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中文名称 英文名称 CAS号 化学式 结构式图片
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1,3,7-trimethylindol-2-yl)methanone —— C18H24N2O3
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1,3,7-trimethylindol-2-yl)methanone
—— (6R)-2-cyclopentyl-8-(3-pyrrolidin-1-ylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H33N5O
(6R)-2-cyclopentyl-8-(3-pyrrolidin-1-ylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(cyclopropylmethyl)-8-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O4
(6R)-2-(cyclopropylmethyl)-8-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— 6-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H18FN5O3
6-[(2R)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6S)-2-(3-methylbutyl)-8-(6-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H29N3O3
(6S)-2-(3-methylbutyl)-8-(6-oxo-1H-pyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(2-cyclopropylacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O2
(6R)-8-(2-cyclopropylacetyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[4-(4-methylpiperazin-1-yl)phenyl]methanone —— C17H25N3O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[4-(4-methylpiperazin-1-yl)phenyl]methanone
—— (6R)-2-(2-hydroxyethyl)-8-[[3-(pyrazol-1-ylmethyl)phenyl]methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H30N4O2
(6R)-2-(2-hydroxyethyl)-8-[[3-(pyrazol-1-ylmethyl)phenyl]methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1,3,7-trimethylindol-2-yl)methanone —— C18H24N2O3
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(1,3,7-trimethylindol-2-yl)methanone
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[3-(1H-imidazol-2-yl)phenyl]methanone —— C20H26N4O3
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[3-(1H-imidazol-2-yl)phenyl]methanone
—— (6-chloro-3-fluoroimidazo[1,2-a]pyridin-2-yl)-[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]methanone —— C14H15ClFN3O3
(6-chloro-3-fluoroimidazo[1,2-a]pyridin-2-yl)-[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]methanone
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(1-methylindol-4-yl)methanone —— C15H18N2O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(1-methylindol-4-yl)methanone
—— 6-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C15H19N5O3
6-[(2S)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— 6-[[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C19H20N4O2S
6-[[(3S)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— (6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-pent-2-ynyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O
(6S)-2-[(5-methylpyrazin-2-yl)methyl]-8-pent-2-ynyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-pent-2-ynyl-2,8-diazaspiro[5.5]undecan-3-one —— C20H28N4O
(6R)-2-[(5-methylpyrazin-2-yl)methyl]-8-pent-2-ynyl-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O3
(6S)-2-(3-methoxypropyl)-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C16H22N4O3
(6R)-6-[[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— 6-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione —— C15H19N5O3
6-[(2R)-2-(2-pyrazol-1-ylethyl)piperidine-1-carbonyl]-1H-pyrimidine-2,4-dione
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(2-methoxy-4-methyl-1,3-thiazol-5-yl)methanone —— C12H18N2O4S
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(2-methoxy-4-methyl-1,3-thiazol-5-yl)methanone
—— 6-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione —— C18H18FN5O3
6-[(2S)-2-(6-fluoro-1H-benzimidazol-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[(3R)-3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H14FN3O2S
6-[(3R)-3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6S)-2-cyclopentyl-8-(3-pyrrolidin-1-ylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H33N5O
(6S)-2-cyclopentyl-8-(3-pyrrolidin-1-ylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(cyclopropylmethyl)-8-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H27N3O4
(6S)-2-(cyclopropylmethyl)-8-[4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methylsulfanyl-1,3-thiazol-4-yl)methanone —— C15H23N3O3S2
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-(2-methylsulfanyl-1,3-thiazol-4-yl)methanone
—— (6R)-2-cyclopropyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N2O3
(6R)-2-cyclopropyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2-phenoxyphenyl)methanone —— C18H19NO4
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2-phenoxyphenyl)methanone
—— 6-[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C18H20N4O2S
6-[(1S)-1-ethyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-2,3-dimethyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (6S)-2-cyclopropyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H26N2O3
(6S)-2-cyclopropyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(3-methoxypropyl)-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H29N3O3
(6R)-2-(3-methoxypropyl)-8-(4-methyl-1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethylamino]methyl]-1,4-oxazepan-6-ol —— C16H22N4O3
(6S)-6-[[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethylamino]methyl]-1,4-oxazepan-6-ol
—— 6-[[(3R)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide —— C19H20N4O2S
6-[[(3R)-3-(1,3-benzothiazol-2-yl)piperidin-1-yl]methyl]-2-oxo-1H-pyridine-3-carboxamide
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methylsulfanyl-1,3-thiazol-4-yl)methanone —— C10H14N2O3S2
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methylsulfanyl-1,3-thiazol-4-yl)methanone
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(2-methoxy-4-methyl-1,3-thiazol-5-yl)methanone —— C12H18N2O4S
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-(2-methoxy-4-methyl-1,3-thiazol-5-yl)methanone
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[4-(4-methylpiperazin-1-yl)phenyl]methanone —— C17H25N3O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[4-(4-methylpiperazin-1-yl)phenyl]methanone
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methyl-4-phenylpyridin-3-yl)methanone —— C18H20N2O3
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methyl-4-phenylpyridin-3-yl)methanone
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[3-(1H-imidazol-2-yl)phenyl]methanone —— C20H26N4O3
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[3-(1H-imidazol-2-yl)phenyl]methanone
—— (6-chloro-3-fluoroimidazo[1,2-a]pyridin-2-yl)-[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]methanone —— C14H15ClFN3O3
(6-chloro-3-fluoroimidazo[1,2-a]pyridin-2-yl)-[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]methanone
—— (6S)-2-butyl-8-(2,6-dimethylpyrimidine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6S)-2-butyl-8-(2,6-dimethylpyrimidine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-butyl-8-(2,6-dimethylpyrimidine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H30N4O2
(6R)-2-butyl-8-(2,6-dimethylpyrimidine-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-hydroxyethyl)-8-(5-propan-2-ylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O2
(6R)-2-(2-hydroxyethyl)-8-(5-propan-2-ylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-[4-(1H-pyrazol-5-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H26N4O2
(6S)-2-cyclopropyl-8-[4-(1H-pyrazol-5-yl)benzoyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-[(1-methylindol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N3O
(6S)-2-cyclopropyl-8-[(1-methylindol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[2-(2H-tetrazol-5-yl)phenyl]methanone —— C18H24N6O3
[(6R)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[2-(2H-tetrazol-5-yl)phenyl]methanone
—— (6S)-2-(2-hydroxyethyl)-8-(5-propan-2-ylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C18H28N4O2
(6S)-2-(2-hydroxyethyl)-8-(5-propan-2-ylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methyl-4-phenylpyridin-3-yl)methanone —— C18H20N2O3
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methyl-4-phenylpyridin-3-yl)methanone
—— (6R)-2-(2-methoxyethyl)-8-[2-(N-methylanilino)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H31N3O3
(6R)-2-(2-methoxyethyl)-8-[2-(N-methylanilino)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methylsulfanyl-1,3-thiazol-4-yl)methanone —— C10H14N2O3S2
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-(2-methylsulfanyl-1,3-thiazol-4-yl)methanone
—— (6R)-2-cyclopropyl-8-[(1-methylindol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N3O
(6R)-2-cyclopropyl-8-[(1-methylindol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[2-(2H-tetrazol-5-yl)phenyl]methanone —— C18H24N6O3
[(6S)-6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-[2-(2H-tetrazol-5-yl)phenyl]methanone