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—— 5-[(2R)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]-1,3-dimethylpyrimidine-2,4-dione —— C17H24N4O3
5-[(2R)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]-1,3-dimethylpyrimidine-2,4-dione
—— 5-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C20H16FN5O3S
5-[(3S)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— (5R)-4,5,6,7-tetrahydrotriazolo[1,5-a]pyridine-5-carboxylic acid —— C7H9N3O2
(5R)-4,5,6,7-tetrahydrotriazolo[1,5-a]pyridine-5-carboxylic acid
—— 5-[(2S)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]-1,3-dimethylpyrimidine-2,4-dione —— C17H24N4O3
5-[(2S)-3-(cyclopropylmethyl)-4-oxo-1,3-diazaspiro[4.4]nonan-2-yl]-1,3-dimethylpyrimidine-2,4-dione
—— (5S)-4,5,6,7-tetrahydrotriazolo[1,5-a]pyridine-5-carboxylic acid —— C7H9N3O2
(5S)-4,5,6,7-tetrahydrotriazolo[1,5-a]pyridine-5-carboxylic acid
—— (5E)-5-({3-Bromo-5-methoxy-4-[2-(3-methoxyphenoxy)ethoxy]phenyl}methylidene)-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H20BrNO5S2
(5E)-5-({3-Bromo-5-methoxy-4-[2-(3-methoxyphenoxy)ethoxy]phenyl}methylidene)-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-3-(3-nitrobenzyl)-5-[4-(pyrrolidin-1-yl)benzylidene]-1,3-thiazolidine-2,4-dione —— C21H19N3O4S
(5E)-3-(3-nitrobenzyl)-5-[4-(pyrrolidin-1-yl)benzylidene]-1,3-thiazolidine-2,4-dione
—— 5-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole —— C20H16FN5O3S
5-[(3R)-2,3-dihydro-1,4-benzodioxin-3-yl]-3-[[5-(2-fluorophenyl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-1,2,4-oxadiazole
—— 5-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methylsulfanyl]-1-methyltetrazole —— C11H12N4OS
5-[[(2S)-2,3-dihydro-1-benzofuran-2-yl]methylsulfanyl]-1-methyltetrazole
—— (5S)-7-methyl-2,3,4,5-tetrahydro-1H-2-benzazepin-5-ol —— C11H15NO
(5S)-7-methyl-2,3,4,5-tetrahydro-1H-2-benzazepin-5-ol
—— (5R)-7-methyl-2,3,4,5-tetrahydro-1H-2-benzazepin-5-ol —— C11H15NO
(5R)-7-methyl-2,3,4,5-tetrahydro-1H-2-benzazepin-5-ol
—— (5E)-1-benzyl-5-[(4-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione —— C19H16N2O3S
(5E)-1-benzyl-5-[(4-methoxyphenyl)methylidene]-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-{(Z)-1-[2-(2-isopropyl-5-methylphenoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]methylidene}-3-methyl-2-thioxo-1,3-thiazolan-4-one —— C23H21N3O3S2
5-{(Z)-1-[2-(2-isopropyl-5-methylphenoxy)-4-oxo-4H-pyrido[1,2-a]pyrimidin-3-yl]methylidene}-3-methyl-2-thioxo-1,3-thiazolan-4-one
—— 5-chloro-2-ethylsulfanyl-N-[(2R,4S)-4-hydroxy-2-methylpentyl]benzamide —— C15H22ClNO2S
5-chloro-2-ethylsulfanyl-N-[(2R,4S)-4-hydroxy-2-methylpentyl]benzamide
—— 5-chloro-2-ethylsulfanyl-N-[(2S,4S)-4-hydroxy-2-methylpentyl]benzamide —— C15H22ClNO2S
5-chloro-2-ethylsulfanyl-N-[(2S,4S)-4-hydroxy-2-methylpentyl]benzamide
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (2R)-1-(adamantane-1-carbonyl)pyrrolidine-2-carboxylate —— C20H27N3O4
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (2R)-1-(adamantane-1-carbonyl)pyrrolidine-2-carboxylate
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl 4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoate —— C18H23N3O4
(5-methyl-1,3,4-oxadiazol-2-yl)methyl 4-[[(2S,6S)-2,6-dimethylmorpholin-4-yl]methyl]benzoate
—— (5E)-3-ethyl-5-[(1Z)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2(3H)-ylidene)butan-2-ylidene]-2-thioxo-1,3-thiazolidin-4-one —— C19H22N2O2S3
(5E)-3-ethyl-5-[(1Z)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2(3H)-ylidene)butan-2-ylidene]-2-thioxo-1,3-thiazolidin-4-one
—— (5Z)-3-(1,3-benzodioxol-5-ylmethyl)-5-[[7-methyl-2-(2-methylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C27H26N4O4S2
(5Z)-3-(1,3-benzodioxol-5-ylmethyl)-5-[[7-methyl-2-(2-methylpiperidin-1-yl)-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-chloro-2-ethylsulfanyl-N-[(2R,4R)-4-hydroxy-2-methylpentyl]benzamide —— C15H22ClNO2S
5-chloro-2-ethylsulfanyl-N-[(2R,4R)-4-hydroxy-2-methylpentyl]benzamide
—— 5-(4-methoxyphenyl)-7-(trifluoromethyl)-N-(2,4,4-trimethylpentan-2-yl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide —— C23H31F3N4O2
5-(4-methoxyphenyl)-7-(trifluoromethyl)-N-(2,4,4-trimethylpentan-2-yl)-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-2-carboxamide
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl 4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]benzoate —— C18H23N3O4
(5-methyl-1,3,4-oxadiazol-2-yl)methyl 4-[[(2S,6R)-2,6-dimethylmorpholin-4-yl]methyl]benzoate
—— 5,7-dimethyl-N'-(1-phenylethylidene)[1,2,4]triazolo[1,5-a]pyrimidine-2-carbohydrazide —— C16H16N6O
5,7-dimethyl-N'-(1-phenylethylidene)[1,2,4]triazolo[1,5-a]pyrimidine-2-carbohydrazide
—— (5Z)-3-cyclopentyl-5-[(2-morpholin-4-yl-4-oxopyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H22N4O3S2
(5Z)-3-cyclopentyl-5-[(2-morpholin-4-yl-4-oxopyrido[1,2-a]pyrimidin-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-chloro-2-ethylsulfanyl-N-[(2S,4R)-4-hydroxy-2-methylpentyl]benzamide —— C15H22ClNO2S
5-chloro-2-ethylsulfanyl-N-[(2S,4R)-4-hydroxy-2-methylpentyl]benzamide
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (2S)-1-(adamantane-1-carbonyl)pyrrolidine-2-carboxylate —— C20H27N3O4
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (2S)-1-(adamantane-1-carbonyl)pyrrolidine-2-carboxylate
—— 5-[(3S)-1-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C14H20N6O2
5-[(3S)-1-[(1S)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (3R)-1-(2,3-dihydro-1H-inden-5-yl)-5-oxopyrrolidine-3-carboxylate —— C18H19N3O4
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (3R)-1-(2,3-dihydro-1H-inden-5-yl)-5-oxopyrrolidine-3-carboxylate
—— (5Z)-3-(2-ethylhexyl)-5-({3-[4-(ethylsulfanyl)phenyl]-1-phenyl-1H-pyrazol-4-yl}methylidene)-2-thioxo-1,3-thiazolidin-4-one —— C29H33N3OS3
(5Z)-3-(2-ethylhexyl)-5-({3-[4-(ethylsulfanyl)phenyl]-1-phenyl-1H-pyrazol-4-yl}methylidene)-2-thioxo-1,3-thiazolidin-4-one
—— (5E)-5-(anilinomethylidene)-1-(3,5-dichlorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione —— C17H11Cl2N3O2S
(5E)-5-(anilinomethylidene)-1-(3,5-dichlorophenyl)-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-[(3S)-1-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide —— C14H20N6O2
5-[(3S)-1-[(1R)-1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]piperidin-3-yl]-1H-pyrazole-3-carboxamide
—— (5-methyl-1,3,4-oxadiazol-2-yl)methyl (3S)-1-(2,3-dihydro-1H-inden-5-yl)-5-oxopyrrolidine-3-carboxylate —— C18H19N3O4
(5-methyl-1,3,4-oxadiazol-2-yl)methyl (3S)-1-(2,3-dihydro-1H-inden-5-yl)-5-oxopyrrolidine-3-carboxylate
—— (5S)-N-[4-(2-methylimidazol-1-yl)butyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole-5-carboxamide —— C17H22F3N5O
(5S)-N-[4-(2-methylimidazol-1-yl)butyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole-5-carboxamide
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone —— C13H19ClN4O
(5-chloro-2-methylpyrimidin-4-yl)-[(3R,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone
—— (5Z)-5-[(2,5-dimethyl-1H-pyrrol-3-yl)methylidene]-3-[2-(1H-indol-3-yl)ethyl]-2-(4-methoxyphenyl)imino-1,3-thiazolidin-4-one —— C27H26N4O2S
(5Z)-5-[(2,5-dimethyl-1H-pyrrol-3-yl)methylidene]-3-[2-(1H-indol-3-yl)ethyl]-2-(4-methoxyphenyl)imino-1,3-thiazolidin-4-one
—— (5Z)-5-{4-[2-(4-bromophenoxy)ethoxy]-3,5-dichlorobenzylidene}-3-methyl-2-thioxo-1,3-thiazolidin-4-one —— C19H14BrCl2NO3S2
(5Z)-5-{4-[2-(4-bromophenoxy)ethoxy]-3,5-dichlorobenzylidene}-3-methyl-2-thioxo-1,3-thiazolidin-4-one
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S,4R)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone —— C13H19ClN4O
(5-chloro-2-methylpyrimidin-4-yl)-[(3S,4R)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone
—— 5-(4-Tert-butylphenyl)-4-[hydroxy-(3-methoxyphenyl)methylidene]-1-pyridin-2-ylpyrrolidine-2,3-dione —— C27H26N2O4
5-(4-Tert-butylphenyl)-4-[hydroxy-(3-methoxyphenyl)methylidene]-1-pyridin-2-ylpyrrolidine-2,3-dione
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone —— C13H19ClN4O
(5-chloro-2-methylpyrimidin-4-yl)-[(3S,4S)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2S)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]methanone —— C15H14ClN3OS
(5-chloro-2-methylpyrimidin-4-yl)-[(2S)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]methanone —— C15H14ClN3OS
(5-chloro-2-methylpyrimidin-4-yl)-[(2R)-2-methyl-2,3-dihydro-1,4-benzothiazin-4-yl]methanone
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R,4R)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone —— C13H19ClN4O
(5-chloro-2-methylpyrimidin-4-yl)-[(3R,4R)-3-(dimethylamino)-4-methylpyrrolidin-1-yl]methanone
—— (5Z)-5-[(2,4-diethoxyphenyl)methylidene]-3-[(4-nitrophenyl)methyl]-1,3-thiazolidine-2,4-dione —— C21H20N2O6S
(5Z)-5-[(2,4-diethoxyphenyl)methylidene]-3-[(4-nitrophenyl)methyl]-1,3-thiazolidine-2,4-dione
—— 5-chloro-N-[(1S)-4,4-dimethyl-2,3-dihydro-1H-naphthalen-1-yl]-2-methylpyrimidine-4-carboxamide —— C18H20ClN3O
5-chloro-N-[(1S)-4,4-dimethyl-2,3-dihydro-1H-naphthalen-1-yl]-2-methylpyrimidine-4-carboxamide
—— (5R)-N-[4-(2-methylimidazol-1-yl)butyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole-5-carboxamide —— C17H22F3N5O
(5R)-N-[4-(2-methylimidazol-1-yl)butyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole-5-carboxamide
—— (5R)-N-[2-(5-tert-butyl-1,2,4-oxadiazol-3-yl)propan-2-yl]-3-(2,4-dichlorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide —— C19H22Cl2N4O3
(5R)-N-[2-(5-tert-butyl-1,2,4-oxadiazol-3-yl)propan-2-yl]-3-(2,4-dichlorophenyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
—— 5-chloro-2-methyl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrimidine-4-carboxamide —— C14H14ClN3O2
5-chloro-2-methyl-N-[(4R)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrimidine-4-carboxamide
—— 5-chloro-2-methyl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrimidine-4-carboxamide —— C14H14ClN3O2
5-chloro-2-methyl-N-[(4S)-4,5,6,7-tetrahydro-1-benzofuran-4-yl]pyrimidine-4-carboxamide
—— 5-chloro-N-[(1R)-4,4-dimethyl-2,3-dihydro-1H-naphthalen-1-yl]-2-methylpyrimidine-4-carboxamide —— C18H20ClN3O
5-chloro-N-[(1R)-4,4-dimethyl-2,3-dihydro-1H-naphthalen-1-yl]-2-methylpyrimidine-4-carboxamide
—— (5S)-5-[(2S)-2-(4-tert-butyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one —— C17H25N3O2S
(5S)-5-[(2S)-2-(4-tert-butyl-1,3-thiazol-2-yl)piperidine-1-carbonyl]pyrrolidin-2-one