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中文名称 英文名称 CAS号 化学式 结构式图片
—— (6S)-2-butyl-8-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N3O2
(6S)-2-butyl-8-[(3,5-dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-[(1,3-dimethylpyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H32N4O
(6R)-2-butyl-8-[(1,3-dimethylpyrazol-4-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(2-ethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2
(6R)-8-[(2-ethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2S)-1-[(1-propylimidazol-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C19H25N5
6-methyl-2-[(2S)-1-[(1-propylimidazol-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6R)-8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N4O2S
(6R)-8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[[1-(benzenesulfonyl)piperidin-4-yl]amino]methyl]-1,4-oxazepan-6-ol —— C17H27N3O4S
(6S)-6-[[[1-(benzenesulfonyl)piperidin-4-yl]amino]methyl]-1,4-oxazepan-6-ol
—— (6S)-8-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one —— C20H33N5O
(6S)-8-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]-2-propan-2-yl-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2R)-1-[(1-propylimidazol-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C19H25N5
6-methyl-2-[(2R)-1-[(1-propylimidazol-2-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-8-[(2-ethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2
(6S)-8-[(2-ethylphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-3-ylmethanone —— C18H24N4O3
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-3-ylmethanone
—— 6-methyl-2-[(3R)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-benzothiazole —— C19H21N3OS
6-methyl-2-[(3R)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-benzothiazole
—— 6-[2-[2-aminoethyl(methyl)amino]ethyl]-3,4-dihydro-1H-quinolin-2-one —— C14H21N3O
6-[2-[2-aminoethyl(methyl)amino]ethyl]-3,4-dihydro-1H-quinolin-2-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-3-ylmethanone —— C18H24N4O3
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-pyrazolo[1,5-a]pyridin-3-ylmethanone
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(5-phenoxyfuran-2-yl)methanone —— C17H19NO5
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(5-phenoxyfuran-2-yl)methanone
—— 6-methyl-2-[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-benzothiazole —— C19H21N3OS
6-methyl-2-[(3S)-3-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,3-benzothiazole
—— 6-[(1R)-1-amino-2-pyrrolidin-1-ylethyl]-3H-1,3-benzoxazol-2-one —— C13H17N3O2
6-[(1R)-1-amino-2-pyrrolidin-1-ylethyl]-3H-1,3-benzoxazol-2-one
—— 6-[(1S)-3-oxocyclopentyl]-4H-1,4-benzothiazin-3-one —— C13H13NO2S
6-[(1S)-3-oxocyclopentyl]-4H-1,4-benzothiazin-3-one
—— 6-[(1S)-1-amino-2-pyrrolidin-1-ylethyl]-3H-1,3-benzoxazol-2-one —— C13H17N3O2
6-[(1S)-1-amino-2-pyrrolidin-1-ylethyl]-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-3-[(2-fluorophenyl)methoxy]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one —— C17H16FN3O3
6-[(2R)-3-[(2-fluorophenyl)methoxy]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2R)-1-aminopiperidin-2-yl]-4H-1,4-benzoxazin-3-one —— C13H17N3O2
6-[(2R)-1-aminopiperidin-2-yl]-4H-1,4-benzoxazin-3-one
—— 6-[2-[(6-nitro-1,3-benzothiazol-2-yl)sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one —— C17H11N3O5S2
6-[2-[(6-nitro-1,3-benzothiazol-2-yl)sulfanyl]acetyl]-4H-1,4-benzoxazin-3-one
—— 6-[[(2S)-2-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one —— C13H17N3O2
6-[[(2S)-2-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-1-aminopiperidin-2-yl]-3-methyl-1,3-benzoxazol-2-one —— C13H17N3O2
6-[(2R)-1-aminopiperidin-2-yl]-3-methyl-1,3-benzoxazol-2-one
—— 6-[(2R)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]pyrido[2,3-d]pyridazin-5-one —— C16H22N4O2
6-[(2R)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-2-(4-bromophenyl)-2-hydroxyethyl]pyrido[2,3-d]pyridazin-5-one —— C15H12BrN3O2
6-[(2S)-2-(4-bromophenyl)-2-hydroxyethyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-1-aminopyrrolidin-2-yl]-4-methyl-1,4-benzoxazin-3-one —— C13H17N3O2
6-[(2S)-1-aminopyrrolidin-2-yl]-4-methyl-1,4-benzoxazin-3-one
—— 6-[[(2R)-2-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one —— C13H17N3O2
6-[[(2R)-2-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-1-aminopyrrolidin-2-yl]-4-methyl-1,4-benzoxazin-3-one —— C13H17N3O2
6-[(2R)-1-aminopyrrolidin-2-yl]-4-methyl-1,4-benzoxazin-3-one
—— 6-[(2R)-2-hydroxy-3-phenylmethoxypropyl]pyrido[2,3-d]pyridazin-5-one —— C17H17N3O3
6-[(2R)-2-hydroxy-3-phenylmethoxypropyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(4R)-4-(aminomethyl)-2-oxopyrrolidin-1-yl]-3H-1,3-benzoxazol-2-one —— C12H13N3O3
6-[(4R)-4-(aminomethyl)-2-oxopyrrolidin-1-yl]-3H-1,3-benzoxazol-2-one
—— 6-[(4S)-4-(aminomethyl)-2-oxopyrrolidin-1-yl]-3H-1,3-benzoxazol-2-one —— C12H13N3O3
6-[(4S)-4-(aminomethyl)-2-oxopyrrolidin-1-yl]-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-3-[benzyl(methyl)amino]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one —— C18H20N4O2
6-[(2R)-3-[benzyl(methyl)amino]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-2-hydroxy-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propyl]pyrido[2,3-d]pyridazin-5-one —— C20H21N3O3
6-[(2S)-2-hydroxy-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-1-aminopiperidin-2-yl]-4H-1,4-benzoxazin-3-one —— C13H17N3O2
6-[(2S)-1-aminopiperidin-2-yl]-4H-1,4-benzoxazin-3-one
—— 6-[(2S)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]pyrido[2,3-d]pyridazin-5-one —— C16H22N4O2
6-[(2S)-2-hydroxy-3-(4-methylpiperidin-1-yl)propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-1-aminopiperidin-2-yl]-3-methyl-1,3-benzoxazol-2-one —— C13H17N3O2
6-[(2S)-1-aminopiperidin-2-yl]-3-methyl-1,3-benzoxazol-2-one
—— 6-[(2S)-2-hydroxy-3-(2-propan-2-ylphenoxy)propyl]pyrido[2,3-d]pyridazin-5-one —— C19H21N3O3
6-[(2S)-2-hydroxy-3-(2-propan-2-ylphenoxy)propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-3-[benzyl(methyl)amino]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one —— C18H20N4O2
6-[(2S)-3-[benzyl(methyl)amino]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2R)-2-(4-bromophenyl)-2-hydroxyethyl]pyrido[2,3-d]pyridazin-5-one —— C15H12BrN3O2
6-[(2R)-2-(4-bromophenyl)-2-hydroxyethyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-3-[(2-fluorophenyl)methoxy]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one —— C17H16FN3O3
6-[(2S)-3-[(2-fluorophenyl)methoxy]-2-hydroxypropyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[(2S)-2-hydroxy-3-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propyl]pyrido[2,3-d]pyridazin-5-one —— C20H21N3O3
6-[(2S)-2-hydroxy-3-[[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[[(3S)-3-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one —— C13H17N3O2
6-[[(3S)-3-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-2-hydroxy-3-(2-propan-2-ylphenoxy)propyl]pyrido[2,3-d]pyridazin-5-one —— C19H21N3O3
6-[(2R)-2-hydroxy-3-(2-propan-2-ylphenoxy)propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[[(3R)-3-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one —— C13H17N3O2
6-[[(3R)-3-methylpiperazin-1-yl]methyl]-3H-1,3-benzoxazol-2-one
—— 6-[(2R)-2-hydroxy-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propyl]pyrido[2,3-d]pyridazin-5-one —— C20H21N3O3
6-[(2R)-2-hydroxy-3-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]oxy]propyl]pyrido[2,3-d]pyridazin-5-one
—— 6-[[Cyclopropyl-[(4-propan-2-ylphenyl)methyl]amino]methyl]-1,3,5-triazine-2,4-diamine —— C17H24N6
6-[[Cyclopropyl-[(4-propan-2-ylphenyl)methyl]amino]methyl]-1,3,5-triazine-2,4-diamine
—— (6R)-2-cyclopentyl-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N2O3
(6R)-2-cyclopentyl-8-(3-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(6,8-Dichloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine —— C10H8Cl2N8S
6-[(6,8-Dichloro-[1,2,4]triazolo[4,3-a]pyridin-3-yl)sulfanylmethyl]-1,3,5-triazine-2,4-diamine
—— 6-[[(4R)-4-amino-2-oxopyrrolidin-1-yl]methyl]-3H-1,3-benzoxazol-2-one —— C12H13N3O3
6-[[(4R)-4-amino-2-oxopyrrolidin-1-yl]methyl]-3H-1,3-benzoxazol-2-one
—— (6R)-8-(2,6-dimethylpyridin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H29N5O
(6R)-8-(2,6-dimethylpyridin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one