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中枢兴奋药

中枢兴奋药是一类能够对中枢神经系统产生兴奋作用的药物。根据其主要作用部位,可分为几大类:主要兴奋大脑皮质的药物、主要兴奋延髓呼吸中枢的药物以及主要兴奋脊髓的药物。这类药物若使用过量,均有可能引发惊厥。

中文名称 英文名称 CAS号 化学式 结构式图片
香草醛.香兰素 1-Ethyl-4-(2-morpholin-4-ylethyl)-3,3-diphenylpyrrolidin-2-one;hydron;chloride;hydrate 7081-53-0 C24H33ClN2O3
香草醛.香兰素
香草二乙胺 etamivan 304-84-7 C12H17NO3
香草二乙胺
醋谷胺 2-acetamidoacetamide 2620-63-5 C4H8N2O2
醋谷胺
贝美格 bemegride 64-65-3 C8H13NO2
贝美格
苦毒浆果[木防已属] Cocculin 124-87-8 C30H34O13
苦毒浆果[木防已属]
盐酸山梗碱 Lobeline hydrochloride 134-63-4 C22H27NO2*ClH
盐酸山梗碱
盐酸士的宁 Brucine hydrochloride 5786-96-9 C23H26N2O4*ClH
盐酸士的宁
盐酸士的宁 strychnine hydrochloride 1421-86-9 C21H22N2O2*ClH
盐酸士的宁
甲氯芬酯 meclofenoxate 51-68-3 C12H16ClNO3
甲氯芬酯
混旋樟脑磺酸钠 D-Camphor-10-sulfonic acid sodium salt 34850-66-3 C10H16NaO4S
混旋樟脑磺酸钠
洛贝林 lobeline 90-69-7 C22H27NO2
洛贝林
氯酯醒 meclofenoxate hydrochloride 3685-84-5 C12H16ClNO3*ClH
氯酯醒
氧气 oxygen 7782-44-7 O2
氧气
戊四唑 pentetrazole 54-95-5 C6H10N4
戊四唑
尼可刹米 N,N-diethylnicotinamide 59-26-7 C10H14N2O
尼可刹米
多沙普仑 doxapram 309-29-5 C24H30N2O2
多沙普仑
二氧化碳 carbon dioxide 124-38-9 CO2
二氧化碳
二棕榈酸磷脂酰胆碱 L-Dipalmitoylphosphatidylcholine 63-89-8 C40H80NO8P
二棕榈酸磷脂酰胆碱
一叶秋碱 (-)-securinine 5610-40-2 C13H15NO2
一叶秋碱
D-樟脑酸 D-(+)-camphoric acid 5394-83-2 C10H16O4
D-樟脑酸
—— (1R,3R,5S,8S,13R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,5S,8S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C30H34O13
(1R,3R,5S,8S,13R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,5S,8S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— (1R,3R,8S,9R,12S,13R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,8S,9R,12S,13R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C30H34O13
(1R,3R,8S,9R,12S,13R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,8S,9R,12S,13R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— (-)-α-lobeline 90-69-7 C22H27NO2
(-)-α-lobeline
—— Picrotoxin 124-87-8 C15H18O7.C15H16O6
Picrotoxin
—— (1R,3R,5S,8S,9S,12R,13R,14S)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,5S,8S,9S,12R,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C30H34O13
(1R,3R,5S,8S,9S,12R,13R,14S)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,5S,8S,9S,12R,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— Cocculus 124-87-8 C15H18O7.C15H16O6
Cocculus
—— Lobeline alpha (-) hydrochoride 134-63-4 C22H28ClNO2
Lobeline alpha (-) hydrochoride
—— (1R,3R,8S,9R,12S,13R,14S)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C30H34O13
(1R,3R,8S,9R,12S,13R,14S)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— (1R,3R,5S,8S,9R,12S,13R,14R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C15H18O7.C15H16O6
(1R,3R,5S,8S,9R,12S,13R,14R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— 2-[(2S)-6-[(2R)-2-hydroxy-2-phenylethyl]-1-methylpiperidin-2-yl]-1-phenylethanone;hydrochloride 134-63-4 C22H28ClNO2
2-[(2S)-6-[(2R)-2-hydroxy-2-phenylethyl]-1-methylpiperidin-2-yl]-1-phenylethanone;hydrochloride
—— strychnine hyudrochloride 1421-86-9 C21H22N2O2*ClH
strychnine hyudrochloride
—— Lobron 90-69-7 C22H27NO2
Lobron
—— (1S,3R,5S,8S,9S,12R,13S,14S)-1-Hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1S,3R,5S,8S,9S,12R,13S,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C30H34O13
(1S,3R,5S,8S,9S,12R,13S,14S)-1-Hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1S,3R,5S,8S,9S,12R,13S,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— 2-[(2<i>RS</i>)-6<i>c</i>-((<i>SR</i>)-β-hydroxy-phenethyl)-1-methyl-[2<i>r</i>]piperidyl]-1-phenyl-ethanone 90-69-7 C22H27NO2
2-[(2<i>RS</i>)-6<i>c</i>-((<i>SR</i>)-β-hydroxy-phenethyl)-1-methyl-[2<i>r</i>]piperidyl]-1-phenyl-ethanone
—— (1R,3R,5S,8S,9R,12S,13R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,5S,8S,9R,12S,13R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione 124-87-8 C30H34O13
(1R,3R,5S,8S,9R,12S,13R)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,5S,8S,9R,12S,13R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione
—— 2-[(2S,6R)-6-(2-hydroxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone 90-69-7 C22H27NO2
2-[(2S,6R)-6-(2-hydroxy-2-phenylethyl)-1-methylpiperidin-2-yl]-1-phenylethanone
—— sodium camphorsulfonate 34850-66-3 C10H15O4S*Na
sodium camphorsulfonate
—— Lobelin-hydrochlorid 134-63-4 C22H27NO2*ClH
Lobelin-hydrochlorid
—— (-)-α-lobeline hydrochloride 134-63-4 C22H27NO2*ClH
(-)-α-lobeline hydrochloride
—— strychnine nitrate 66-32-0 C21H22N2O2*HNO3
strychnine nitrate
—— hydroperoxyl radical 7782-44-7 HO2
hydroperoxyl radical