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—— 6-[[(6R)-6-hydroxy-1,4-oxazepan-6-yl]methyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one —— C13H22N4O3
6-[[(6R)-6-hydroxy-1,4-oxazepan-6-yl]methyl]-1,2,4,5,7,8-hexahydropyrazolo[3,4-d]azepin-3-one
—— (6-aminopyridin-3-yl)-[4-[(1R)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]methanone —— C18H29N5O
(6-aminopyridin-3-yl)-[4-[(1R)-1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl]methanone
—— (6S)-2-cyclopropyl-8-[2-(2,3-dihydro-1,4-benzoxazin-4-yl)-2-oxoethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H29N3O3
(6S)-2-cyclopropyl-8-[2-(2,3-dihydro-1,4-benzoxazin-4-yl)-2-oxoethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[[3-(2H-tetrazol-5-yl)phenyl]methylamino]methyl]-1,4-oxazepan-6-ol —— C14H20N6O2
(6S)-6-[[[3-(2H-tetrazol-5-yl)phenyl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-2-(3-methoxypropyl)-8-(tetrazolo[1,5-a]pyridine-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N6O3
(6R)-2-(3-methoxypropyl)-8-(tetrazolo[1,5-a]pyridine-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H27FN2O2
(6S)-2-cyclopropyl-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-[(1-propylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6S)-2-(3-methoxypropyl)-8-[(1-propylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-(2-indol-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one —— C21H27N3O3
(6S)-2-(2-hydroxyethyl)-8-(2-indol-1-ylacetyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-2-(2-methoxyethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C15H23N3O2S
(6R)-2-(2-methoxyethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(3-methoxypropyl)-8-(tetrazolo[1,5-a]pyridine-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N6O3
(6S)-2-(3-methoxypropyl)-8-(tetrazolo[1,5-a]pyridine-6-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-[[[3-(2H-tetrazol-5-yl)phenyl]methylamino]methyl]-1,4-oxazepan-6-ol —— C14H20N6O2
(6R)-6-[[[3-(2H-tetrazol-5-yl)phenyl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-8-(6-aminopyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H25N7O
(6S)-8-(6-aminopyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-[(1-ethylimidazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O
(6R)-8-[(1-ethylimidazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,4-oxazepan-6-ol —— C12H15N3O3
(6S)-4-(2,1,3-benzoxadiazol-4-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-2-(3-methoxypropyl)-8-[(1-propylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O2
(6R)-2-(3-methoxypropyl)-8-[(1-propylimidazol-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[3-(1-methylpyrrol-2-yl)-1H-pyrazol-5-yl]methanone —— C15H20N4O3
[(6R)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[3-(1-methylpyrrol-2-yl)-1H-pyrazol-5-yl]methanone
—— (6S)-2-(2-hydroxyethyl)-8-[(2-propan-2-ylpyrimidin-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O2
(6S)-2-(2-hydroxyethyl)-8-[(2-propan-2-ylpyrimidin-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C19H26N4O3
(6R)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-2-(2-methoxyethyl)-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6R)-2-(2-methoxyethyl)-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[3-(1-methylpyrrol-2-yl)-1H-pyrazol-5-yl]methanone —— C15H20N4O3
[(6S)-6-(hydroxymethyl)-1,4-oxazepan-4-yl]-[3-(1-methylpyrrol-2-yl)-1H-pyrazol-5-yl]methanone
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[6-(methoxymethyl)pyridin-2-yl]methanone —— C13H18N2O4
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[6-(methoxymethyl)pyridin-2-yl]methanone
—— (6S)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C19H26N4O3
(6S)-4-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C18H24N4O3
(6S)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-2-cyclopropyl-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C20H27FN2O2
(6R)-2-cyclopropyl-8-[2-(4-fluorophenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[2-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]-1,3-thiazol-4-yl]methanone —— C14H15F3N4O3S
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[2-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]-1,3-thiazol-4-yl]methanone
—— (6R)-2-cyclopropyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O
(6R)-2-cyclopropyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(1-ethylimidazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C20H34N4O
(6S)-8-[(1-ethylimidazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-6-[[[2-fluoro-5-(trifluoromethyl)phenyl]methylamino]methyl]-1,4-oxazepan-6-ol —— C14H18F4N2O2
(6S)-6-[[[2-fluoro-5-(trifluoromethyl)phenyl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-2-(2-hydroxyethyl)-8-[(2-propan-2-ylpyrimidin-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C19H30N4O2
(6R)-2-(2-hydroxyethyl)-8-[(2-propan-2-ylpyrimidin-5-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H30N2O3
(6S)-2-(2-methoxyethyl)-8-[2-(3-methylphenyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C21H28N4O
(6S)-2-cyclopropyl-8-[(8-methylimidazo[1,2-a]pyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
—— [(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[2-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]-1,3-thiazol-4-yl]methanone —— C14H15F3N4O3S
[(6S)-6-hydroxy-1,4-oxazepan-4-yl]-[2-[3-methyl-5-(trifluoromethyl)pyrazol-1-yl]-1,3-thiazol-4-yl]methanone
—— (6R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol —— C18H24N4O3
(6R)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
—— (6S)-2-(2-methoxyethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one —— C15H23N3O2S
(6S)-2-(2-methoxyethyl)-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-8-(6-aminopyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one —— C18H25N7O
(6R)-8-(6-aminopyrimidin-4-yl)-2-[2-(1H-imidazol-5-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
—— (6R)-6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-oxazepan-6-ol —— C14H23N3O2S
(6R)-6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-2-(2-hydroxyethyl)-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4
(6R)-2-(2-hydroxyethyl)-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— [(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[6-(methoxymethyl)pyridin-2-yl]methanone —— C13H18N2O4
[(6R)-6-hydroxy-1,4-oxazepan-4-yl]-[6-(methoxymethyl)pyridin-2-yl]methanone
—— (6R)-6-[[[5-(methoxymethyl)-1H-pyrazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol —— C12H22N4O3
(6R)-6-[[[5-(methoxymethyl)-1H-pyrazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6S)-6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-oxazepan-6-ol —— C14H23N3O2S
(6S)-6-(pyrrolidin-1-ylmethyl)-4-(1,3-thiazol-4-ylmethyl)-1,4-oxazepan-6-ol
—— (6R)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H35N3O2
(6R)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-cyclopropyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H23N3O2
(6S)-2-cyclopropyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-hydroxyethyl)-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one —— C19H26N2O4
(6S)-2-(2-hydroxyethyl)-8-(2-hydroxy-4-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-4-[[3-ethoxy-4-(3-methylbut-2-enoxy)phenyl]methyl]-1,4-oxazepan-6-ol —— C19H29NO4
(6S)-4-[[3-ethoxy-4-(3-methylbut-2-enoxy)phenyl]methyl]-1,4-oxazepan-6-ol
—— 6-[(3S)-3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one —— C18H16FN3O2S
6-[(3S)-3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-5-methyl-3H-thieno[2,3-d]pyrimidin-4-one
—— (6R)-4-[[3-ethoxy-4-(3-methylbut-2-enoxy)phenyl]methyl]-1,4-oxazepan-6-ol —— C19H29NO4
(6R)-4-[[3-ethoxy-4-(3-methylbut-2-enoxy)phenyl]methyl]-1,4-oxazepan-6-ol
—— (6S)-6-[[[5-(methoxymethyl)-1H-pyrazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol —— C12H22N4O3
(6S)-6-[[[5-(methoxymethyl)-1H-pyrazol-3-yl]methylamino]methyl]-1,4-oxazepan-6-ol
—— (6R)-2-cyclopropyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one —— C17H23N3O2
(6R)-2-cyclopropyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one —— C22H35N3O2
(6S)-8-[(3,5-dimethyl-4-oxo-1H-pyridin-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
—— (6S)-2-(2-methoxyethyl)-8-[(2-propoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one —— C22H34N2O3
(6S)-2-(2-methoxyethyl)-8-[(2-propoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one