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—— (E)-1-[4-[(4R,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]piperidin-1-yl]-3-phenylprop-2-en-1-one —— C25H34N2O2
(E)-1-[4-[(4R,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]piperidin-1-yl]-3-phenylprop-2-en-1-one
—— ethyl 2-[[4-(dimethylsulfamoyl)benzoyl]amino]-3-(methylcarbamoylcarbamoyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate —— C22H27N5O7S2
ethyl 2-[[4-(dimethylsulfamoyl)benzoyl]amino]-3-(methylcarbamoylcarbamoyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxylate
—— (E)-ethyl 2-((4-cyanobenzoyl)imino)-3-methyl-2,3-dihydrobenzo[d]thiazole-6-carboxylate —— C19H15N3O3S
(E)-ethyl 2-((4-cyanobenzoyl)imino)-3-methyl-2,3-dihydrobenzo[d]thiazole-6-carboxylate
—— ethyl 4-[4-[[(1R,2R)-2-methylcyclopropanecarbonyl]amino]benzoyl]oxypiperidine-1-carboxylate —— C20H26N2O5
ethyl 4-[4-[[(1R,2R)-2-methylcyclopropanecarbonyl]amino]benzoyl]oxypiperidine-1-carboxylate
—— Ethyl 2-[[2-(2,4-dimethylphenyl)quinoline-4-carbonyl]amino]-4-(4-fluorophenyl)thiophene-3-carboxylate —— C31H25FN2O3S
Ethyl 2-[[2-(2,4-dimethylphenyl)quinoline-4-carbonyl]amino]-4-(4-fluorophenyl)thiophene-3-carboxylate
—— ethyl 4-[4-[[(1R,2S)-2-methylcyclopropanecarbonyl]amino]benzoyl]oxypiperidine-1-carboxylate —— C20H26N2O5
ethyl 4-[4-[[(1R,2S)-2-methylcyclopropanecarbonyl]amino]benzoyl]oxypiperidine-1-carboxylate
—— (E)-N-[3-[4-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-oxopropyl]-3-(furan-2-yl)prop-2-enamide —— C22H31N3O5
(E)-N-[3-[4-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-oxopropyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl 2-(4-oxo-4H-chromene-3-carboxamido)thiazole-4-carboxylate —— C16H12N2O5S
ethyl 2-(4-oxo-4H-chromene-3-carboxamido)thiazole-4-carboxylate
—— Ethyl 2-[[2-(4-bromobenzoyl)oxyacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H22BrNO5S
Ethyl 2-[[2-(4-bromobenzoyl)oxyacetyl]amino]-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(1S)-1-[2-(difluoromethoxy)phenyl]propyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C17H18F2N2O2S
(E)-N-[(1S)-1-[2-(difluoromethoxy)phenyl]propyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— ethyl 2-[[2-(2-ethoxy-2-oxoethyl)sulfanylacetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate —— C18H25NO5S2
ethyl 2-[[2-(2-ethoxy-2-oxoethyl)sulfanylacetyl]amino]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophene-3-carboxylate
—— (E)-N-[(1R)-1-[2-(difluoromethoxy)phenyl]propyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide —— C17H18F2N2O2S
(E)-N-[(1R)-1-[2-(difluoromethoxy)phenyl]propyl]-3-(2-methyl-1,3-thiazol-4-yl)prop-2-enamide
—— Ethyl 2-[[(2-methoxyphenyl)methyl-(1-methylpiperidin-4-yl)carbamothioyl]amino]acetate —— C19H29N3O3S
Ethyl 2-[[(2-methoxyphenyl)methyl-(1-methylpiperidin-4-yl)carbamothioyl]amino]acetate
—— (E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-cyclopropyl-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide —— C24H26N2O4
(E)-3-[4-(cyanomethoxy)-3-methoxyphenyl]-N-cyclopropyl-N-[[5-[(1R,2R)-2-methylcyclopropyl]furan-2-yl]methyl]prop-2-enamide
—— (E)-3-(3-fluorophenyl)-N-[3-(2-oxo-2-pyrrolidin-1-ylethoxy)phenyl]prop-2-enamide —— C21H21FN2O3
(E)-3-(3-fluorophenyl)-N-[3-(2-oxo-2-pyrrolidin-1-ylethoxy)phenyl]prop-2-enamide
—— (E)-1-[4-[(4S,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]piperidin-1-yl]-3-phenylprop-2-en-1-one —— C25H34N2O2
(E)-1-[4-[(4S,4aR,8aS)-4-methyl-3,4,4a,5,6,7,8,8a-octahydro-2H-quinoline-1-carbonyl]piperidin-1-yl]-3-phenylprop-2-en-1-one
—— ethyl 1'-benzyl-2-(2,2-diphenylacetyl)spiro[4,9-dihydro-3H-pyrido[3,4-b]indole-1,4'-piperidine]-3'-carboxylate —— C39H39N3O3
ethyl 1'-benzyl-2-(2,2-diphenylacetyl)spiro[4,9-dihydro-3H-pyrido[3,4-b]indole-1,4'-piperidine]-3'-carboxylate
—— (E)-3-(1,3-benzodioxol-5-yl)-N-[(2R)-3-methylbutan-2-yl]prop-2-enamide —— C15H19NO3
(E)-3-(1,3-benzodioxol-5-yl)-N-[(2R)-3-methylbutan-2-yl]prop-2-enamide
—— Ethyl 2-[4-[benzyl(ethyl)sulfamoyl]benzoyl]imino-3-(2-ethoxy-2-oxoethyl)-1,3-benzothiazole-6-carboxylate —— C30H31N3O7S2
Ethyl 2-[4-[benzyl(ethyl)sulfamoyl]benzoyl]imino-3-(2-ethoxy-2-oxoethyl)-1,3-benzothiazole-6-carboxylate
—— ethyl 2-(2-methylpropanoylamino)-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate —— C17H26N2O3S
ethyl 2-(2-methylpropanoylamino)-6-propan-2-yl-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carboxylate
—— ethyl 5-(3-((furan-2-ylmethyl)amino)-2-hydroxypropoxy)-2-methyl-1-(p-tolyl)-1H-indole-3-carboxylate —— C27H30N2O5
ethyl 5-(3-((furan-2-ylmethyl)amino)-2-hydroxypropoxy)-2-methyl-1-(p-tolyl)-1H-indole-3-carboxylate
—— Ethyl 6-methyl-2-[[2-(2,2,2-trichloroacetyl)oxyacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C16H18Cl3NO5S
Ethyl 6-methyl-2-[[2-(2,2,2-trichloroacetyl)oxyacetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— ethyl 2-((Z)-2-(((Z)-3-(4-nitrophenyl)acryloyl)imino)-6-sulfamoylbenzo[d]thiazol-3(2H)-yl)acetate —— C20H18N4O7S2
ethyl 2-((Z)-2-(((Z)-3-(4-nitrophenyl)acryloyl)imino)-6-sulfamoylbenzo[d]thiazol-3(2H)-yl)acetate
—— ethyl 2-(4-ethoxyanilino)-5-[(3-ethoxy-4-prop-2-enoxyphenyl)methylidene]-4-oxothiophene-3-carboxylate —— C27H29NO6S
ethyl 2-(4-ethoxyanilino)-5-[(3-ethoxy-4-prop-2-enoxyphenyl)methylidene]-4-oxothiophene-3-carboxylate
—— Ethyl 4-(3,4-dimethoxyphenyl)-6-(3-nitrophenyl)-2-oxocyclohex-3-ene-1-carboxylate —— C23H23NO7
Ethyl 4-(3,4-dimethoxyphenyl)-6-(3-nitrophenyl)-2-oxocyclohex-3-ene-1-carboxylate
—— Ethyl 2-(2-{[4-(4-ethoxyphenyl)-5-{[(2-fluorophenyl)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}acetamido)-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate —— C30H30FN5O5S2
Ethyl 2-(2-{[4-(4-ethoxyphenyl)-5-{[(2-fluorophenyl)formamido]methyl}-4H-1,2,4-triazol-3-YL]sulfanyl}acetamido)-4H,5H,6H-cyclopenta[B]thiophene-3-carboxylate
—— Ethyl 5-(4-bromobenzamido)-3-(4-fluorophenyl)-4-oxo-3,4-dihydrothieno[3,4-d]pyridazine-1-carboxylate —— C22H15BrFN3O4S
Ethyl 5-(4-bromobenzamido)-3-(4-fluorophenyl)-4-oxo-3,4-dihydrothieno[3,4-d]pyridazine-1-carboxylate
—— ethyl 4-[4-[[(1S,2S)-2-methylcyclopropanecarbonyl]amino]benzoyl]oxypiperidine-1-carboxylate —— C20H26N2O5
ethyl 4-[4-[[(1S,2S)-2-methylcyclopropanecarbonyl]amino]benzoyl]oxypiperidine-1-carboxylate
—— Ethyl 4-[4-[(7-methyl-[1,3]thiazolo[5,4-e][1,3]benzothiazol-2-yl)carbamoyl]phenyl]sulfonylpiperazine-1-carboxylate —— C23H23N5O5S3
Ethyl 4-[4-[(7-methyl-[1,3]thiazolo[5,4-e][1,3]benzothiazol-2-yl)carbamoyl]phenyl]sulfonylpiperazine-1-carboxylate
—— Ethyl 2-cyano-3-(4-ethoxy-3-methoxyphenyl)prop-2-enoate —— C15H17NO4
Ethyl 2-cyano-3-(4-ethoxy-3-methoxyphenyl)prop-2-enoate
—— ethyl 2-[2-[2-[(3-methoxycarbonyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-2-oxoethyl]sulfanylacetyl]imino-3-(2-methoxy-2-oxoethyl)-1,3-benzothiazole-6-carboxylate —— C26H27N3O8S3
ethyl 2-[2-[2-[(3-methoxycarbonyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-2-oxoethyl]sulfanylacetyl]imino-3-(2-methoxy-2-oxoethyl)-1,3-benzothiazole-6-carboxylate
—— (E)-1-[4-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(2-ethoxyphenyl)prop-2-en-1-one —— C23H32N2O4
(E)-1-[4-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(2-ethoxyphenyl)prop-2-en-1-one
—— (E)-1-[4-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(4-methylphenyl)prop-2-en-1-one —— C22H30N2O3
(E)-1-[4-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(4-methylphenyl)prop-2-en-1-one
—— (E)-1-[4-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(2,4-dimethylphenyl)prop-2-en-1-one —— C23H32N2O3
(E)-1-[4-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(2,4-dimethylphenyl)prop-2-en-1-one
—— (E)-3-(2,3-dimethoxyphenyl)-1-[4-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]prop-2-en-1-one —— C23H32N2O5
(E)-3-(2,3-dimethoxyphenyl)-1-[4-[(2S,6S)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]prop-2-en-1-one
—— (E)-3-(2,3-dimethoxyphenyl)-1-[4-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]prop-2-en-1-one —— C23H32N2O5
(E)-3-(2,3-dimethoxyphenyl)-1-[4-[(2R,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]prop-2-en-1-one
—— ethyl 2-[[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfonyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C20H18FN3O6S2
ethyl 2-[[2-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]sulfonyl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl 5-(N-((4-methoxyphenyl)sulfonyl)butyramido)-2-methylbenzofuran-3-carboxylate —— C23H25NO7S
ethyl 5-(N-((4-methoxyphenyl)sulfonyl)butyramido)-2-methylbenzofuran-3-carboxylate
—— ethyl N-[(2R)-4-methyl-1-[[(E)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enoyl]amino]pentan-2-yl]carbamate —— C19H25N3O7
ethyl N-[(2R)-4-methyl-1-[[(E)-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enoyl]amino]pentan-2-yl]carbamate
—— ethyl N-[(2R)-1-[[(E)-3-[1-(2-cyanoethyl)indol-3-yl]prop-2-enoyl]amino]-4-methylpentan-2-yl]carbamate —— C23H30N4O3
ethyl N-[(2R)-1-[[(E)-3-[1-(2-cyanoethyl)indol-3-yl]prop-2-enoyl]amino]-4-methylpentan-2-yl]carbamate
—— ethyl N-[(2R)-1-[3-(1,4-dioxo-3H-phthalazin-2-yl)propanoylamino]-4-methylpentan-2-yl]carbamate —— C20H28N4O5
ethyl N-[(2R)-1-[3-(1,4-dioxo-3H-phthalazin-2-yl)propanoylamino]-4-methylpentan-2-yl]carbamate
—— ethyl N-[(2R)-1-[[2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetyl]amino]-4-methylpentan-2-yl]carbamate —— C22H32N4O3
ethyl N-[(2R)-1-[[2-(3,5-dimethyl-1-phenylpyrazol-4-yl)acetyl]amino]-4-methylpentan-2-yl]carbamate
—— ethyl N-[(2S)-1-[[5-(2,2-dimethylpropanoylamino)-3-methylthiophene-2-carbonyl]amino]-4-methylpentan-2-yl]carbamate —— C20H33N3O4S
ethyl N-[(2S)-1-[[5-(2,2-dimethylpropanoylamino)-3-methylthiophene-2-carbonyl]amino]-4-methylpentan-2-yl]carbamate
—— ethyl N-[(2R)-4-methyl-1-[3-[(4-methylphenyl)sulfonylamino]propanoylamino]pentan-2-yl]carbamate —— C19H31N3O5S
ethyl N-[(2R)-4-methyl-1-[3-[(4-methylphenyl)sulfonylamino]propanoylamino]pentan-2-yl]carbamate
—— ethyl N-[(2S)-1-[[4-(2,5-dioxopyrrolidin-1-yl)benzoyl]amino]-4-methylpentan-2-yl]carbamate —— C20H27N3O5
ethyl N-[(2S)-1-[[4-(2,5-dioxopyrrolidin-1-yl)benzoyl]amino]-4-methylpentan-2-yl]carbamate
—— (E)-1-[4-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(2-ethoxyphenyl)prop-2-en-1-one —— C23H32N2O4
(E)-1-[4-[(2S,6R)-2,6-dimethylmorpholine-4-carbonyl]piperidin-1-yl]-3-(2-ethoxyphenyl)prop-2-en-1-one
—— ethyl N-[(2R)-1-[[(E)-3-[4-(cyclopropylcarbamoyl)phenyl]prop-2-enoyl]amino]-4-methylpentan-2-yl]carbamate —— C22H31N3O4
ethyl N-[(2R)-1-[[(E)-3-[4-(cyclopropylcarbamoyl)phenyl]prop-2-enoyl]amino]-4-methylpentan-2-yl]carbamate
—— ethyl N-[6-ethyl-2-[(4-pyrrolidin-1-ylsulfonylbenzoyl)amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonyl]carbamate —— C24H30N4O6S2
ethyl N-[6-ethyl-2-[(4-pyrrolidin-1-ylsulfonylbenzoyl)amino]-5,7-dihydro-4H-thieno[2,3-c]pyridine-3-carbonyl]carbamate
—— Ethyl 4-[4-[[3-(dimethylcarbamoylcarbamoyl)-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridin-2-yl]carbamoyl]phenyl]sulfonylpiperazine-1-carboxylate —— C29H40N6O7S2
Ethyl 4-[4-[[3-(dimethylcarbamoylcarbamoyl)-5,5,7,7-tetramethyl-4,6-dihydrothieno[2,3-c]pyridin-2-yl]carbamoyl]phenyl]sulfonylpiperazine-1-carboxylate
—— ethyl N-[(2R)-1-[[5-(2,2-dimethylpropanoylamino)-3-methylthiophene-2-carbonyl]amino]-4-methylpentan-2-yl]carbamate —— C20H33N3O4S
ethyl N-[(2R)-1-[[5-(2,2-dimethylpropanoylamino)-3-methylthiophene-2-carbonyl]amino]-4-methylpentan-2-yl]carbamate