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—— (6S)-2-(3-methoxypropyl)-8-(2-pyrimidin-2-ylsulfanylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O3S
(6S)-2-(3-methoxypropyl)-8-(2-pyrimidin-2-ylsulfanylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(4R,8aS)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole —— C14H18N4
6-[(4R,8aS)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole
—— 6-[(4R,8aR)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole —— C14H18N4
6-[(4R,8aR)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole
—— 6-chloro-N-[[(6R)-1,4-oxazepan-6-yl]methyl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide —— C11H15ClN4O3S2
6-chloro-N-[[(6R)-1,4-oxazepan-6-yl]methyl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
—— 6-chloro-N-[[(6S)-1,4-oxazepan-6-yl]methyl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide —— C11H15ClN4O3S2
6-chloro-N-[[(6S)-1,4-oxazepan-6-yl]methyl]imidazo[2,1-b][1,3]thiazole-5-sulfonamide
—— 6-[(4S,8aS)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole —— C14H18N4
6-[(4S,8aS)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole
—— (6R)-8-(2-aminopyridine-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O3
(6R)-8-(2-aminopyridine-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-hex-5-enyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O
(6R)-8-hex-5-enyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(3-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-hex-5-enyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N4O
(6S)-8-hex-5-enyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(1-methyl-3-phenylthieno[2,3-c]pyrazol-5-yl)methanone —— C18H19N3O3S
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(1-methyl-3-phenylthieno[2,3-c]pyrazol-5-yl)methanone
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(1-methyl-3-phenylthieno[2,3-c]pyrazol-5-yl)methanone —— C18H19N3O3S
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(1-methyl-3-phenylthieno[2,3-c]pyrazol-5-yl)methanone
—— (6R)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H29N5O
(6R)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-(spiro[indene-1,4'-piperidine]-1'-ylmethyl)-1,4-oxazepan-6-ol —— C19H26N2O2
(6R)-6-(spiro[indene-1,4'-piperidine]-1'-ylmethyl)-1,4-oxazepan-6-ol
—— (6S)-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4OS
(6S)-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-(spiro[indene-1,4'-piperidine]-1'-ylmethyl)-1,4-oxazepan-6-ol —— C19H26N2O2
(6S)-6-(spiro[indene-1,4'-piperidine]-1'-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4OS
(6R)-8-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C23H29N5O
(6S)-8-(6,7-dihydro-5H-cyclopenta[d]pyrimidin-4-yl)-2-(2-pyridin-2-ylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O
(6R)-2-butyl-8-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(4S,8aR)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole —— C14H18N4
6-[(4S,8aR)-1,2,3,4,6,7,8,8a-octahydropyrrolo[1,2-a]pyrazin-4-yl]-1H-benzimidazole
—— (6S)-2-cyclopropyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O3
(6S)-2-cyclopropyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopentyl-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O
(6S)-2-cyclopentyl-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopentyl-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O
(6R)-2-cyclopentyl-8-(2,6-dimethylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethylamino)methyl]-1,4-oxazepan-6-ol —— C14H22N4O2
(6S)-6-[(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethylamino)methyl]-1,4-oxazepan-6-ol
—— (6R)-2-cyclopropyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H26N4O3
(6R)-2-cyclopropyl-8-[5-(pyrazol-1-ylmethyl)furan-2-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-[(2-methoxy-3,5-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N2O3
(6S)-2-(2-hydroxyethyl)-8-[(2-methoxy-3,5-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-(2-aminopyridine-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O3
(6S)-8-(2-aminopyridine-4-carbonyl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethylamino)methyl]-1,4-oxazepan-6-ol —— C14H22N4O2
(6R)-6-[(6,7-dihydro-5H-cyclopenta[d]pyrimidin-2-ylmethylamino)methyl]-1,4-oxazepan-6-ol
—— (6S)-2-butyl-8-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H32N4O
(6S)-2-butyl-8-[(2-methylimidazo[1,2-a]pyridin-3-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[4-[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H21N3O3
6-[4-[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6R)-2-(2-hydroxyethyl)-8-[(2-methoxy-3,5-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H32N2O3
(6R)-2-(2-hydroxyethyl)-8-[(2-methoxy-3,5-dimethylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-methyl-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H25N5O2
(6R)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-methyl-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-(4-methoxyphenoxy)acetate —— C21H20O7
(6-Ethyl-7-hydroxy-2-oxochromen-4-yl)methyl 2-(4-methoxyphenoxy)acetate
—— 6-[4-[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one —— C17H21N3O3
6-[4-[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-6-methyl-1H-pyrimidin-2-ylidene]cyclohexa-2,4-dien-1-one
—— (6S)-2-(2-hydroxyethyl)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O3S
(6S)-2-(2-hydroxyethyl)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-5-phenylpyrrol-2-yl)methanone —— C18H22N2O3
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-5-phenylpyrrol-2-yl)methanone
—— (6R)-2-(2-hydroxyethyl)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N3O3S
(6R)-2-(2-hydroxyethyl)-8-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[[4-(2-phenylethyl)-1,2,4-triazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol —— C17H25N5O2
(6S)-6-[[[4-(2-phenylethyl)-1,2,4-triazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-methyl-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide —— C20H25N5O2
(6S)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-methyl-3-oxo-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
—— (6R)-6-[[[4-(2-phenylethyl)-1,2,4-triazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol —— C17H25N5O2
(6R)-6-[[[4-(2-phenylethyl)-1,2,4-triazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-5-phenylpyrrol-2-yl)methanone —— C18H22N2O3
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1-methyl-5-phenylpyrrol-2-yl)methanone
—— (6R)-2-(2-hydroxyethyl)-8-[3-(4-methylphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6R)-2-(2-hydroxyethyl)-8-[3-(4-methylphenyl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethylamino)methyl]-1,4-oxazepan-6-ol —— C15H24N2O2S
(6R)-6-[(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethylamino)methyl]-1,4-oxazepan-6-ol
—— (6R)-2-(2-hydroxyethyl)-8-(7-methylthieno[3,2-d]pyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24N4O2S
(6R)-2-(2-hydroxyethyl)-8-(7-methylthieno[3,2-d]pyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N2O2
(6S)-2-cyclopropyl-8-[(4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-hydroxypropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O2
(6R)-8-(3-hydroxypropyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-(7-methylthieno[3,2-d]pyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24N4O2S
(6S)-2-(2-hydroxyethyl)-8-(7-methylthieno[3,2-d]pyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-N,N-dimethyl-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-sulfonamide —— C17H26N4O3S
(6S)-N,N-dimethyl-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-sulfonamide
—— 6-[(3S)-3-(3-phenylpropanoyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C19H21N3O4
6-[(3S)-3-(3-phenylpropanoyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-[(2S)-2-(2-pyrrolidin-1-ylethyl)piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C20H26N4O3
6-[(2S)-2-(2-pyrrolidin-1-ylethyl)piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione