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中文名称 英文名称 CAS号 化学式 结构式图片
—— (E)-1-(4-bromophenyl)-3-[(1R)-6-hydroxy-7-methoxy-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl]prop-2-en-1-one —— C20H20BrNO3
(E)-1-(4-bromophenyl)-3-[(1R)-6-hydroxy-7-methoxy-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl]prop-2-en-1-one
—— (E)-N-[3-methyl-2-(pyrrolidine-1-carbonyl)phenyl]-3-quinolin-8-ylprop-2-enamide —— C24H23N3O2
(E)-N-[3-methyl-2-(pyrrolidine-1-carbonyl)phenyl]-3-quinolin-8-ylprop-2-enamide
—— (E)-3-(2,5-dimethoxyphenyl)-N-[[6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]prop-2-enamide —— C23H29N3O4
(E)-3-(2,5-dimethoxyphenyl)-N-[[6-[(2S,6S)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]prop-2-enamide
—— ethyl (2E,5R)-2-[(3-chloro-4-hydroxy-5-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H21ClN2O5S
ethyl (2E,5R)-2-[(3-chloro-4-hydroxy-5-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5R)-2-[(1,3-dimethylpyrazol-4-yl)methylidene]-5-(4-hydroxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C22H22N4O4S
ethyl (2E,5R)-2-[(1,3-dimethylpyrazol-4-yl)methylidene]-5-(4-hydroxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C20H27N3O3
(E)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— Ethyl 2-[(5-propylthiophene-3-carbonyl)amino]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate —— C21H27NO3S2
Ethyl 2-[(5-propylthiophene-3-carbonyl)amino]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophene-3-carboxylate
—— ethyl (6R)-6-ethyl-2-[[5-(5-ethylthiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H27F3N4O3S2
ethyl (6R)-6-ethyl-2-[[5-(5-ethylthiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (2E,5S)-2-[(3-chloro-4-hydroxy-5-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H21ClN2O5S
ethyl (2E,5S)-2-[(3-chloro-4-hydroxy-5-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (6R)-2-[[2-(5-ethylthiophen-2-yl)quinoline-4-carbonyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C28H28N2O3S2
ethyl (6R)-2-[[2-(5-ethylthiophen-2-yl)quinoline-4-carbonyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-(7-methyl-5-oxo-1,2,3,4,9,11-hexahydroisochromeno[4,3-g][1,3]benzoxazin-10-yl)benzoate —— C25H25NO5
Ethyl 2-(7-methyl-5-oxo-1,2,3,4,9,11-hexahydroisochromeno[4,3-g][1,3]benzoxazin-10-yl)benzoate
—— Ethyl 2-[(5-methyl-4-phenylthiophene-3-carbonyl)amino]-5-phenylthiophene-3-carboxylate —— C25H21NO3S2
Ethyl 2-[(5-methyl-4-phenylthiophene-3-carbonyl)amino]-5-phenylthiophene-3-carboxylate
—— ethyl (2E,5S)-5-(4-fluorophenyl)-7-methyl-3-oxo-2-[(5-phenyl-1H-pyrazol-4-yl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H21FN4O3S
ethyl (2E,5S)-5-(4-fluorophenyl)-7-methyl-3-oxo-2-[(5-phenyl-1H-pyrazol-4-yl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(2,5-dimethoxyphenyl)-N-[[6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]prop-2-enamide —— C23H29N3O4
(E)-3-(2,5-dimethoxyphenyl)-N-[[6-[(2S,6R)-2,6-dimethylmorpholin-4-yl]pyridin-3-yl]methyl]prop-2-enamide
—— (E)-3-[(1R,6S)-2,6-dimethylcyclohex-2-en-1-yl]prop-2-enoic acid —— C11H16O2
(E)-3-[(1R,6S)-2,6-dimethylcyclohex-2-en-1-yl]prop-2-enoic acid
—— ethyl 2-[[4-[(2-bromophenoxy)methyl]benzoyl]amino]-5-[(1R)-1-phenylethyl]thiophene-3-carboxylate —— C29H26BrNO4S
ethyl 2-[[4-[(2-bromophenoxy)methyl]benzoyl]amino]-5-[(1R)-1-phenylethyl]thiophene-3-carboxylate
—— ethyl (4S)-2-amino-4-[5-[(4-chloro-2-methylphenoxy)methyl]-2,4-dimethylphenyl]-5-oxo-4,6,7,8-tetrahydrochromene-3-carboxylate —— C28H30ClNO5
ethyl (4S)-2-amino-4-[5-[(4-chloro-2-methylphenoxy)methyl]-2,4-dimethylphenyl]-5-oxo-4,6,7,8-tetrahydrochromene-3-carboxylate
—— (E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C23H32N4O2
(E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— (E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C19H29N3O5S
(E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— ethyl 4-[[(3R,3aR,4aR,5R,8aS,9aS)-8a-methyl-2-oxospiro[3a,4,4a,6,7,8,9,9a-octahydro-3H-benzo[f][1]benzofuran-5,2'-oxirane]-3-yl]methyl]piperazine-1-carboxylate —— C22H34N2O5
ethyl 4-[[(3R,3aR,4aR,5R,8aS,9aS)-8a-methyl-2-oxospiro[3a,4,4a,6,7,8,9,9a-octahydro-3H-benzo[f][1]benzofuran-5,2'-oxirane]-3-yl]methyl]piperazine-1-carboxylate
—— ethyl (2R)-2-cyano-2-[3-(3,5-ditert-butyl-4-hydroxyphenyl)-1,4-dioxonaphthalen-2-yl]acetate —— C29H31NO5
ethyl (2R)-2-cyano-2-[3-(3,5-ditert-butyl-4-hydroxyphenyl)-1,4-dioxonaphthalen-2-yl]acetate
—— ethyl 2-({3-[(4-chlorophenoxy)methyl]benzoyl}amino)-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C26H26ClNO4S
ethyl 2-({3-[(4-chlorophenoxy)methyl]benzoyl}amino)-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— (E)-1-[(4aR,8aR)-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-3-phenylprop-2-en-1-one —— C18H23NO2
(E)-1-[(4aR,8aR)-4a-hydroxy-1,3,4,5,6,7,8,8a-octahydroisoquinolin-2-yl]-3-phenylprop-2-en-1-one
—— ethyl 2-{[({4-[(4-bromo-1H-pyrazol-1-yl)methyl]benzoyl}amino)carbothioyl]amino}-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C24H25BrN4O3S2
ethyl 2-{[({4-[(4-bromo-1H-pyrazol-1-yl)methyl]benzoyl}amino)carbothioyl]amino}-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— (E)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide —— C20H27N3O3
(E)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]-3-[4-(2-oxopyrrolidin-1-yl)phenyl]prop-2-enamide
—— ethyl (2Z,5S)-2-[[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H32N2O5S
ethyl (2Z,5S)-2-[[3-[(2,3-dimethylphenoxy)methyl]-4-methoxyphenyl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (6S)-6-methyl-2-[[2-(3-propan-2-yloxyphenyl)quinoline-4-carbonyl]carbamothioylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C32H33N3O4S2
ethyl (6S)-6-methyl-2-[[2-(3-propan-2-yloxyphenyl)quinoline-4-carbonyl]carbamothioylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-({[2-(2-methoxyphenyl)-4-quinolinyl]carbonyl}amino)-4-(4-methylphenyl)-3-thiophenecarboxylate —— C31H26N2O4S
Ethyl 2-({[2-(2-methoxyphenyl)-4-quinolinyl]carbonyl}amino)-4-(4-methylphenyl)-3-thiophenecarboxylate
—— Ethyl 4-(4-cyclohexylphenyl)-2-({4-nitrobenzoyl}amino)-5-methyl-3-thiophenecarboxylate —— C27H28N2O5S
Ethyl 4-(4-cyclohexylphenyl)-2-({4-nitrobenzoyl}amino)-5-methyl-3-thiophenecarboxylate
—— (E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C23H32N4O2
(E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— (E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C21H28N4O2
(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— ethyl (2Z,5S)-2-[[5-[(4-chloro-2-nitrophenoxy)methyl]furan-2-yl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H22ClN3O7S
ethyl (2Z,5S)-2-[[5-[(4-chloro-2-nitrophenoxy)methyl]furan-2-yl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (6R)-2-[(2-chloro-5-methylsulfanylbenzoyl)carbamothioylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H23ClN2O3S3
ethyl (6R)-2-[(2-chloro-5-methylsulfanylbenzoyl)carbamothioylamino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-(1,3-benzoxazol-2-yl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C17H21N3O3
(E)-3-(1,3-benzoxazol-2-yl)-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— ethyl 2-[(2-phenylquinoline-4-carbonyl)carbamothioylamino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C29H27N3O3S2
ethyl 2-[(2-phenylquinoline-4-carbonyl)carbamothioylamino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— (E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C21H26N4O3S
(E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(2R)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— ethyl (2Z,5S)-2-[[5-[(2,3-dichlorophenoxy)methyl]furan-2-yl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H22Cl2N2O5S
ethyl (2Z,5S)-2-[[5-[(2,3-dichlorophenoxy)methyl]furan-2-yl]methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide —— C21H26N4O3S
(E)-3-[2-(N-acetylanilino)-1,3-thiazol-4-yl]-N-[(2S)-1-morpholin-4-ylpropan-2-yl]prop-2-enamide
—— Ethyl 2-[[2-(4-chlorophenoxy)-2-methylpropanoyl]amino]-4-(4-methoxyphenyl)thiophene-3-carboxylate —— C24H24ClNO5S
Ethyl 2-[[2-(4-chlorophenoxy)-2-methylpropanoyl]amino]-4-(4-methoxyphenyl)thiophene-3-carboxylate
—— ethyl (3R)-3-(aminomethyl)piperidine-1-carboxylate —— C9H18N2O2
ethyl (3R)-3-(aminomethyl)piperidine-1-carboxylate
—— (E)-1-[(3S)-3-(aminomethyl)piperidin-1-yl]but-2-en-1-one —— C10H18N2O
(E)-1-[(3S)-3-(aminomethyl)piperidin-1-yl]but-2-en-1-one
—— ethyl (2E,5S)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H25FN4O3S
ethyl (2E,5S)-2-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methylidene]-5-(4-fluorophenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 4-(3,4-dimethylphenyl)-5-methyl-2-[(5-methylthiophene-2-carbonyl)amino]thiophene-3-carboxylate —— C22H23NO3S2
Ethyl 4-(3,4-dimethylphenyl)-5-methyl-2-[(5-methylthiophene-2-carbonyl)amino]thiophene-3-carboxylate
—— ethyl (6S)-6-methyl-2-[[2-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H27N3O3S3
ethyl (6S)-6-methyl-2-[[2-(5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-ylsulfanyl)acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-(2-piperidin-1-ylethyl)prop-2-enamide —— C19H29N3O4S
(E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N-(2-piperidin-1-ylethyl)prop-2-enamide
—— ethyl (2S)-2-[[(2Z)-2-[(2,3-dimethoxyphenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxy]propanoate —— C22H22O7
ethyl (2S)-2-[[(2Z)-2-[(2,3-dimethoxyphenyl)methylidene]-3-oxo-1-benzofuran-6-yl]oxy]propanoate
—— (E)-1-[(3R)-3-(aminomethyl)piperidin-1-yl]but-2-en-1-one —— C10H18N2O
(E)-1-[(3R)-3-(aminomethyl)piperidin-1-yl]but-2-en-1-one
—— Ethyl 2-({[7-(difluoromethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-3-yl]carbonyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C25H22F2N4O3S
Ethyl 2-({[7-(difluoromethyl)-5-phenylpyrazolo[1,5-a]pyrimidin-3-yl]carbonyl}amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (2S)-2-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbothioyl]amino]-3-phenylpropanoate —— C23H27N3O3S
ethyl (2S)-2-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbothioyl]amino]-3-phenylpropanoate
—— ethyl (4R)-2-amino-4-[3-[(3-chloro-4-fluorophenoxy)methyl]-4-methoxyphenyl]-7,7-dimethyl-5-oxo-6,8-dihydro-4H-chromene-3-carboxylate —— C28H29ClFNO6
ethyl (4R)-2-amino-4-[3-[(3-chloro-4-fluorophenoxy)methyl]-4-methoxyphenyl]-7,7-dimethyl-5-oxo-6,8-dihydro-4H-chromene-3-carboxylate