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—— ethyl (2E,5S)-2-[(2-chloro-4,5-dimethoxyphenyl)methylidene]-5-(3-methoxy-4-methylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27ClN2O6S
ethyl (2E,5S)-2-[(2-chloro-4,5-dimethoxyphenyl)methylidene]-5-(3-methoxy-4-methylphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N,N-bis(prop-2-enyl)prop-2-enamide —— C18H24N2O4S
(E)-3-[3-(dimethylsulfamoyl)-4-methoxyphenyl]-N,N-bis(prop-2-enyl)prop-2-enamide
—— (E)-N-[2-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C22H22N6O3
(E)-N-[2-[3-(5-amino-4-cyano-1-phenylpyrazol-3-yl)propylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl 6-[4-[3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]propanoyl]piperazin-1-yl]pyridine-3-carboxylate —— C23H29N3O4
ethyl 6-[4-[3-[5-[(1R,2S)-2-methylcyclopropyl]furan-2-yl]propanoyl]piperazin-1-yl]pyridine-3-carboxylate
—— ethyl 4-[(3R)-5-acetyl-3-[5-chloro-2-[(2-chlorophenyl)methoxy]phenyl]-4-phenyl-3H-1,2,4-triazol-2-yl]benzoate —— C32H27Cl2N3O4
ethyl 4-[(3R)-5-acetyl-3-[5-chloro-2-[(2-chlorophenyl)methoxy]phenyl]-4-phenyl-3H-1,2,4-triazol-2-yl]benzoate
—— ethyl 5-[(3-chlorophenyl)carbamoyl]-4-methyl-2-[[(2R)-2,3,3,3-tetrafluoro-2-methoxypropanoyl]amino]thiophene-3-carboxylate —— C19H17ClF4N2O5S
ethyl 5-[(3-chlorophenyl)carbamoyl]-4-methyl-2-[[(2R)-2,3,3,3-tetrafluoro-2-methoxypropanoyl]amino]thiophene-3-carboxylate
—— ethyl (2E,5S)-2-[(5-bromo-2-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H21BrN2O4S
ethyl (2E,5S)-2-[(5-bromo-2-methoxyphenyl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— Ethyl 4-(4-methoxy-2,6-dimethylphenyl)sulfonylpiperazine-1-carboxylate —— C16H24N2O5S
Ethyl 4-(4-methoxy-2,6-dimethylphenyl)sulfonylpiperazine-1-carboxylate
—— ethyl (2E,5S)-2-[[2-[(2-fluorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C33H31FN2O4S
ethyl (2E,5S)-2-[[2-[(2-fluorophenyl)methoxy]phenyl]methylidene]-7-methyl-3-oxo-5-(4-propan-2-ylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 2-[(4R)-2-amino-4-(5-bromothiophen-2-yl)-3-cyano-7,7-dimethyl-5-oxo-6,8-dihydro-4H-quinolin-1-yl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C27H28BrN3O3S2
ethyl 2-[(4R)-2-amino-4-(5-bromothiophen-2-yl)-3-cyano-7,7-dimethyl-5-oxo-6,8-dihydro-4H-quinolin-1-yl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 2-[[6-[[2-(1-methyltetrazol-5-yl)sulfanylacetyl]amino]-1,3-benzothiazol-2-yl]sulfanyl]acetate —— C15H16N6O3S3
Ethyl 2-[[6-[[2-(1-methyltetrazol-5-yl)sulfanylacetyl]amino]-1,3-benzothiazol-2-yl]sulfanyl]acetate
—— ethyl (2Z,5R)-2-[(2-hydroxy-5-nitrophenyl)methylidene]-5-(3-methoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H23N3O7S
ethyl (2Z,5R)-2-[(2-hydroxy-5-nitrophenyl)methylidene]-5-(3-methoxyphenyl)-3-oxo-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5S)-5-(4-fluorophenyl)-7-methyl-3-oxo-2-[(2-prop-2-ynoxynaphthalen-1-yl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H23FN2O4S
ethyl (2Z,5S)-5-(4-fluorophenyl)-7-methyl-3-oxo-2-[(2-prop-2-ynoxynaphthalen-1-yl)methylidene]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5E)-2-[(4-tert-butylbenzoyl)amino]-5-[(3,5-dichloro-2-methoxyphenyl)methylidene]-4-oxothiophene-3-carboxylate —— C26H25Cl2NO5S
ethyl (5E)-2-[(4-tert-butylbenzoyl)amino]-5-[(3,5-dichloro-2-methoxyphenyl)methylidene]-4-oxothiophene-3-carboxylate
—— ethyl (6R)-6-methyl-2-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbothioyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H29N3O3S2
ethyl (6R)-6-methyl-2-[[(1R,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-diene-11-carbothioyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl (3S)-1-[[(3R,3aR,8aS,9aS)-5,8a-dimethyl-2-oxo-3,3a,4,6,7,8,9,9a-octahydrobenzo[f][1]benzofuran-3-yl]methyl]piperidin-1-ium-3-carboxylate —— C23H36NO4+
ethyl (3S)-1-[[(3R,3aR,8aS,9aS)-5,8a-dimethyl-2-oxo-3,3a,4,6,7,8,9,9a-octahydrobenzo[f][1]benzofuran-3-yl]methyl]piperidin-1-ium-3-carboxylate
—— ethyl (2R)-2-[(5E)-5-[(3-methoxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C16H17NO5S
ethyl (2R)-2-[(5E)-5-[(3-methoxyphenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— (E)-3-(4-chlorophenyl)-2-[1-(2-hydroxyethyl)pyridin-1-ium-4-yl]prop-2-ene-1-sulfonate —— C16H16ClNO4S
(E)-3-(4-chlorophenyl)-2-[1-(2-hydroxyethyl)pyridin-1-ium-4-yl]prop-2-ene-1-sulfonate
—— ethyl 1-[(2S)-2-(3-methylphenoxy)propanoyl]piperidine-4-carboxylate —— C18H25NO4
ethyl 1-[(2S)-2-(3-methylphenoxy)propanoyl]piperidine-4-carboxylate
—— ethyl 1-[(2S)-2-(4-methylphenoxy)propanoyl]piperidine-4-carboxylate —— C18H25NO4
ethyl 1-[(2S)-2-(4-methylphenoxy)propanoyl]piperidine-4-carboxylate
—— ethyl 1-[(2R)-2-(4-methylphenoxy)propanoyl]piperidine-4-carboxylate —— C18H25NO4
ethyl 1-[(2R)-2-(4-methylphenoxy)propanoyl]piperidine-4-carboxylate
—— ethyl (2E,5R)-2-[(5-bromothiophen-2-yl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H21BrN2O5S2
ethyl (2E,5R)-2-[(5-bromothiophen-2-yl)methylidene]-5-(3,4-dimethoxyphenyl)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2E,5S)-2-[[5-(2-methoxycarbonylphenyl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H24N2O6S2
ethyl (2E,5S)-2-[[5-(2-methoxycarbonylphenyl)furan-2-yl]methylidene]-3-oxo-7-phenyl-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl 1-[(2R)-2-(3-methylphenoxy)propanoyl]piperidine-4-carboxylate —— C18H25NO4
ethyl 1-[(2R)-2-(3-methylphenoxy)propanoyl]piperidine-4-carboxylate
—— Ethyl 1-[3-(2-chlorophenyl)propanoyl]piperidine-4-carboxylate —— C17H22ClNO3
Ethyl 1-[3-(2-chlorophenyl)propanoyl]piperidine-4-carboxylate
—— Ethyl 4-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}anilino)-4-oxobutanoate —— C16H19N3O6S
Ethyl 4-(4-{[(5-methyl-3-isoxazolyl)amino]sulfonyl}anilino)-4-oxobutanoate
—— ethyl 4-[[(2S)-2-[[(1S,2R,6R,8S,9R)-4,4,11,11-tetramethyl-3,5,7,10,12-pentaoxatricyclo[7.3.0.02,6]dodecane-8-carbonyl]amino]propanoyl]amino]benzoate —— C24H32N2O9
ethyl 4-[[(2S)-2-[[(1S,2R,6R,8S,9R)-4,4,11,11-tetramethyl-3,5,7,10,12-pentaoxatricyclo[7.3.0.02,6]dodecane-8-carbonyl]amino]propanoyl]amino]benzoate
—— (E,4E)-4-[(5-chlorofuran-2-yl)methylidene]-3-methylpent-2-enedioate —— C11H7ClO5-2
(E,4E)-4-[(5-chlorofuran-2-yl)methylidene]-3-methylpent-2-enedioate
—— ethyl 2-[[(2Z)-2-[[(2R)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-1-benzofuran-6-yl]oxy]acetate —— C23H20O6
ethyl 2-[[(2Z)-2-[[(2R)-2-methyl-2H-chromen-3-yl]methylidene]-3-oxo-1-benzofuran-6-yl]oxy]acetate
—— ethyl (4S)-6-amino-5-cyano-2-[(3-cyano-6-methyl-7,8-dihydro-5H-1,6-naphthyridin-2-yl)sulfanylmethyl]-4-pyridin-4-yl-4H-pyran-3-carboxylate —— C25H24N6O3S
ethyl (4S)-6-amino-5-cyano-2-[(3-cyano-6-methyl-7,8-dihydro-5H-1,6-naphthyridin-2-yl)sulfanylmethyl]-4-pyridin-4-yl-4H-pyran-3-carboxylate
—— Ethyl 2-[[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-5-(dimethylcarbamoyl)-4-methylthiophene-3-carboxylate —— C23H19ClF3N5O4S2
Ethyl 2-[[5-(5-chlorothiophen-2-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carbonyl]amino]-5-(dimethylcarbamoyl)-4-methylthiophene-3-carboxylate
—— Ethyl 4-(2,4-dichlorophenyl)-2-[(2,5-dimethyl-3-furoyl)amino]-3-thiophenecarboxylate —— C20H17Cl2NO4S
Ethyl 4-(2,4-dichlorophenyl)-2-[(2,5-dimethyl-3-furoyl)amino]-3-thiophenecarboxylate
—— ethyl 3-[[1-(4-fluorophenyl)-6-oxopyridazine-3-carbonyl]amino]benzoate —— C20H16FN3O4
ethyl 3-[[1-(4-fluorophenyl)-6-oxopyridazine-3-carbonyl]amino]benzoate
—— ethyl (6S)-6-methyl-2-(9H-xanthene-9-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C26H25NO4S
ethyl (6S)-6-methyl-2-(9H-xanthene-9-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-3-(furan-2-yl)-N-[2-[[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]prop-2-enamide —— C21H22N4O4
(E)-3-(furan-2-yl)-N-[2-[[(S)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]prop-2-enamide
—— ethyl 2-[({[3-cyano-4-(4-methoxyphenyl)-6-(2-thienyl)-2-pyridinyl]sulfanyl}acetyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C29H25N3O4S3
ethyl 2-[({[3-cyano-4-(4-methoxyphenyl)-6-(2-thienyl)-2-pyridinyl]sulfanyl}acetyl)amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl (2Z,5S)-5-(4-ethoxyphenyl)-2-[(4-hydroxy-3-methoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26N2O6S
ethyl (2Z,5S)-5-(4-ethoxyphenyl)-2-[(4-hydroxy-3-methoxyphenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E,4Z)-4-[(2,4-dimethoxyphenyl)methylidene]-3-methylpent-2-enedioate —— C15H14O6-2
(E,4Z)-4-[(2,4-dimethoxyphenyl)methylidene]-3-methylpent-2-enedioate
—— Ethyl 2-({[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]carbonyl}amino)-4-(1-naphthyl)-3-thiophenecarboxylate —— C28H20ClFN2O4S
Ethyl 2-({[3-(2-chloro-6-fluorophenyl)-5-methyl-4-isoxazolyl]carbonyl}amino)-4-(1-naphthyl)-3-thiophenecarboxylate
—— ethyl (2S)-2-[(5Z)-5-[[1-(4-iodophenyl)pyrrol-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate —— C19H17IN2O4S
ethyl (2S)-2-[(5Z)-5-[[1-(4-iodophenyl)pyrrol-2-yl]methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]propanoate
—— ethyl 2-[[1-(2-phenoxyacetyl)piperidine-4-carbonyl]amino]benzoate —— C23H26N2O5
ethyl 2-[[1-(2-phenoxyacetyl)piperidine-4-carbonyl]amino]benzoate
—— (E)-3-(2,3-dimethoxyphenyl)-N-[(2R)-3-ethyl-2-morpholin-4-ylpentyl]prop-2-enamide —— C22H34N2O4
(E)-3-(2,3-dimethoxyphenyl)-N-[(2R)-3-ethyl-2-morpholin-4-ylpentyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[(2-pyrrolidin-1-ylpyridin-4-yl)methylamino]ethyl]prop-2-enamide —— C19H22N4O3
(E)-3-(furan-2-yl)-N-[2-oxo-2-[(2-pyrrolidin-1-ylpyridin-4-yl)methylamino]ethyl]prop-2-enamide
—— Ethyl 2-{[(4-bromophenoxy)acetyl]amino}-4-(4-fluorophenyl)-5-methyl-3-thiophenecarboxylate —— C22H19BrFNO4S
Ethyl 2-{[(4-bromophenoxy)acetyl]amino}-4-(4-fluorophenyl)-5-methyl-3-thiophenecarboxylate
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[3-(2-pyridin-2-ylethynyl)anilino]ethyl]prop-2-enamide —— C22H17N3O3
(E)-3-(furan-2-yl)-N-[2-oxo-2-[3-(2-pyridin-2-ylethynyl)anilino]ethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[3-[(2-methoxyacetyl)amino]anilino]-2-oxoethyl]prop-2-enamide —— C18H19N3O5
(E)-3-(furan-2-yl)-N-[2-[3-[(2-methoxyacetyl)amino]anilino]-2-oxoethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[2-(2-oxopyrrolidin-1-yl)anilino]ethyl]prop-2-enamide —— C19H19N3O4
(E)-3-(furan-2-yl)-N-[2-oxo-2-[2-(2-oxopyrrolidin-1-yl)anilino]ethyl]prop-2-enamide
—— (E)-N-[2-[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C20H19N3O3S
(E)-N-[2-[(2R)-2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl (3R)-1-[5-(2-chlorophenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxylate —— C18H19ClN2O4
ethyl (3R)-1-[5-(2-chlorophenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxylate
—— (E)-N-[2-[[(R)-(4-chlorophenyl)-phenylmethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C22H19ClN2O3
(E)-N-[2-[[(R)-(4-chlorophenyl)-phenylmethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide