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—— 6-[[(3S)-3-hydroxy-3-methylpiperidin-1-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide —— C20H25N5O3S
6-[[(3S)-3-hydroxy-3-methylpiperidin-1-yl]methyl]-N-[(2-methylimidazo[2,1-b][1,3]thiazol-6-yl)methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6R)-4-(2-phenylquinazolin-4-yl)-1,4-oxazepan-6-ol —— C19H19N3O2
(6R)-4-(2-phenylquinazolin-4-yl)-1,4-oxazepan-6-ol
—— (6R)-8-[(1-ethylindol-6-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H31N3O2
(6R)-8-[(1-ethylindol-6-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-aminopyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H27N5O2
(6R)-8-(6-aminopyrimidin-4-yl)-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-[(2,4,6-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H23F3N2O2
(6S)-2-(2-hydroxyethyl)-8-[(2,4,6-trifluorophenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-N-tert-butyl-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide —— C20H30N4O2
(6S)-N-tert-butyl-3-oxo-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-8-carboxamide
—— (6S)-8-[3-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6S)-8-[3-(dimethylamino)benzoyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-[2-(2-oxopyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O4
(6R)-2-(2-methoxyethyl)-8-[2-(2-oxopyridin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O3
(6R)-2-butyl-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(3-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H29FN2O2
(6R)-8-(3-fluorobenzoyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopentyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O3
(6S)-2-cyclopentyl-8-(2-methyl-6-oxo-1H-pyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(2,4-dimethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O4
(6R)-8-[(2,4-dimethoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O3
(6S)-2-butyl-8-(2-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C16H23N3O3
(6S)-2-(2-hydroxyethyl)-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N5O3
(6S)-8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-butyl-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H32N4O2
(6S)-2-butyl-8-[3-(2-methylimidazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(1-ethylbenzimidazol-2-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6R)-8-[(1-ethylbenzimidazol-2-yl)methyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2R)-1-[(2-pyrrolidin-1-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C21H26N6
6-methyl-2-[(2R)-1-[(2-pyrrolidin-1-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— 6-[[(3R)-3-hydroxypyrrolidin-3-yl]methyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one —— C12H20N4O2
6-[[(3R)-3-hydroxypyrrolidin-3-yl]methyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one
—— (6R)-8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H27N5O3
(6R)-8-[2-(ethylamino)pyrimidine-5-carbonyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]sulfonyl-3H-1,3-benzothiazol-2-one —— C16H21N3O4S2
6-[(2R)-2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]sulfonyl-3H-1,3-benzothiazol-2-one
—— (6R)-8-[2-(dimethylamino)ethyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H33N3O
(6R)-8-[2-(dimethylamino)ethyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-ethyl-2-methyl-N-[(3S)-2-oxopyrrolidin-3-yl]quinoline-4-carboxamide —— C17H19N3O2
6-ethyl-2-methyl-N-[(3S)-2-oxopyrrolidin-3-yl]quinoline-4-carboxamide
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methanone —— C20H28N2O5
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methanone
—— (6R)-6-[[(3,5-dimethyl-1,2-oxazol-4-yl)methyl-methylamino]methyl]-1,4-oxazepan-6-ol —— C13H23N3O3
(6R)-6-[[(3,5-dimethyl-1,2-oxazol-4-yl)methyl-methylamino]methyl]-1,4-oxazepan-6-ol
—— [6-(hydroxymethyl)pyridin-2-yl]-[(2R)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone —— C18H22N2O2S
[6-(hydroxymethyl)pyridin-2-yl]-[(2R)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone
—— 6-[[(3S)-3-hydroxypyrrolidin-3-yl]methyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one —— C12H20N4O2
6-[[(3S)-3-hydroxypyrrolidin-3-yl]methyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N6O
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[(2-methylsulfanylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N2O2S
(6S)-2-(2-methoxyethyl)-8-[(2-methylsulfanylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N6O
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(1H-pyrazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [6-(hydroxymethyl)pyridin-2-yl]-[(2S)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone —— C18H22N2O2S
[6-(hydroxymethyl)pyridin-2-yl]-[(2S)-2-(2-thiophen-2-ylethyl)piperidin-1-yl]methanone
—— (6R)-2-cyclopropyl-8-(4-methyl-2-propan-2-ylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N4O2
(6R)-2-cyclopropyl-8-(4-methyl-2-propan-2-ylpyrimidine-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— 6-methyl-2-[(2S)-1-[(2-pyrrolidin-1-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole —— C21H26N6
6-methyl-2-[(2S)-1-[(2-pyrrolidin-1-ylpyrimidin-5-yl)methyl]pyrrolidin-2-yl]-1H-benzimidazole
—— (6S)-4-(2-phenylquinazolin-4-yl)-1,4-oxazepan-6-ol —— C19H19N3O2
(6S)-4-(2-phenylquinazolin-4-yl)-1,4-oxazepan-6-ol
—— 6-methyl-5-[[4-[(1S)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]methyl]quinoline —— C23H34N4
6-methyl-5-[[4-[(1S)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]methyl]quinoline
—— (6R)-4-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol —— C18H23FN4O2
(6R)-4-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methanone —— C20H28N2O5
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methanone
—— (6S)-8-[2-(dimethylamino)ethyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H33N3O
(6S)-8-[2-(dimethylamino)ethyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol —— C18H23FN4O2
(6S)-4-[1-(7-fluoroquinazolin-2-yl)piperidin-4-yl]-1,4-oxazepan-6-ol
—— 6-methyl-5-[[4-[(1R)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]methyl]quinoline —— C23H34N4
6-methyl-5-[[4-[(1R)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]methyl]quinoline
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(3-methyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-2-yl)methanone —— C17H26N4O3S
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(3-methyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-2-yl)methanone
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(3-methyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-2-yl)methanone —— C17H26N4O3S
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(3-methyl-5,6-dihydroimidazo[2,1-b][1,3]thiazol-2-yl)methanone
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)methanone —— C13H18N2O4
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)methanone
—— (6R)-2-(2-hydroxyethyl)-8-[3-(tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one —— C15H26N6O2
(6R)-2-(2-hydroxyethyl)-8-[3-(tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-(4,5-Dimethoxy-2-methylphenyl)-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline —— C20H23NO4
6-(4,5-Dimethoxy-2-methylphenyl)-2,3,6,7,8,9-hexahydro-[1,4]dioxino[2,3-g]isoquinoline
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)methanone —— C13H18N2O4
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)methanone
—— [(6R)-4-[[1-(4-butylphenyl)pyrazol-4-yl]methyl]-1,4-oxazepan-6-yl]methanol —— C20H29N3O2
[(6R)-4-[[1-(4-butylphenyl)pyrazol-4-yl]methyl]-1,4-oxazepan-6-yl]methanol
—— (6S)-2-(2-hydroxyethyl)-8-[3-(tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one —— C15H26N6O2
(6S)-2-(2-hydroxyethyl)-8-[3-(tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-hydroxypropyl)-8-(3-pyrrol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N3O2
(6R)-2-(3-hydroxypropyl)-8-(3-pyrrol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-hydroxypropyl)-8-(3-pyrrol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H31N3O2
(6S)-2-(3-hydroxypropyl)-8-(3-pyrrol-1-ylpropyl)-2,8-diazaspiro[5.5]undecan-3-one