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—— (5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methanone —— C15H18ClN5O
(5-chloro-2-methylpyrimidin-4-yl)-[(3S)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methanone
—— 5-(3,5-dimethylpyrazol-1-yl)-N-[2-[[(2S)-oxolan-2-yl]methoxy]ethyl]pyridin-2-amine —— C17H24N4O2
5-(3,5-dimethylpyrazol-1-yl)-N-[2-[[(2S)-oxolan-2-yl]methoxy]ethyl]pyridin-2-amine
—— 5-methyl-7-[(2S)-2-(3-phenylpropyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H25N5
5-methyl-7-[(2S)-2-(3-phenylpropyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-methyl-N-[(1S)-1-naphthalen-1-ylethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C18H17N5
5-methyl-N-[(1S)-1-naphthalen-1-ylethyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5-bromofuran-2-yl)-[(3S)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methanone —— C14H16BrN3O2
(5-bromofuran-2-yl)-[(3S)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methanone
—— 5-[(2,4-dichlorophenoxy)methyl]-1,3,4-oxadiazol-2-yl (1E)-N-(4-nitrophenyl)-2-oxo-2-phenylethanehydrazonothioate —— C23H15Cl2N5O5S
5-[(2,4-dichlorophenoxy)methyl]-1,3,4-oxadiazol-2-yl (1E)-N-(4-nitrophenyl)-2-oxo-2-phenylethanehydrazonothioate
—— (5Z)-3-amino-5-[(3-methylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C11H10N2OS2
(5Z)-3-amino-5-[(3-methylphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-methyl-N-[(2R)-1-(4-phenylphenyl)propan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C21H21N5
5-methyl-N-[(2R)-1-(4-phenylphenyl)propan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5-methyl-1H-pyrazol-3-yl)-[(3R)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone —— C12H16N6O
(5-methyl-1H-pyrazol-3-yl)-[(3R)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone
—— 5-[(4R)-3,4-dihydro-2H-chromen-4-yl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole —— C19H17N5O2
5-[(4R)-3,4-dihydro-2H-chromen-4-yl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole
—— 5-cyclopropyl-3-[(2S)-1-[(5,7-dimethylimidazo[1,2-a]pyrimidin-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole —— C18H22N6O
5-cyclopropyl-3-[(2S)-1-[(5,7-dimethylimidazo[1,2-a]pyrimidin-2-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazole
—— (5Z)-5-[(Z)-2-bromo-3-phenylprop-2-enylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H12BrNOS2
(5Z)-5-[(Z)-2-bromo-3-phenylprop-2-enylidene]-3-phenyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-methyl-7-[(2R)-2-(3-phenylpropyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H25N5
5-methyl-7-[(2R)-2-(3-phenylpropyl)piperidin-1-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 5-[(1S)-1-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole —— C17H18N6O2
5-[(1S)-1-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole
—— 5-methyl-N-(4-methylcyclohexyl)-N-[[(2R)-oxolan-2-yl]methyl]-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C19H26F3N5O
5-methyl-N-(4-methylcyclohexyl)-N-[[(2R)-oxolan-2-yl]methyl]-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-methyl-N-[(2R)-4-methyl-4-phenylpentan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C18H23N5
5-methyl-N-[(2R)-4-methyl-4-phenylpentan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5S)-N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C18H22N4O2
(5S)-N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-methyl-N-[(2S)-1-(4-phenylphenyl)propan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C21H21N5
5-methyl-N-[(2S)-1-(4-phenylphenyl)propan-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— 5-[(4S)-3,4-dihydro-2H-chromen-4-yl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole —— C19H17N5O2
5-[(4S)-3,4-dihydro-2H-chromen-4-yl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole
—— (5Z)-5-[[3-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-3-[(4-nitrophenyl)methyl]-1,3-thiazolidine-2,4-dione —— C24H16Cl2N2O5S
(5Z)-5-[[3-[(2,4-dichlorophenyl)methoxy]phenyl]methylidene]-3-[(4-nitrophenyl)methyl]-1,3-thiazolidine-2,4-dione
—— (5-methyl-1H-pyrazol-3-yl)-[(3S)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone —— C12H16N6O
(5-methyl-1H-pyrazol-3-yl)-[(3S)-3-(1,2,4-triazol-1-yl)piperidin-1-yl]methanone
—— (5Z)-5-{[5-(2,4-dichlorophenyl)furan-2-yl]methylidene}-2-(4-methoxyphenyl)[1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one —— C22H13Cl2N3O3S
(5Z)-5-{[5-(2,4-dichlorophenyl)furan-2-yl]methylidene}-2-(4-methoxyphenyl)[1,3]thiazolo[3,2-b][1,2,4]triazol-6(5H)-one
—— (5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methanone —— C15H18ClN5O
(5-chloro-2-methylpyrimidin-4-yl)-[(3R)-3-(5-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methanone
—— 5-[(1R)-1-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole —— C17H18N6O2
5-[(1R)-1-(3,5-dimethyl-1,2-oxazol-4-yl)ethyl]-3-(5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl)-1,2,4-oxadiazole
—— (5R)-N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C18H22N4O2
(5R)-N-[(2R)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-methyl-N-(4-methylcyclohexyl)-N-[[(2S)-oxolan-2-yl]methyl]-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine —— C19H26F3N5O
5-methyl-N-(4-methylcyclohexyl)-N-[[(2S)-oxolan-2-yl]methyl]-2-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
—— (5S)-N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C18H22N4O2
(5S)-N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— (5R)-N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide —— C18H22N4O2
(5R)-N-[(2S)-1-(3,5-dimethylpyrazol-1-yl)propan-2-yl]-5-phenyl-4,5-dihydro-1,2-oxazole-3-carboxamide
—— 5-[4-(dimethylamino)phenyl]-N-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]pyridine-3-carboxamide —— C23H29N5O
5-[4-(dimethylamino)phenyl]-N-[(2S)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]pyridine-3-carboxamide
—— 5-[4-(dimethylamino)phenyl]-N-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]pyridine-3-carboxamide —— C23H29N5O
5-[4-(dimethylamino)phenyl]-N-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]pyridine-3-carboxamide
—— 5-methyl-N-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]pyridine-3-carboxamide —— C20H23N3O2
5-methyl-N-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
—— 5-[(2,5-Dihydroxyphenyl)methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione —— C13H12N2O4S
5-[(2,5-Dihydroxyphenyl)methylidene]-1,3-dimethyl-2-sulfanylidene-1,3-diazinane-4,6-dione
—— 5-methyl-N-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]pyridine-3-carboxamide —— C20H23N3O2
5-methyl-N-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
—— (5E)-5-{[5-(4-bromophenyl)furan-2-yl]methylidene}-3-(3-fluorophenyl)-2-thioxo-1,3-thiazolidin-4-one —— C20H11BrFNO2S2
(5E)-5-{[5-(4-bromophenyl)furan-2-yl]methylidene}-3-(3-fluorophenyl)-2-thioxo-1,3-thiazolidin-4-one
—— 5-[[methyl-[(1R,2S)-2-methylsulfonylcyclohexyl]amino]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C15H22N4O3S
5-[[methyl-[(1R,2S)-2-methylsulfonylcyclohexyl]amino]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5E)-5-butan-2-ylidene-3-(4-chlorobenzoyl)-2-sulfanylidene-1,3-thiazolidin-4-one —— C14H12ClNO2S2
(5E)-5-butan-2-ylidene-3-(4-chlorobenzoyl)-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-(3,4-dimethoxyphenyl)-3-hydroxy-1-(2-hydroxypropyl)-4-[(4-methylphenyl)carbonyl]-1,5-dihydro-2H-pyrrol-2-one —— C23H25NO6
5-(3,4-dimethoxyphenyl)-3-hydroxy-1-(2-hydroxypropyl)-4-[(4-methylphenyl)carbonyl]-1,5-dihydro-2H-pyrrol-2-one
—— (5Z)-5-{4-[(2,4-dichlorobenzyl)oxy]-3-methoxy-5-(prop-2-en-1-yl)benzylidene}-3-(3-nitrobenzyl)-1,3-thiazolidine-2,4-dione —— C28H22Cl2N2O6S
(5Z)-5-{4-[(2,4-dichlorobenzyl)oxy]-3-methoxy-5-(prop-2-en-1-yl)benzylidene}-3-(3-nitrobenzyl)-1,3-thiazolidine-2,4-dione
—— 5-[[methyl-[(1S,2S)-2-methylsulfonylcyclohexyl]amino]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one —— C15H22N4O3S
5-[[methyl-[(1S,2S)-2-methylsulfonylcyclohexyl]amino]methyl]-1H-pyrazolo[1,5-a]pyrimidin-7-one
—— (5Z)-3-[4-(difluoromethoxy)phenyl]-5-[(4-methoxyphenyl)methylidene]-2-(2-oxooxolan-3-yl)sulfanylimidazol-4-one —— C22H18F2N2O5S
(5Z)-3-[4-(difluoromethoxy)phenyl]-5-[(4-methoxyphenyl)methylidene]-2-(2-oxooxolan-3-yl)sulfanylimidazol-4-one
—— 5-(5-{(E)-[3-(4-fluorobenzyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}furan-2-yl)benzene-1,3-dicarboxylic acid —— C23H14FNO7S
5-(5-{(E)-[3-(4-fluorobenzyl)-2,4-dioxo-1,3-thiazolidin-5-ylidene]methyl}furan-2-yl)benzene-1,3-dicarboxylic acid
—— (5E)-5-[(2E)-2-(6-methoxy-1-methylquinolin-2-ylidene)ethylidene]quinolin-1-ium-8-one —— C22H19N2O2+
(5E)-5-[(2E)-2-(6-methoxy-1-methylquinolin-2-ylidene)ethylidene]quinolin-1-ium-8-one
—— (5Z)-5-[[5-(4-chlorophenyl)sulfanylthiophen-2-yl]methylidene]-3-(cyclohexylmethyl)-1,3-thiazolidine-2,4-dione —— C21H20ClNO2S3
(5Z)-5-[[5-(4-chlorophenyl)sulfanylthiophen-2-yl]methylidene]-3-(cyclohexylmethyl)-1,3-thiazolidine-2,4-dione
—— (5Z)-3-[2-(azepan-1-yl)-2-oxoethyl]-5-[(5-bromofuran-2-yl)methylidene]-1,3-thiazolidine-2,4-dione —— C16H17BrN2O4S
(5Z)-3-[2-(azepan-1-yl)-2-oxoethyl]-5-[(5-bromofuran-2-yl)methylidene]-1,3-thiazolidine-2,4-dione
—— (5Z)-5-[(4-butoxy-3-methoxyphenyl)methylidene]-3-(4-methoxyphenyl)-2-phenyl-1,3-thiazolidin-4-one —— C28H29NO4S
(5Z)-5-[(4-butoxy-3-methoxyphenyl)methylidene]-3-(4-methoxyphenyl)-2-phenyl-1,3-thiazolidin-4-one
—— 5-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]thiophene-3-carbonitrile —— C12H12N2OS
5-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]thiophene-3-carbonitrile
—— 5-[(1S,4R)-2-azabicyclo[2.2.1]heptane-2-carbonyl]thiophene-3-carbonitrile —— C12H12N2OS
5-[(1S,4R)-2-azabicyclo[2.2.1]heptane-2-carbonyl]thiophene-3-carbonitrile
—— (5S)-5-[(4,6-dimethylpyrimidin-2-yl)amino]-1-methylpiperidin-2-one —— C12H18N4O
(5S)-5-[(4,6-dimethylpyrimidin-2-yl)amino]-1-methylpiperidin-2-one
—— (5S)-5-[(2,6-dimethylpyrimidin-4-yl)amino]-1-methylpiperidin-2-one —— C12H18N4O
(5S)-5-[(2,6-dimethylpyrimidin-4-yl)amino]-1-methylpiperidin-2-one
—— (5R)-5-(1,3-benzoxazol-2-ylamino)-1-methylpiperidin-2-one —— C13H15N3O2
(5R)-5-(1,3-benzoxazol-2-ylamino)-1-methylpiperidin-2-one