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—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[(1-pyridin-2-ylpiperidin-4-yl)amino]ethyl]prop-2-enamide —— C19H22N4O3
(E)-3-(furan-2-yl)-N-[2-oxo-2-[(1-pyridin-2-ylpiperidin-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C22H25N3O4
(E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 2-[[2-[(4R)-4-[4-(difluoromethoxy)phenyl]-4-methyl-2,5-dioxoimidazolidin-1-yl]acetyl]amino]-4,5-dimethylthiophene-3-carboxylate —— C22H23F2N3O6S
ethyl 2-[[2-[(4R)-4-[4-(difluoromethoxy)phenyl]-4-methyl-2,5-dioxoimidazolidin-1-yl]acetyl]amino]-4,5-dimethylthiophene-3-carboxylate
—— (E)-3-(3-fluorophenyl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoic acid —— C18H18FNO4S2
(E)-3-(3-fluorophenyl)-2-(5-piperidin-1-ylsulfonylthiophen-2-yl)prop-2-enoic acid
—— (E)-3-[4-(cyclopropylsulfamoyl)phenyl]-N-[(5-ethylthiophen-2-yl)methyl]prop-2-enamide —— C19H22N2O3S2
(E)-3-[4-(cyclopropylsulfamoyl)phenyl]-N-[(5-ethylthiophen-2-yl)methyl]prop-2-enamide
—— ethyl (6R)-6-methyl-2-[(5-nitrofuran-2-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C17H18N2O6S
ethyl (6R)-6-methyl-2-[(5-nitrofuran-2-carbonyl)amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-(1-pyridin-2-ylpiperidin-4-yl)-3-[4-(trifluoromethylsulfanyl)phenyl]prop-2-enamide —— C20H20F3N3OS
(E)-N-(1-pyridin-2-ylpiperidin-4-yl)-3-[4-(trifluoromethylsulfanyl)phenyl]prop-2-enamide
—— (E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)prop-2-enamide —— C23H26N4OS
(E)-3-[3,5-dimethyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)prop-2-enamide
—— Ethyl 5-[(4-methylphenyl)sulfonylamino]-2-propyl-1-benzofuran-3-carboxylate —— C21H23NO5S
Ethyl 5-[(4-methylphenyl)sulfonylamino]-2-propyl-1-benzofuran-3-carboxylate
—— (E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C24H29N3O3
(E)-3-[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-3-[5-(4-fluorophenyl)thiophen-2-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C22H21FN4OS
(E)-3-[5-(4-fluorophenyl)thiophen-2-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(2-bromophenyl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C18H19BrN4O
(E)-3-(2-bromophenyl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 2-[[2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C18H17N3O4S3
ethyl 2-[[2-[(5-thiophen-2-yl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 2-[[2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C21H23N5O4S2
ethyl 2-[[2-[[4-amino-5-(2-methoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl (3S)-3-(3-bromophenyl)-2,2-difluoro-3-[(3-methoxydibenzofuran-2-yl)amino]propanoate —— C24H20BrF2NO4
ethyl (3S)-3-(3-bromophenyl)-2,2-difluoro-3-[(3-methoxydibenzofuran-2-yl)amino]propanoate
—— ethyl (6S)-6-methyl-2-[[(2S)-2-morpholin-4-ium-4-ylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C19H29N2O4S+
ethyl (6S)-6-methyl-2-[[(2S)-2-morpholin-4-ium-4-ylpropanoyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— Ethyl 5-[(4-ethoxyphenyl)sulfonylamino]-2-phenyl-1-benzofuran-3-carboxylate —— C25H23NO6S
Ethyl 5-[(4-ethoxyphenyl)sulfonylamino]-2-phenyl-1-benzofuran-3-carboxylate
—— (E)-N-benzhydryl-N-methyl-3-thiophen-2-ylprop-2-enamide —— C21H19NOS
(E)-N-benzhydryl-N-methyl-3-thiophen-2-ylprop-2-enamide
—— ethyl 4-[(2R)-3-[furan-2-ylmethyl(2-methoxyethyl)amino]-2-hydroxypropoxy]benzoate —— C20H27NO6
ethyl 4-[(2R)-3-[furan-2-ylmethyl(2-methoxyethyl)amino]-2-hydroxypropoxy]benzoate
—— (E)-3-(2-methoxy-5-methylphenyl)-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C21H25N3O2
(E)-3-(2-methoxy-5-methylphenyl)-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C23H26ClN3O7S2
ethyl 2-[[2-[(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]prop-2-enoyl]oxyacetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 6-[(6-chloro-3,4-dihydro-2H-quinolin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C17H20ClN3O3
ethyl 6-[(6-chloro-3,4-dihydro-2H-quinolin-1-yl)methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-N-(1-pyrimidin-2-ylpiperidin-4-yl)-3-[2-(trifluoromethoxy)phenyl]prop-2-enamide —— C19H19F3N4O2
(E)-N-(1-pyrimidin-2-ylpiperidin-4-yl)-3-[2-(trifluoromethoxy)phenyl]prop-2-enamide
—— (E)-N-[[4-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C21H27N3OS
(E)-N-[[4-[[(2S)-2-methylpiperidin-1-yl]methyl]phenyl]methyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— (E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C21H24N4O4
(E)-3-(5-methoxy-2,3-dihydro-1,4-benzodioxin-7-yl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 2,5-dimethyl-4-[2-(5-nitro-1,3-dioxoisoindol-2-yl)acetyl]-1H-pyrrole-3-carboxylate —— C19H17N3O7
ethyl 2,5-dimethyl-4-[2-(5-nitro-1,3-dioxoisoindol-2-yl)acetyl]-1H-pyrrole-3-carboxylate
—— (E)-3-(4-ethoxy-3-methoxyphenyl)-N-[[4-(propan-2-ylcarbamoylamino)phenyl]methyl]prop-2-enamide —— C23H29N3O4
(E)-3-(4-ethoxy-3-methoxyphenyl)-N-[[4-(propan-2-ylcarbamoylamino)phenyl]methyl]prop-2-enamide
—— (E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide —— C24H29N3O3
(E)-3-[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]-N-(1-pyridin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 4-[(2S)-3-[furan-2-ylmethyl(2-methoxyethyl)amino]-2-hydroxypropoxy]benzoate —— C20H27NO6
ethyl 4-[(2S)-3-[furan-2-ylmethyl(2-methoxyethyl)amino]-2-hydroxypropoxy]benzoate
—— ethyl 5-[4-[(2E,4E)-hexa-2,4-dienoyl]piperazin-1-yl]sulfonylfuran-2-carboxylate —— C17H22N2O6S
ethyl 5-[4-[(2E,4E)-hexa-2,4-dienoyl]piperazin-1-yl]sulfonylfuran-2-carboxylate
—— (E)-3-(4-methoxyphenyl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide —— C18H26N2O4S
(E)-3-(4-methoxyphenyl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide
—— (E)-N-prop-2-enyl-3-quinoxalin-2-ylprop-2-enamide —— C14H13N3O
(E)-N-prop-2-enyl-3-quinoxalin-2-ylprop-2-enamide
—— ethyl 1-ethyl-2,5-dimethyl-4-[(Z)-3-[2-methyl-4-(methylcarbamoyl)anilino]-3-oxoprop-1-enyl]pyrrole-3-carboxylate —— C23H29N3O4
ethyl 1-ethyl-2,5-dimethyl-4-[(Z)-3-[2-methyl-4-(methylcarbamoyl)anilino]-3-oxoprop-1-enyl]pyrrole-3-carboxylate
—— (E)-3-(2-fluorophenyl)-N-[[3-(piperidine-1-carbonyl)phenyl]methyl]prop-2-enamide —— C22H23FN2O2
(E)-3-(2-fluorophenyl)-N-[[3-(piperidine-1-carbonyl)phenyl]methyl]prop-2-enamide
—— (E)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-[[4-(propan-2-ylcarbamoylamino)phenyl]methyl]prop-2-enamide —— C20H25N5O4
(E)-3-(1,3-dimethyl-2,4-dioxopyrimidin-5-yl)-N-[[4-(propan-2-ylcarbamoylamino)phenyl]methyl]prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[(2S)-2-(4-phenylpiperazin-1-yl)propyl]prop-2-enamide —— C22H26FN3O
(E)-3-(4-fluorophenyl)-N-[(2S)-2-(4-phenylpiperazin-1-yl)propyl]prop-2-enamide
—— (E)-3-(3-ethoxy-4-methoxyphenyl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide —— C20H30N2O5S
(E)-3-(3-ethoxy-4-methoxyphenyl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide
—— (E)-3-[4-(difluoromethoxy)phenyl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C19H20F2N4O2
(E)-3-[4-(difluoromethoxy)phenyl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(3,5-dichlorophenyl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C18H18Cl2N4O
(E)-3-(3,5-dichlorophenyl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(2,4-dimethylphenyl)-1-[4-(5-nitrothiophene-2-carbonyl)piperazin-1-yl]prop-2-en-1-one —— C20H21N3O4S
(E)-3-(2,4-dimethylphenyl)-1-[4-(5-nitrothiophene-2-carbonyl)piperazin-1-yl]prop-2-en-1-one
—— (E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(2,4-dimethylphenyl)prop-2-en-1-one —— C19H21BrN4O
(E)-1-[4-(5-bromopyrimidin-2-yl)piperazin-1-yl]-3-(2,4-dimethylphenyl)prop-2-en-1-one
—— (E)-3-(3,5-dimethoxyphenyl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C20H24N4O3
(E)-3-(3,5-dimethoxyphenyl)-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 5-[4-[(2Z,4Z)-hexa-2,4-dienoyl]piperazin-1-yl]sulfonylfuran-2-carboxylate —— C17H22N2O6S
ethyl 5-[4-[(2Z,4Z)-hexa-2,4-dienoyl]piperazin-1-yl]sulfonylfuran-2-carboxylate
—— (E)-3-(3-fluoro-4-methoxyphenyl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide —— C18H25FN2O4S
(E)-3-(3-fluoro-4-methoxyphenyl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(4-cyanophenyl)-N-[[2-(phenylmethoxymethyl)phenyl]methyl]prop-2-enamide —— C25H22N2O2
(E)-3-(4-cyanophenyl)-N-[[2-(phenylmethoxymethyl)phenyl]methyl]prop-2-enamide
—— (E)-3-[4-(cyanomethoxy)phenyl]-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide —— C19H25N3O4S
(E)-3-[4-(cyanomethoxy)phenyl]-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(2S)-2-[(2S)-2-methylpiperidin-1-yl]propyl]prop-2-enamide —— C19H26N2O3
(E)-3-(1,3-benzodioxol-5-yl)-N-[(2S)-2-[(2S)-2-methylpiperidin-1-yl]propyl]prop-2-enamide
—— (E)-3-(1,3-benzoxazol-2-yl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide —— C18H23N3O4S
(E)-3-(1,3-benzoxazol-2-yl)-N-(1-propylsulfonylpiperidin-4-yl)prop-2-enamide
—— (E)-3-[5-(2-fluorophenyl)furan-2-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide —— C22H21FN4O2
(E)-3-[5-(2-fluorophenyl)furan-2-yl]-N-(1-pyrimidin-2-ylpiperidin-4-yl)prop-2-enamide
—— ethyl 1-ethyl-2,5-dimethyl-4-[(E)-3-[2-methyl-4-(methylcarbamoyl)anilino]-3-oxoprop-1-enyl]pyrrole-3-carboxylate —— C23H29N3O4
ethyl 1-ethyl-2,5-dimethyl-4-[(E)-3-[2-methyl-4-(methylcarbamoyl)anilino]-3-oxoprop-1-enyl]pyrrole-3-carboxylate