-4-(4-phenoxybutyl)-1,4-oxazepan-6-ol —— C15H23NO3
(6S)-4-(4-phenoxybutyl)-1,4-oxazepan-6-ol
—— (6S)-6-[[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol —— C19H26N4O3
(6S)-6-[[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol
—— 6-[(3R)-3-(imidazol-1-ylmethyl)piperidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one —— C17H19N5O2S
6-[(3R)-3-(imidazol-1-ylmethyl)piperidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-(hydroxymethyl)-N-[[(3S)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]pyridine-2-carboxamide —— C17H21N5O3
6-(hydroxymethyl)-N-[[(3S)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]pyridine-2-carboxamide
—— (6S)-2-(cyclopropylmethyl)-8-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6S)-2-(cyclopropylmethyl)-8-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-(1-phenyltetrazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C17H24N6O2
(6S)-4-(1-phenyltetrazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-4-(1-phenyltetrazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C17H24N6O2
(6R)-4-(1-phenyltetrazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-6-[[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol —— C19H26N4O3
(6R)-6-[[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol
—— (6S)-2-(cyclopropylmethyl)-8-(8-methoxyquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H29N3O2
(6S)-2-(cyclopropylmethyl)-8-(8-methoxyquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(2,6-difluoro-4-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26F2N2O3
(6S)-8-[(2,6-difluoro-4-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone —— C17H26N2O4
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[5-[(4-methylpiperidin-1-yl)methyl]furan-2-yl]methanone
—— (6S)-8-(4-methylpyridin-2-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N4O
(6S)-8-(4-methylpyridin-2-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methylbutyl)-8-[3-(tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H30N6O2
(6S)-2-(3-methylbutyl)-8-[3-(tetrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[methyl-[(3-thiophen-2-yl-1H-pyrazol-5-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol —— C15H22N4O2S
(6R)-6-[[methyl-[(3-thiophen-2-yl-1H-pyrazol-5-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-4,5,6,7-tetrahydroindazol-3-yl)methanone —— C15H23N3O3
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-4,5,6,7-tetrahydroindazol-3-yl)methanone
—— (6S)-8-(5-chloropyridin-2-yl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24ClN3O
(6S)-8-(5-chloropyridin-2-yl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[methyl-[(3-thiophen-2-yl-1H-pyrazol-5-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol —— C15H22N4O2S
(6S)-6-[[methyl-[(3-thiophen-2-yl-1H-pyrazol-5-yl)methyl]amino]methyl]-1,4-oxazepan-6-ol
—— (6S)-6-[[2-(2H-triazol-4-ylsulfanyl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C10H19N5O2S
(6S)-6-[[2-(2H-triazol-4-ylsulfanyl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-8-(4-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24N2O4
(6S)-8-(4-hydroxybenzoyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N5O
(6R)-2-cyclopropyl-8-[4-(ethylamino)pyrimidin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methylbutyl)-8-(2-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O2
(6R)-2-(3-methylbutyl)-8-(2-methylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6R)-2-(cyclopropylmethyl)-8-[(5-methoxy-4-oxo-1H-pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]methanone —— C15H23N3O3S
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]methanone
—— (6R)-6-[[2-(2H-triazol-4-ylsulfanyl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C10H19N5O2S
(6R)-6-[[2-(2H-triazol-4-ylsulfanyl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-8-(4-methylpyridin-2-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H28N4O
(6R)-8-(4-methylpyridin-2-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-N-ethyl-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C18H26N4O2
(6R)-N-ethyl-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— (6R)-2-(cyclopropylmethyl)-8-[2-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O3
(6R)-2-(cyclopropylmethyl)-8-[2-(3-methyl-5-oxo-1,2-dihydropyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26ClFN2O2
(6S)-8-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(hydroxymethyl)-N-[[(3R)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]pyridine-2-carboxamide —— C17H21N5O3
6-(hydroxymethyl)-N-[[(3R)-1-(1-methyl-6-oxopyridazin-4-yl)pyrrolidin-3-yl]methyl]pyridine-2-carboxamide
—— (6R)-2-(2-hydroxyethyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6R)-2-(2-hydroxyethyl)-8-[4-(1H-pyrazol-4-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-N-ethyl-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C18H26N4O2
(6S)-N-ethyl-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-(pyrimidin-2-ylsulfanylmethyl)furan-2-yl]methanone —— C16H19N3O4S
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[5-(pyrimidin-2-ylsulfanylmethyl)furan-2-yl]methanone
—— (6S)-2-cyclopentyl-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O
(6S)-2-cyclopentyl-8-[(1-propan-2-ylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(2,2,2-trimethoxyethyl)-3H-1,3-benzoxazol-2-one —— C12H15NO5
6-(2,2,2-trimethoxyethyl)-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-2-amino-1-methoxypropan-2-yl]-4H-1,4-benzothiazin-3-one —— C12H16N2O2S
6-[(2R)-2-amino-1-methoxypropan-2-yl]-4H-1,4-benzothiazin-3-one