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—— (E)-3-(furan-2-yl)-N-[2-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-oxoethyl]prop-2-enamide —— C17H19N3O3
(E)-3-(furan-2-yl)-N-[2-[(1S)-1-methyl-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazin-2-yl]-2-oxoethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[2-(2-nitroanilino)ethylamino]-2-oxoethyl]prop-2-enamide —— C17H18N4O5
(E)-3-(furan-2-yl)-N-[2-[2-(2-nitroanilino)ethylamino]-2-oxoethyl]prop-2-enamide
—— ethyl 3-[3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propylcarbamoyl]-5-nitrobenzoate —— C19H27N3O6
ethyl 3-[3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propylcarbamoyl]-5-nitrobenzoate
—— (E)-N-[2-[[(1S)-1-[4-(difluoromethoxy)phenyl]ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C18H18F2N2O4
(E)-N-[2-[[(1S)-1-[4-(difluoromethoxy)phenyl]ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[4-(naphthalene-1-carbonyl)piperazin-1-yl]-2-oxoethyl]prop-2-enamide —— C24H23N3O4
(E)-3-(furan-2-yl)-N-[2-[4-(naphthalene-1-carbonyl)piperazin-1-yl]-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-[[(1R)-1-[4-(difluoromethoxy)phenyl]ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C18H18F2N2O4
(E)-N-[2-[[(1R)-1-[4-(difluoromethoxy)phenyl]ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]prop-2-enamide —— C21H22N4O4
(E)-3-(furan-2-yl)-N-[2-[[(R)-(2-methoxyphenyl)-(1-methylimidazol-2-yl)methyl]amino]-2-oxoethyl]prop-2-enamide
—— Ethyl 2-(cinnamoylamino)-4-(4-methoxyphenyl)-5-methyl-3-thiophenecarboxylate —— C24H23NO4S
Ethyl 2-(cinnamoylamino)-4-(4-methoxyphenyl)-5-methyl-3-thiophenecarboxylate
—— ethyl (3S)-1-[5-(2-chlorophenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxylate —— C18H19ClN2O4
ethyl (3S)-1-[5-(2-chlorophenyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxylate
—— (E)-N-[2-[[(S)-(4-chlorophenyl)-phenylmethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C22H19ClN2O3
(E)-N-[2-[[(S)-(4-chlorophenyl)-phenylmethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[[1-[2-(diethylamino)ethyl]benzimidazol-2-yl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C22H27N5O3
(E)-N-[2-[[1-[2-(diethylamino)ethyl]benzimidazol-2-yl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl (2Z,5S)-5-(4-fluorophenyl)-2-(furan-2-ylmethylidene)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C21H17FN2O4S
ethyl (2Z,5S)-5-(4-fluorophenyl)-2-(furan-2-ylmethylidene)-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-N-[2-[[5-(4-chlorophenyl)furan-2-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C20H17ClN2O4
(E)-N-[2-[[5-(4-chlorophenyl)furan-2-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl]prop-2-enamide —— C19H22N4O3
(E)-3-(furan-2-yl)-N-[2-oxo-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]ethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[2-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]ethylamino]-2-oxoethyl]prop-2-enamide —— C21H21N3O3S
(E)-3-(furan-2-yl)-N-[2-[2-[4-(2-methyl-1,3-thiazol-4-yl)phenyl]ethylamino]-2-oxoethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-(3-piperidin-1-ylsulfonylanilino)ethyl]prop-2-enamide —— C20H23N3O5S
(E)-3-(furan-2-yl)-N-[2-oxo-2-(3-piperidin-1-ylsulfonylanilino)ethyl]prop-2-enamide
—— (E)-N-[2-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C21H24N2O5
(E)-N-[2-[[(2R)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[3-(2-oxopyrrolidin-1-yl)anilino]ethyl]prop-2-enamide —— C19H19N3O4
(E)-3-(furan-2-yl)-N-[2-oxo-2-[3-(2-oxopyrrolidin-1-yl)anilino]ethyl]prop-2-enamide
—— ethyl (2Z,5R)-2-[(1,3-dimethyl-2-oxobenzimidazol-5-yl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H24N4O4S
ethyl (2Z,5R)-2-[(1,3-dimethyl-2-oxobenzimidazol-5-yl)methylidene]-7-methyl-3-oxo-5-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(furan-2-yl)-N-[2-[4-(4-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl]prop-2-enamide —— C22H24N2O5
(E)-3-(furan-2-yl)-N-[2-[4-(4-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl]prop-2-enamide
—— ethyl (6S)-6-(2-methylbutan-2-yl)-2-(thiophene-2-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C21H27NO3S2
ethyl (6S)-6-(2-methylbutan-2-yl)-2-(thiophene-2-carbonylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[2-[[(1S)-1-(4-bromophenyl)ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C17H17BrN2O3
(E)-N-[2-[[(1S)-1-(4-bromophenyl)ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[2-[(2S)-2-(4-ethoxyphenoxy)propanoyl]hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C20H23N3O6
(E)-N-[2-[2-[(2S)-2-(4-ethoxyphenoxy)propanoyl]hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl 3-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propylcarbamoyl]-5-nitrobenzoate —— C19H27N3O6
ethyl 3-[3-[(2S,6S)-2,6-dimethylmorpholin-4-yl]propylcarbamoyl]-5-nitrobenzoate
—— (E)-N-[2-[[(1R)-1-(1-adamantyl)ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C21H28N2O3
(E)-N-[2-[[(1R)-1-(1-adamantyl)ethyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl [(5E)-5-{3-bromo-4-[(2-fluorobenzyl)oxy]benzylidene}-2,4-dioxo-1,3-thiazolidin-3-yl]acetate —— C21H17BrFNO5S
ethyl [(5E)-5-{3-bromo-4-[(2-fluorobenzyl)oxy]benzylidene}-2,4-dioxo-1,3-thiazolidin-3-yl]acetate
—— (E)-3-(furan-2-yl)-N-[2-[[(2S)-2-(4-methoxyphenyl)-2-piperidin-1-ylethyl]amino]-2-oxoethyl]prop-2-enamide —— C23H29N3O4
(E)-3-(furan-2-yl)-N-[2-[[(2S)-2-(4-methoxyphenyl)-2-piperidin-1-ylethyl]amino]-2-oxoethyl]prop-2-enamide
—— ethyl (5Z)-5-[(1-cyclopropyl-2,5-dimethylpyrrol-3-yl)methylidene]-2-(4-methoxyanilino)-4-oxothiophene-3-carboxylate —— C24H26N2O4S
ethyl (5Z)-5-[(1-cyclopropyl-2,5-dimethylpyrrol-3-yl)methylidene]-2-(4-methoxyanilino)-4-oxothiophene-3-carboxylate
—— (E)-3-(furan-2-yl)-N-[2-[2-(3-methoxy-4-propoxybenzoyl)hydrazinyl]-2-oxoethyl]prop-2-enamide —— C20H23N3O6
(E)-3-(furan-2-yl)-N-[2-[2-(3-methoxy-4-propoxybenzoyl)hydrazinyl]-2-oxoethyl]prop-2-enamide
—— (E)-N-[2-[[5-(1,3-benzothiazol-2-yl)furan-2-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C21H17N3O4S
(E)-N-[2-[[5-(1,3-benzothiazol-2-yl)furan-2-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[[(1S)-1-(4-bromophenyl)propyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C18H19BrN2O3
(E)-N-[2-[[(1S)-1-(4-bromophenyl)propyl]amino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[2-[(4-methylphenyl)methylsulfanyl]ethylamino]-2-oxoethyl]prop-2-enamide —— C19H22N2O3S
(E)-3-(furan-2-yl)-N-[2-[2-[(4-methylphenyl)methylsulfanyl]ethylamino]-2-oxoethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]-2-oxoethyl]prop-2-enamide —— C20H23N3O5S
(E)-3-(furan-2-yl)-N-[2-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]-2-oxoethyl]prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl]prop-2-enamide —— C16H13F3N2O4
(E)-3-(furan-2-yl)-N-[2-oxo-2-[4-(trifluoromethoxy)anilino]ethyl]prop-2-enamide
—— (E)-N-[2-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C21H24N2O5
(E)-N-[2-[[(2S)-5-ethoxy-2-methyl-2,3-dihydro-1-benzofuran-6-yl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[2-(4-chlorophenyl)sulfanylethylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C17H17ClN2O3S
(E)-N-[2-[2-(4-chlorophenyl)sulfanylethylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-2-[(4-fluorophenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H23FN2O5S
ethyl (2E,5S)-5-(3,4-dimethoxyphenyl)-2-[(4-fluorophenyl)methylidene]-7-methyl-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[4-[(2S)-oxolane-2-carbonyl]piperazin-1-yl]ethyl]prop-2-enamide —— C18H23N3O5
(E)-3-(furan-2-yl)-N-[2-oxo-2-[4-[(2S)-oxolane-2-carbonyl]piperazin-1-yl]ethyl]prop-2-enamide
—— (E)-N-[2-[2-(3,4-diethoxyphenyl)ethylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C21H26N2O5
(E)-N-[2-[2-(3,4-diethoxyphenyl)ethylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[3-oxo-3-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]propyl]prop-2-enamide —— C16H20F3N3O3
(E)-3-(furan-2-yl)-N-[3-oxo-3-[4-(2,2,2-trifluoroethyl)piperazin-1-yl]propyl]prop-2-enamide
—— ethyl 3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propylcarbamoyl]-5-nitrobenzoate —— C19H27N3O6
ethyl 3-[3-[(2R,6R)-2,6-dimethylmorpholin-4-yl]propylcarbamoyl]-5-nitrobenzoate
—— (E)-N-[2-[2-[2-(4-chlorophenyl)acetyl]hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C17H16ClN3O4
(E)-N-[2-[2-[2-(4-chlorophenyl)acetyl]hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl 4-[(E)-[2-oxo-5-phenyl-1-(4-propan-2-ylphenyl)pyrrol-3-ylidene]methyl]benzoate —— C29H27NO3
ethyl 4-[(E)-[2-oxo-5-phenyl-1-(4-propan-2-ylphenyl)pyrrol-3-ylidene]methyl]benzoate
—— (E)-N-[2-[[4-(difluoromethoxy)phenyl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C17H16F2N2O4
(E)-N-[2-[[4-(difluoromethoxy)phenyl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[2-[(2R)-2-(4-ethoxyphenoxy)propanoyl]hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C20H23N3O6
(E)-N-[2-[2-[(2R)-2-(4-ethoxyphenoxy)propanoyl]hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[2-(3,4-dimethoxybenzoyl)hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C18H19N3O6
(E)-N-[2-[2-(3,4-dimethoxybenzoyl)hydrazinyl]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-N-[2-[[4-(difluoromethoxy)-3-methoxyphenyl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide —— C18H18F2N2O5
(E)-N-[2-[[4-(difluoromethoxy)-3-methoxyphenyl]methylamino]-2-oxoethyl]-3-(furan-2-yl)prop-2-enamide
—— ethyl (2Z,5S)-5-(4-acetyloxyphenyl)-7-methyl-2-(1-methyl-2-oxoindol-3-ylidene)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H23N3O6S
ethyl (2Z,5S)-5-(4-acetyloxyphenyl)-7-methyl-2-(1-methyl-2-oxoindol-3-ylidene)-3-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[4-[2-oxo-2-(propan-2-ylamino)ethyl]piperazin-1-yl]ethyl]prop-2-enamide —— C18H26N4O4
(E)-3-(furan-2-yl)-N-[2-oxo-2-[4-[2-oxo-2-(propan-2-ylamino)ethyl]piperazin-1-yl]ethyl]prop-2-enamide
—— Ethyl (4Z)-4-{[4-(methoxycarbonyl)phenyl]methylidene}-1-(2-methoxyethyl)-2-methyl-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate —— C20H23NO6
Ethyl (4Z)-4-{[4-(methoxycarbonyl)phenyl]methylidene}-1-(2-methoxyethyl)-2-methyl-5-oxo-4,5-dihydro-1H-pyrrole-3-carboxylate