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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C19H30N4O2
(6S)-4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6S)-2-(cyclopropylmethyl)-8-(2-oxo-1,3-dihydroimidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H24N4O3
(6S)-2-(cyclopropylmethyl)-8-(2-oxo-1,3-dihydroimidazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethylamino]pyridine-3-carbonitrile —— C17H20N6O2
6-[2-[(2R)-4-(1-methyl-6-oxopyridazin-4-yl)morpholin-2-yl]ethylamino]pyridine-3-carbonitrile
—— (6R)-8-[3-(2-ethylimidazol-1-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O3
(6R)-8-[3-(2-ethylimidazol-1-yl)propanoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-2-(3-methoxyphenyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C19H19N3O3S
6-[(2R)-2-(3-methoxyphenyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 6-ethyl-2-methyl-N-[(1R)-2-methyl-1-(2-methyl-1,2,4-triazol-3-yl)propyl]quinoline-4-carboxamide —— C20H25N5O
6-ethyl-2-methyl-N-[(1R)-2-methyl-1-(2-methyl-1,2,4-triazol-3-yl)propyl]quinoline-4-carboxamide
—— (6R)-2-(2-hydroxyethyl)-8-[(2-methylnaphthalen-1-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C23H30N2O2
(6R)-2-(2-hydroxyethyl)-8-[(2-methylnaphthalen-1-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-4-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-1,4-oxazepan-6-yl]methanol —— C13H17F3N2O2
[(6R)-4-[[6-(trifluoromethyl)pyridin-3-yl]methyl]-1,4-oxazepan-6-yl]methanol
—— (6R)-N-cyclopentyl-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C21H30N4O2
(6R)-N-cyclopentyl-3-oxo-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— (6R)-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H33N5O2
(6R)-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-3-hydroxybutyl]sulfamoyl]-N-propyl-3,4-dihydro-1H-isoquinoline-2-carboxamide —— C17H27N3O4S
6-[[(3R)-3-hydroxybutyl]sulfamoyl]-N-propyl-3,4-dihydro-1H-isoquinoline-2-carboxamide
—— (6R)-2-(2-methoxyethyl)-8-[(1-propylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H32N4O2
(6R)-2-(2-methoxyethyl)-8-[(1-propylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H33N5O2
(6S)-8-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-2-methylquinolin-4-yl)-[(2S)-2-(1-methylpyrazol-3-yl)piperidin-1-yl]methanone —— C22H26N4O
(6-ethyl-2-methylquinolin-4-yl)-[(2S)-2-(1-methylpyrazol-3-yl)piperidin-1-yl]methanone
—— 6-[(2S)-2-(3-methoxyphenyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C19H19N3O3S
6-[(2S)-2-(3-methoxyphenyl)piperidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6R)-N-tert-butyl-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C20H30N4O2
(6R)-N-tert-butyl-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— 6-methyl-5-[(2S)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile —— C20H22N4O2
6-methyl-5-[(2S)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile
—— (6R)-2-(2-hydroxyethyl)-8-[(2,4,6-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H23F3N2O2
(6R)-2-(2-hydroxyethyl)-8-[(2,4,6-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-5-[(2R)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile —— C20H22N4O2
6-methyl-5-[(2R)-2-methyl-4-(2-methylphenyl)piperazine-1-carbonyl]-2-oxo-1H-pyridine-3-carbonitrile
—— 6-ethyl-2-methyl-N-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide —— C18H20N4O2
6-ethyl-2-methyl-N-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide
—— (6S)-8-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O
(6S)-8-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-2-methylquinolin-4-yl)-[(2R)-2-(1-methylpyrazol-3-yl)piperidin-1-yl]methanone —— C22H26N4O
(6-ethyl-2-methylquinolin-4-yl)-[(2R)-2-(1-methylpyrazol-3-yl)piperidin-1-yl]methanone
—— (6S)-8-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N5O2
(6S)-8-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]methanone —— C17H22F3N3O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl]methanone
—— (6S)-8-(3-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6S)-8-(3-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H34N4O
(6R)-8-[(2-ethylpyrimidin-5-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-3-hydroxy-3-methylpiperidin-1-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide —— C20H25N5O3S
6-[[(3R)-3-hydroxy-3-methylpiperidin-1-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-6-[[(2-phenyl-1,3-oxazol-4-yl)methylamino]methyl]-1,4-oxazepan-6-ol —— C16H21N3O3
(6R)-6-[[(2-phenyl-1,3-oxazol-4-yl)methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-6-[[(3,5-dimethyl-1,2-oxazol-4-yl)methyl-methylamino]methyl]-1,4-oxazepan-6-ol —— C13H23N3O3
(6S)-6-[[(3,5-dimethyl-1,2-oxazol-4-yl)methyl-methylamino]methyl]-1,4-oxazepan-6-ol
—— 6-[(3S)-3-[(2-methylimidazol-1-yl)methyl]piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C19H21N5O3
6-[(3S)-3-[(2-methylimidazol-1-yl)methyl]piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione
—— (6S)-2-(2-methoxyethyl)-8-[2-(2-oxopyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O4
(6S)-2-(2-methoxyethyl)-8-[2-(2-oxopyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-quinolin-4-yl-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N3O2
(6S)-2-(3-methoxypropyl)-8-quinolin-4-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[(2-phenyl-1,3-oxazol-4-yl)methylamino]methyl]-1,4-oxazepan-6-ol —— C16H21N3O3
(6S)-6-[[(2-phenyl-1,3-oxazol-4-yl)methylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-8-[3-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6R)-8-[3-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-(2-ethylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O2
(6R)-2-butyl-8-(2-ethylpyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(2,4-dimethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O4
(6S)-8-[(2,4-dimethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-hydroxyethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C16H23N3O3
(6R)-2-(2-hydroxyethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2S)-2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]sulfonyl-3H-1,3-benzothiazol-2-one —— C16H21N3O4S2
6-[(2S)-2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]sulfonyl-3H-1,3-benzothiazol-2-one
—— (6R)-2-(3-methoxypropyl)-8-quinolin-4-yl-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N3O2
(6R)-2-(3-methoxypropyl)-8-quinolin-4-yl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopentyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O3
(6R)-2-cyclopentyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6R)-2-butyl-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-2-methyl-N-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide —— C18H20N4O2
6-ethyl-2-methyl-N-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]quinoline-4-carboxamide
—— (6R)-2-(2-methoxyethyl)-8-[(2-methylsulfanylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2S
(6R)-2-(2-methoxyethyl)-8-[(2-methylsulfanylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(3-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24ClFN2O2
(6R)-8-[(3-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6-aminopyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H27N5O2
(6S)-8-(6-aminopyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(3R)-3-[(2-methylimidazol-1-yl)methyl]piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C19H21N5O3
6-[(3R)-3-[(2-methylimidazol-1-yl)methyl]piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione
—— (6S)-8-[(3-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24ClFN2O2
(6S)-8-[(3-chloro-4-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(1-ethylindol-6-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H31N3O2
(6S)-8-[(1-ethylindol-6-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(1-ethylbenzimidazol-2-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6S)-8-[(1-ethylbenzimidazol-2-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-2-methyl-N-[(3R)-2-oxopyrrolidin-3-yl]quinoline-4-carboxamide —— C17H19N3O2
6-ethyl-2-methyl-N-[(3R)-2-oxopyrrolidin-3-yl]quinoline-4-carboxamide