(4-cyclopropylphenyl)methanesulfonyl chloride | 1521474-21-4

• 分子结构分类: 有机化合物 - 苯类化合物 - 苯和取代衍生物
• 英文名称: (4-cyclopropylphenyl)methanesulfonyl chloride
• CAS: 1521474-21-4
• 化学式: C₁₀H₁₁ClO₂S
• 分子量: 230.715
• InChiKey: ACXMSQQWIKYWTM-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  2.8
• 重原子数：
  14
• 可旋转键数：
  3
• 环数：
  2.0
• sp3杂化的碳原子比例：
  0.4
• 拓扑面积：
  42.5
• 氢给体数：
  0
• 氢受体数：
  2

反应信息

• 作为反应物：
  描述：

  6-amino-1-propyl-3,4-dihydroquinolin-2-one 、 (4-cyclopropylphenyl)methanesulfonyl chloride 在 N,N-二异丙基乙胺 作用下， 以 乙酸乙酯 为溶剂， 以77%的产率得到1-(4-cyclopropylphenyl)-N-(2-oxo-1-propyl-3,4-dihydroquinolin-6-yl)methanesulfonamide
  参考文献：
  名称：

  WO2016/22910

  摘要：

  公开号：

文献信息

• 2-oxo-3,4-dihydroquinolin-6-yl sulphonamide CPDS and their use as plant growth regulators
  申请人：THE REGENTS OF THE UNIVERSITY OF CALIFORNIA

  公开号：US10167261B2

  公开（公告）日：2019-01-01

  The present invention relates to sulfonamide derivatives of formula (I) where the substituents R1-R6 and R8, L, A and n are as defined in the application, to plant growth regulator compositions comprising them and to methods of using them for controlling the growth of plants, improving plant tolerance to abiotic stress (including environmental and chemical stresses), inhibiting seed germination and/or safening a plant against phytotoxic effects of chemicals.

  本发明涉及式（I）的磺酰胺衍生物（其中取代基 R1-R6 和 R8、L、A 和 n 如本申请中所定义），涉及包含它们的植物生长调节剂组合物，涉及使用它们控制植物生长、提高植物对非生物胁迫（包括环境和化学胁迫）的耐受性、抑制种子萌发和/或使植物免受化学品植物毒性影响的方法。
• 2-OXO-3,4-DIHYDROQUINOLIN-6-YL SULPHONAMIDE CPDS AND THEIR USE AS PLANT GROWTH REGULATORS.
  申请人：The Regents of the University of California

  公开号：EP3180313A2

  公开（公告）日：2017-06-21
• 2-OXO-3,4-DIHYDROQUINOLIN-6-YL SULPHONAMIDE CPDS AND THEIR USE AS PLANT GROWTH REGULATORS
  申请人：The Regents of the University of California

  公开号：EP3180313B1

  公开（公告）日：2021-01-06
• [EN] PLANT GROWTH REGULATOR COMPOUNDS<br/>[FR] COMPOSÉS RÉGULATEURS DE LA CROISSANCE VÉGÉTALE
  申请人：UNIV CALIFORNIA

  公开号：WO2016022910A2

  公开（公告）日：2016-02-11

  The present invention relates to novel sulfonamide derivatives, to processes and intermediates for preparing them, to plant growth regulator compositions comprising them and to methods of using them for controlling the growth of plants, improving plant tolerance to abiotic stress (including environmental and chemical stresses), inhibiting seed germination and/or safening a plant against phytotoxic effects of chemicals.