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中文名称 英文名称 CAS号 化学式 结构式图片
—— 6-[(2R)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C17H18N4O5
6-[(2R)-4-(4-methoxyphenyl)-2-methyl-3-oxopiperazine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-methyl-2-[(2R)-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C20H25N5
6-methyl-2-[(2R)-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— 6-[[(3R)-3-(aminomethyl)pyrrolidin-1-yl]methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1H-pyridine-3-carboxamide —— C19H25N5O4S
6-[[(3R)-3-(aminomethyl)pyrrolidin-1-yl]methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1H-pyridine-3-carboxamide
—— [6-[(6R)-6-hydroxy-1,4-oxazepan-4-yl]pyrazin-2-yl]-morpholin-4-ylmethanone —— C14H20N4O4
[6-[(6R)-6-hydroxy-1,4-oxazepan-4-yl]pyrazin-2-yl]-morpholin-4-ylmethanone
—— (6R)-2-(cyclopropylmethyl)-8-[1-(2-hydroxyethyl)benzimidazol-2-yl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O2
(6R)-2-(cyclopropylmethyl)-8-[1-(2-hydroxyethyl)benzimidazol-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[(4-propan-2-ylthiadiazol-5-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C16H28N4O2S
(6R)-4-[(4-propan-2-ylthiadiazol-5-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6S)-6-[[2-phenylethyl(pyridin-2-ylmethyl)amino]methyl]-1,4-oxazepan-6-ol —— C20H27N3O2
(6S)-6-[[2-phenylethyl(pyridin-2-ylmethyl)amino]methyl]-1,4-oxazepan-6-ol
—— (6R)-8-but-3-enoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6R)-8-but-3-enoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2S)-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C20H25N5
6-methyl-2-[(2S)-1-[(2-propan-2-ylpyrimidin-4-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-6-[[(5-chloro-1-benzothiophen-3-yl)methylamino]methyl]-1,4-oxazepan-6-ol —— C15H19ClN2O2S
(6S)-6-[[(5-chloro-1-benzothiophen-3-yl)methylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O
(6R)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-(3-pyrazol-1-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6S)-2-(2-methoxyethyl)-8-(3-pyrazol-1-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-but-3-enoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6S)-8-but-3-enoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-(3-pyrazol-1-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O3
(6R)-2-(2-methoxyethyl)-8-(3-pyrazol-1-ylpropanoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopentyl-8-[(5-methoxy-4-oxopyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O4
(6R)-2-cyclopentyl-8-[(5-methoxy-4-oxopyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol —— C17H27N3O3
(6S)-6-[[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol
—— (6R)-6-[[(5-chloro-1-benzothiophen-3-yl)methylamino]methyl]-1,4-oxazepan-6-ol —— C15H19ClN2O2S
(6R)-6-[[(5-chloro-1-benzothiophen-3-yl)methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H27N5O
(6S)-2-[2-(1H-imidazol-5-yl)ethyl]-8-(5-methylpyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[(4-propan-2-ylthiadiazol-5-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C16H28N4O2S
(6S)-4-[(4-propan-2-ylthiadiazol-5-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-6-[[2-phenylethyl(pyridin-2-ylmethyl)amino]methyl]-1,4-oxazepan-6-ol —— C20H27N3O2
(6R)-6-[[2-phenylethyl(pyridin-2-ylmethyl)amino]methyl]-1,4-oxazepan-6-ol
—— (6-ethyl-2-methylquinolin-4-yl)-[(3R)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methanone —— C23H28N4O
(6-ethyl-2-methylquinolin-4-yl)-[(3R)-3-[(2-methylimidazol-1-yl)methyl]piperidin-1-yl]methanone
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(1-phenyltriazol-4-yl)methanone —— C14H16N4O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(1-phenyltriazol-4-yl)methanone
—— [6-[(6S)-6-hydroxy-1,4-oxazepan-4-yl]pyrazin-2-yl]-morpholin-4-ylmethanone —— C14H20N4O4
[6-[(6S)-6-hydroxy-1,4-oxazepan-4-yl]pyrazin-2-yl]-morpholin-4-ylmethanone
—— (6S)-2-cyclopentyl-8-[(5-methoxy-4-oxopyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O4
(6S)-2-cyclopentyl-8-[(5-methoxy-4-oxopyran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3S)-3-(aminomethyl)pyrrolidin-1-yl]methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1H-pyridine-3-carboxamide —— C19H25N5O4S
6-[[(3S)-3-(aminomethyl)pyrrolidin-1-yl]methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1H-pyridine-3-carboxamide
—— (6R)-8-butanoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6R)-8-butanoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-butanoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H28N4O2
(6S)-8-butanoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[(1-methylindol-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H31N3O2
(6S)-2-(2-methoxyethyl)-8-[(1-methylindol-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[[3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl]methyl]-1,4-oxazepan-6-ol —— C16H17F3N2O4
(6R)-4-[[3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl]methyl]-1,4-oxazepan-6-ol
—— (6S)-4-[[3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl]methyl]-1,4-oxazepan-6-ol —— C16H17F3N2O4
(6S)-4-[[3-[2-(trifluoromethoxy)phenyl]-1,2-oxazol-5-yl]methyl]-1,4-oxazepan-6-ol
—— (6R)-6-[[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol —— C17H27N3O3
(6R)-6-[[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl]-1,4-oxazepan-6-ol
—— 6-[(3S)-3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione —— C17H17N5O3
6-[(3S)-3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-1,4-dihydroquinoxaline-2,3-dione
—— (6R)-2-(2-methoxyethyl)-8-[(1-methylindol-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H31N3O2
(6R)-2-(2-methoxyethyl)-8-[(1-methylindol-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(1-phenyltriazol-4-yl)methanone —— C14H16N4O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(1-phenyltriazol-4-yl)methanone
—— 6-methyl-4-[(2S)-2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-quinolin-2-one —— C21H27N3O3
6-methyl-4-[(2S)-2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1H-quinolin-2-one
—— (6R)-8-(2-aminopyridine-4-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6R)-8-(2-aminopyridine-4-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1,4-oxazepan-6-ol —— C13H23N3O2
(6S)-4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1,4-oxazepan-6-ol
—— (6S)-8-(2-aminopyridine-4-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N4O2
(6S)-8-(2-aminopyridine-4-carbonyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-2-methylquinolin-4-yl)-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone —— C21H23N3O2
(6-ethyl-2-methylquinolin-4-yl)-[(2S)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone
—— (6R)-4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1,4-oxazepan-6-ol —— C13H23N3O2
(6R)-4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1,4-oxazepan-6-ol
—— (6S)-2-cyclopropyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24N4O3
(6S)-2-cyclopropyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6-ethyl-2-methylquinolin-4-yl)-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone —— C21H23N3O2
(6-ethyl-2-methylquinolin-4-yl)-[(2R)-2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methanone
—— (6S)-N,N-dimethyl-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-sulfonamide —— C17H26N4O3S
(6S)-N,N-dimethyl-3-oxo-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-sulfonamide
—— (6R)-2-(2-hydroxyethyl)-8-(2,3,4-trifluorobenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H21F3N2O3
(6R)-2-(2-hydroxyethyl)-8-(2,3,4-trifluorobenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-cyclopropyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H24N4O3
(6R)-2-cyclopropyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-ethoxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O3
(6R)-8-(3-ethoxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[[(3R)-3-aminopyrrolidin-1-yl]methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1H-pyridine-3-carboxamide —— C18H23N5O4S
6-[[(3R)-3-aminopyrrolidin-1-yl]methyl]-2-oxo-N-[(4-sulfamoylphenyl)methyl]-1H-pyridine-3-carboxamide
—— (6S)-2-cyclopentyl-8-(5-oxo-1,2-dihydropyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H26N4O3
(6S)-2-cyclopentyl-8-(5-oxo-1,2-dihydropyrazole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-aminopyrimidin-4-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N5O
(6R)-8-(6-aminopyrimidin-4-yl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-(4-hydroxy-3-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N2O4
(6S)-2-(cyclopropylmethyl)-8-(4-hydroxy-3-methoxybenzoyl)-2,8-diazaspiro[5.5]undecan-3-one