6-Amino-2-(1-benzothiophen-5-yl)-5-methoxypyrimidine-4-carboxylic acid

• 分子结构分类: 有机化合物 - 有机杂环化合物 - 二嗪类
• 英文名称: 6-Amino-2-(1-benzothiophen-5-yl)-5-methoxypyrimidine-4-carboxylic acid
• 英文别名: 6-amino-2-(1-benzothiophen-5-yl)-5-methoxypyrimidine-4-carboxylic acid
• 化学式: C₁₄H₁₁N₃O₃S
• 分子量: 301.326
• InChiKey: YHGNMUQDLLOSJB-UHFFFAOYSA-N

计算性质

• 辛醇/水分配系数(LogP)：
  2.4
• 重原子数：
  21
• 可旋转键数：
  3
• 环数：
  3.0
• sp3杂化的碳原子比例：
  0.07
• 拓扑面积：
  127
• 氢给体数：
  2
• 氢受体数：
  7

文献信息

• 4-AMINO-6-(HETEROCYCLIC)PICOLINATES AND 6-AMINO-2-(HETEROCYCLIC)PYRIMIDINE-4-CARBOXYLATES AND THEIR USE AS HERBICIDES
  申请人：Dow AgroSciences, LLC

  公开号：US20150126372A1

  公开（公告）日：2015-05-07

  4-Amino-6-(heterocyclic)picolinic acids and their derivatives; 6-amino-2-(heterocyclic)pyrimidine-4-carboxylates and their derivatives; and methods of using the same as herbicides.

  4-氨基-6-(杂环)吡啶甲酸及其衍生物；6-氨基-2-(杂环)嘧啶-4-羧酸酯及其衍生物；以及将其作为除草剂的方法。
• SAFENED HERBICIDAL COMPOSITIONS COMPRISING PYRIDINE CARBOXYLIC ACIDS
  申请人：Dow AgroSciences LLC

  公开号：EP3508063A1

  公开（公告）日：2019-07-10

  Disclosed herein are safened herbicidal compositions comprising (a) a pyridine carboxylic acid herbicide, or an agriculturally acceptable N-oxide, salt or ester thereof, and (b) an azole carboxylate safener, or agriculturally acceptable salt or ester thereof. Also disclosed herein are methods of controlling undesirable vegetation, comprising applying to vegetation or an area adjacent the vegetation or applying in soil or water to control the emergence or growth of vegetation (a) a pyridine carboxylic acid herbicide, or an agriculturally acceptable N-oxide, salt or ester thereof, and (b) an azole carboxylate safener, or agriculturally acceptable salt or ester thereof.

  本文公开了安全除草组合物，包括(a)吡啶甲酸除草剂，或其农业上可接受的 N-氧化物、盐或酯，和(b)唑羧酸盐安全剂，或其农业上可接受的盐或酯。本文还公开了控制不良植被的方法，包括向植被或植被邻近区域施用，或在土壤或水中施用，以控制植被的出现或生长：(a) 吡啶甲酸除草剂，或其农业上可接受的 N-氧化物、盐或酯，以及 (b) 唑类羧酸酯安全剂，或其农业上可接受的盐或酯。
• Synergistic weed control from applications of pyridine carboxylic acid herbicides and synthetic auxin herbicides and/or auxin transport inhibitors
  申请人：Dow AgroSciences LLC

  公开号：US10231451B2

  公开（公告）日：2019-03-19

  Disclosed herein are herbicidal compositions comprising a herbicidally effective amount of (a) a pyridine carboxylic acid herbicide or an agriculturally acceptable N-oxide, salt or ester thereof, and (b) a synthetic auxin herbicide, an auxin transport inhibitor, agriculturally acceptable salts or esters thereof, or combinations thereof. Also disclosed herein are methods of controlling undesirable vegetation which comprise applying to vegetation or an area adjacent the vegetation or applying to soil or water to prevent the emergence or growth of vegetation (a) a pyridine carboxylic acid herbicide or an agriculturally acceptable N-oxide, salt or ester thereof, and (b) a synthetic auxin herbicide, an auxin transport inhibitor, agriculturally acceptable salts or esters thereof, or combinations thereof, wherein (a) and (b) are each added in an amount sufficient to provide a herbicidal effect.

  本文公开了除草组合物，该组合物包含除草有效量的(a)吡啶羧酸除草剂或其农业上可接受的 N-氧化物、盐或酯，和(b)合成辅助素除草剂、辅助素转运抑制剂、其农业上可接受的盐或酯，或其组合。本文还公开了控制不良植被的方法，包括向植被或植被邻近区域施用，或向土壤或水中施用，以防止植被出现或生长 (a) 吡啶羧酸除草剂或农业上可接受的 N-氧化物、(b) 合成辅助素除草剂、辅助素转运抑制剂、农业上可接受的盐或酯，或它们的组合，其中(a)和(b)的添加量足以提供除草效果。
• Synergistic weed control from applications of pyridine carboxylic acid herbicides and photosystem II inhibitors
  申请人：Dow AgroSciences, LLC

  公开号：US10455836B2

  公开（公告）日：2019-10-29

  Disclosed herein are herbicidal compositions comprising a herbicidally effective amount of (a) a pyridine carboxylic acid herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof, and (b) a photosystem II inhibitor, or an agriculturally acceptable salt or ester thereof. Also disclosed herein are methods of controlling undesirable vegetation which comprise applying to vegetation or an area adjacent the vegetation or applying to soil or water to prevent the emergence or growth of vegetation (a) a pyridine carboxylic acid herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof, and (b) a photosystem II inhibitor, or an agriculturally acceptable salt or ester thereof, wherein (a) and (b) are each added in an amount sufficient to provide a herbicidal effect.

  本文公开了除草组合物，该组合物包含除草有效量的(a)吡啶羧酸除草剂或其农业上可接受的 N-氧化物、盐或酯，以及(b)光系统 II 抑制剂或其农业上可接受的盐或酯。本文还公开了控制不良植被的方法，包括向植被或植被邻近区域施用，或向土壤或水中施用，以防止植被出现或生长：(a) 吡啶羧酸除草剂或其农业上可接受的 N-氧化物、盐或酯；(b) 光系统 II 抑制剂或其农业上可接受的盐或酯，其中(a)和(b)的添加量足以提供除草效果。
• Synergistic weed control from applications of pyridine carboxylic acid herbicides and ALS inhibitors
  申请人：Dow AgroSciences LLC

  公开号：US10448638B2

  公开（公告）日：2019-10-22

  Disclosed herein are herbicidal compositions comprising a herbicidally effective amount of (a) a pyridine carboxylic acid herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof, and (b) an acetolactate synthase (ALS) inhibitor or an agriculturally acceptable salt or ester thereof. Also disclosed herein are methods of controlling undesirable vegetation which comprise applying to vegetation or an area adjacent the vegetation or applying to soil or water to prevent the emergence or growth of vegetation (a) a pyridine carboxylic acid herbicide or an agriculturally acceptable N-oxide, salt, or ester thereof, and (b) an acetolactate synthase (ALS) inhibitor or an agriculturally acceptable salt or ester thereof, wherein (a) and (b) are each added in an amount sufficient to provide a herbicidal effect.

  本文公开的除草组合物包含除草有效量的(a)吡啶羧酸除草剂或其农业上可接受的 N-氧化物、盐或酯，和(b)乙酰乳酸合成酶(ALS)抑制剂或其农业上可接受的盐或酯。本文还公开了控制不良植被的方法，包括向植被或植被邻近区域施用或向土壤或水中施用以防止植被出现或生长 (a) 吡啶羧酸除草剂或其农业上可接受的 N-氧化物、盐或酯，以及 (b) 乙酰乳酸合成酶 (ALS) 抑制剂或其农业上可接受的盐或酯，其中 (a) 和 (b) 的添加量足以提供除草效果。